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Cat. No. Product Name Target Signaling Pathways
T1636 Paroxetine hydrochloride

Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀

5-HT Receptor; Serotonin Transporter; GRK; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Paroxetine hydrochloride (Paroxetine HCl) 是一种血清素摄取抑制剂,能抑制 GRK2 活性,IC50值为 14 μM。它可研究抑郁症。
T1636L Paroxetine hydrochloride hemihydrate

Paroxetine Hydrochloride,Paxil,Paroxetine HCl,Seroxat

5-HT Receptor GPCR/G Protein; Neuroscience
Paroxetine hydrochloride hemihydrate (Paxil) 是一种抗抑郁药,为高效的五羟色胺再摄取抑制剂,能抑制 GRK2 活性,IC50 为 14 μM。
T37308 Desmethylene Paroxetine hydrochloride

Drug Metabolite Metabolism
Desmethylene Paroxetine hydrochlorideParoxetine 的非共轭代谢产物,是一种儿茶酚中间体。
T35875 CCG258208 hydrochloride

GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).GRKs-IN-1 hydrochloride is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine[1]. [1]. Waldschmidt HV, et al. Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2Inhibitors Based on Paroxetine. J Med Chem. 2017 Apr 13;60(7):305...

化合物

Paroxetine hydrochloride
Cat.No: T1636
Synonym: Paroxetine HCl,BRL29060 hydrochloride,FG-7051,BRL29060A,盐酸帕罗西汀
Target: 5-HT Receptor, Serotonin Transporter, GRK, AChR, Autophagy
Paroxetine hydrochloride hemihydrate
Cat.No: T1636L
Synonym: Paroxetine Hydrochloride,Paxil,Paroxetine HCl,Seroxat
Target: 5-HT Receptor
Desmethylene Paroxetine hydrochloride
Cat.No: T37308
Synonym:
Target: Drug Metabolite
CCG258208 hydrochloride
Cat.No: T35875
Synonym:
Target:
TargetMol Loading
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