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Cat. No. Product Name Target Signaling Pathways
T74830 PDK-IN-1

PDK-IN-1(compound 7o)是一种针对丙酮酸脱氢酶激酶(PDK)的抑制剂,其对PDK1和HSP90的IC50值分别为0.03和0.1μM。通过靶向PDH/PDK轴,PDK-IN-1能有效降低肿瘤质量。
T12412L PDK4-IN-1 hydrochloride

Apoptosis; PDK Apoptosis; PI3K/Akt/mTOR signaling
PDK4-IN-1 hydrochloride 是一种蒽醌衍生物,对丙酮酸脱氢酶激酶 4有抑制作用,IC50为 84 nM,具有口服活性。它抑制细胞转化和细胞增殖并诱导细胞凋亡。它具有抗过敏,抗糖尿病和抗癌作用。
T12412 PDK4-IN-1

Others Others
PDK4-IN-1 is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4)(IC50 value of 84 nM).
T16450 PDK1-IN-RS2

PDK PI3K/Akt/mTOR signaling
PDK1-IN-RS2 inhibits the activation of the downstream kinases S6K1 by PDK1. PDK1-IN-RS2 is a mimic of the peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor (Kd: 9 μM).
T17224 VER-246608

Dehydrogenase; PDK Metabolism; PI3K/Akt/mTOR signaling
VER-246608 是ATP 竞争性的丙酮酸脱氢酶激酶抑制剂,对PDK-1PDK-3,PDK-2,和PDK-4的IC50分别为 35 nM,40 nM,84 nM 和 91 nM。
T79723 PDK-IN-2

PDK-IN-2(Compound 1F)是一种具有IC50为68 nM的PDK抑制剂。该化合物能够抑制PDK1PDK4在细胞内的表达,增强线粒体生物能并降低糖酵解表型,同时诱导细胞走向线粒体途径的apoptosis。此外,PDK-IN-2在4T1同基因小鼠模型中能够有效抑制肿瘤生长。

化合物

PDK-IN-1
Cat.No: T74830
Synonym:
Target:
PDK4-IN-1 hydrochloride
Cat.No: T12412L
Synonym:
Target: Apoptosis, PDK
PDK4-IN-1
Cat.No: T12412
Synonym:
Target: Others
PDK1-IN-RS2
Cat.No: T16450
Synonym:
Target: PDK
VER-246608
Cat.No: T17224
Synonym:
Target: Dehydrogenase, PDK
PDK-IN-2
Cat.No: T79723
Synonym:
Target:
TargetMol Loading
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