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Search Results for " p-300 "

13

抑制剂 & 化合物

1

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T69691	Pocenbrodib FT-7051,P-300	Epigenetic Reader Domain	Chromatin/Epigenetic
	Pocenbrodib (FT-7051) 是一种有效的 CBP/p300 家族的溴结构域抑制剂，具有潜在的抗肿瘤活性，可口用于研究癌症。
T12345	CBP/p300-IN-3 P300/CBP-IN-3	Histone Acetyltransferase	Chromatin/Epigenetic
	CBP/p300-IN-3 (P300/CBP-IN-3) 是一种组蛋白乙酰转移酶抑制剂。
T40144	CBP/p300 ligand 2
	CBP/p300 ligand 2 is a selective ligand that binds to the target protein for PROTAC of dCBP-1, a potent and selective heterobifunctional degrader of p300/CBP.
T12346	CBP/p300-IN-5 P300/CBP-IN-5	Epigenetic Reader Domain	Chromatin/Epigenetic
	P300/CBP-IN-5 is a potent inhibitor of p300/CBP histone acetyltransferase (IC50 of 18.8 nM).
T40344	CBP/p300-IN-14 CBP/p300-IN-14
	CBP/p300-IN-14, efficiently inhibits CBP/EP300 (lysine acetyltransferase) with an IC50 value of 3.3 nM.
T39826	CBP/p300-IN-8 CBP/p300-IN-8
	CBP/p300-IN-8 is a potent inhibitor of the CBP/P300 family of bromodomains . CBP/p300-IN-8 inhibits CBP ( IC 50 =0.01-0.1 μΜ) and BRD4 ( IC 50 =1-1000 μΜ) activity.
T10702	CBP/p300-IN-2 CBP/EP300-IN-2	Epigenetic Reader Domain; c-Myc	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc).
T40143	PROTAC CBP/P300 Degrader-1 PROTAC CBP/P300 Degrader-1
	PROTAC CBP/P300 Degrader-1 is an effective compound that degrades CBP/P300 in a potent manner. It significantly reduces cell viability in various cancer cell lines.
T40142	Thalidomide-NH-CBP/p300 ligand 2 Thalidomide-NH-CBP/p300 ligand 2
	Thalidomide-NH-CBP/p300 ligand 2 (P-007) is a PROTAC-based compound designed to degrade CBP and p300, acting as a functional antagonist (WO2020173440).
T14042	4-P-PDOT 4-phenyl-2- propionamidotetralin	Melatonin Receptor; MT Receptor	GPCR/G Protein; Neuroscience
	4-P-PDOT (4-phenyl-2- propionamidotetralin) 是一种选择性和亲和性的褪黑激素受体拮抗剂，可显著抵消褪黑激素介导的抗氧化作用。它对MT2的选择性是 MT1 的 300 倍以上。
T27389	Frequentin
	Frequentin, an antibiotic originally isolated from P. frequentans, is active against bacteria (MICs = 200 and 300 µg/ml for B. subtilis and S. aureus, respectively) and fungi.
T38347	Zelkovamycin
	Zelkovamycin is a cyclic peptide antibiotic originally isolated from Streptomyces.1 It inhibits growth of X. oryzae, P. oryzae, S. aureus, and A. laidlawii in a concentration-dependent manner when used at concentrations ranging from 0.01 to 300 μg/ml.References1. Zhang, H., Tomoda, H., Tabata, N., et al. Zelkovamycin, a new cyclic peptide antibiotic from Streptomyces sp. K96-0670. I. Production, isolation and biological properties. J. Antibiot. (Tokyo) 52(1), 29-33 (1999). Zelkovamycin is a cycl...
T78135	Nicotelline Nicotellin
	Nicotelline（Nicotellin）是一种与尼古丁相关的生物碱，作为人类cDNA表达的细胞色素P-450 2A6（CYP2A6）的弱抑制剂，不显著抑制该酶介导的香豆素7-羟基化反应，在300 μM浓度下效果更是如此。此外，Nicotelline还被用作烟草烟雾中颗粒物（PM）的示踪剂和生物标记物。

化合物

Cat.No: T69691

Synonym: FT-7051,P-300

Target: Epigenetic Reader Domain

Cat.No: T12345

Synonym: P300/CBP-IN-3

Target: Histone Acetyltransferase

CBP/p300 ligand 2

Cat.No: T40144

Cat.No: T12346

Synonym: P300/CBP-IN-5

Target: Epigenetic Reader Domain

Cat.No: T40344

Synonym: CBP/p300-IN-14

Cat.No: T39826

Synonym: CBP/p300-IN-8

Cat.No: T10702

Synonym: CBP/EP300-IN-2

Target: Epigenetic Reader Domain, c-Myc

PROTAC CBP/P300 Degrader-1

Cat.No: T40143

Synonym: PROTAC CBP/P300 Degrader-1

Thalidomide-NH-CBP/p300 ligand 2

Cat.No: T40142

Synonym: Thalidomide-NH-CBP/p300 ligand 2

Cat.No: T14042

Synonym: 4-phenyl-2- propionamidotetralin

Target: Melatonin Receptor, MT Receptor

Cat.No: T27389

Cat.No: T38347

Cat.No: T78135

Synonym: Nicotellin

Cat. No.	Product Name	Target	Signaling Pathways
T2911	Stevioside 甜菊苷,蛇菊苷	TLR	Immunology/Inflammation
	Stevioside 是一种天然甜味剂，从甜叶菊叶中提取的获得，具有抗癌作用。

天然产物

Cat.No: T2911

Synonym: 甜菊苷,蛇菊苷

Target: TLR

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