首页 工具
登录
购物车

搜索结果

Search Results for " myelofibrosis "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T9705 TL-895

BTK Angiogenesis; Tyrosine Kinase/Adaptors
TL-895 是口服有效的,ATP 竞争性的,以及高度选择性和不可逆的BTK 抑制剂,IC50和Ki 分别为 1.5 nM 和 11.9 nM。TL-895在 JAKi 复发/难治性骨髓纤维化、急性髓系白血病、COVID-19 和癌症方面有研究的价值。
T3069 AZD-1480

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
AZD1480 是 ATP 竞争型JAK1和JAK2抑制剂,IC50分别为 1.3 和 0.4 nM。
T2709 TAK-901

TAK901

JAK; CDK; Src; Aurora Kinase Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
TAK-901是一种多靶点的极光激酶抑制剂,对极光激酶 A 和 B 的 IC50值分别为 21 和 15 nM。它用于研究淋巴瘤、骨髓纤维化、多发性骨髓瘤、骨髓化生和晚期实体瘤等治疗的试验。
T70823 Momelotinib HCl

Momelotinib HCl is a JAK1/2 inhibitor, reducing anemia in myelofibrosis (MF) patients.
T11687 Itacitinib adipate

Phosphatase Metabolism
Itacitinib adipate is an orally bioavailable and selective JAK1 inhibitor,Itacitinib adipate has been tested for efficacy and safety in a phase II trial in myelofibrosis.
T64283 Pacritinib hydrochloride

Pacritinib hydrochloride 是一种野生型 JAK2 (IC50: 23 nM) 和 JAK2V617F 突变型 (IC50: 19 nM) 的有效抑制剂。Pacritinib hydrochloride 也能够抑制 FLT3 (IC50: 22 nM) 及其突变型 FLT3D835Y (IC50: 6 nM)。Pacritinib hydrochloride 能够用于研究急性髓系白血病(AML)和骨髓纤维化(MF)。
T70008 Bomedemstat ditosylate

Bomedemstat, also known as IMG-7289, is a lysine-specific histone demethylase 1 (LSD1) inhibitor with antineoplastic activity. Bomedemstat may be useful in the treatment of acute myeloid leukaemia, myelodysplastic syndrome, and Myelofibrosis. IMG-7289 selectively inhibited proliferation and induced apoptosis of JAK2 V617F cells by concomitantly increasing expression and methylation of p53, and, independently, the pro-apoptotic factor PUMA and by decreasing the levels of its antiapoptotic antago...
T9634 Bomedemstat

Bomedemstat (IMG-7289) 是一种有效的,具有口服活性的且不可逆的赖氨酸特异性脱甲基酶 1 (LSD1) 抑制剂,具有表观遗传活性。Bomedemstat 具有抗癌活性,可用于急性髓性白血病 (AML) 和骨髓纤维化 (MF) 的研究。

化合物

TL-895
Cat.No: T9705
Synonym:
Target: BTK
AZD-1480
Cat.No: T3069
Synonym:
Target: JAK
TAK-901
Cat.No: T2709
Synonym: TAK901
Target: JAK, CDK, Src, Aurora Kinase
Momelotinib HCl
Cat.No: T70823
Synonym:
Target:
Itacitinib adipate
Cat.No: T11687
Synonym:
Target: Phosphatase
Pacritinib hydrochloride
Cat.No: T64283
Synonym:
Target:
Bomedemstat ditosylate
Cat.No: T70008
Synonym:
Target:
Bomedemstat
Cat.No: T9634
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼