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Cat. No. Product Name Target Signaling Pathways
T11964 MCH-1 antagonist 1

P450 Metabolism
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
T11966 MCHR1 antagonist 2

HER; Melanin-concentrating Hormone Receptor (MCHR) Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors
MCHR1 antagonist 2 是有效的黑色素聚集激素受体 1 拮抗剂,IC50为 65 nM。它也抑制hERG,在IMR-32 细胞中的IC50为 4.0 nM。
T22591 ATC 0175 hydrochloride

GPR; 5-HT Receptor; Melanin-concentrating Hormone Receptor (MCHR) Endocrinology/Hormones; GPCR/G Protein; Neuroscience
ATC 0175 hydrochloride 是一种具有口服活性的黑色素细胞浓缩激素1受体拮抗剂,具有强效性和选择性,ATC 0175 hydrochloride 对MCH1R、MCH2R、MCH1、5-HT2B 受体和5-HT1A 受体 具有亲和力 ,IC50分别为为13.5nM、>10,000 nM、13 nM、9.66 nM 和16.9 nM。ATC 0175 hydrochloride 在动物模型中表现出抗抑郁和抗焦虑作用。ATC0175可用于研究抑郁症和/或焦虑症。
T10173 MCHR1 antagonist 1

Others Others
MCHR1 antagonist 1 is a selective antagonist of melanin-concentrating hormone-1 (MCH1) receptor (Kb: 1 nM, Ki: 4 nM at human MCH1).
T26703 AZ13483342

AZ-13483342,AZ 13483342

AZ13483342 is an antagonist of the melanin concentrating hormone receptor 1 (MCH1) with a potential diabetes therapeutic activity.
T5406 SNAP 94847

SNAP-94847

GPR; Melanin-concentrating Hormone Receptor (MCHR) Endocrinology/Hormones; GPCR/G Protein
SNAP 94847 (SNAP-94847) 是一种选择性黑色素浓缩激素受体1 拮抗剂,Ki 为 2.2 nM。它具有抗焦虑和抗抑郁活性,可减少小鼠的食物摄入。
T7749 ALB-127158

ALB-127158(a) 是一种有效的选择性黑色素浓缩激素 1 (MCH1) 受体拮抗剂,可能是炎症性肠病 (IBD) 的潜在治疗方法

化合物

MCH-1 antagonist 1
Cat.No: T11964
Synonym:
Target: P450
MCHR1 antagonist 2
Cat.No: T11966
Synonym:
Target: HER, Melanin-concentrating Hormone Receptor (MCHR)
ATC 0175 hydrochloride
Cat.No: T22591
Synonym:
Target: GPR, 5-HT Receptor, Melanin-concentrating Hormone Receptor (MCHR)
MCHR1 antagonist 1
Cat.No: T10173
Synonym:
Target: Others
AZ13483342
Cat.No: T26703
Synonym: AZ-13483342,AZ 13483342
Target:
SNAP 94847
Cat.No: T5406
Synonym: SNAP-94847
Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)
ALB-127158
Cat.No: T7749
Synonym:
Target:
TargetMol Loading
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