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抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T65008 L-Adenosine

L-Adenosine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65008,CAS号为 3080-29-3。
T26266 TH-162

L-PIA,(R)​-PIA,(R)​- PIA,(R)​-​PIA,L-2-N6-(Phenylisopropyl)adenosine

TH-162, also known as (R)​-​PIA and Adenosine, N-(1-methyl-2-phenylethyl)-, (R)-, is an agonist of the A1 adenosine receptor. Affinity for adenosine receptors is approx. 100× that of the (+)-isomer.
TNU0351 3’-Azido-3’-deoxy-beta-L-adenosine

3'-Azido-3'-deoxy-beta-L-adenosine is a Nucleoside Derivative - L-nucleoside, Azido-nucleoside.
T28881 Sulmazole

Vardax,AR-L 115BS,AR-L 115-BS

PDE; Parasite; Adenosine Receptor GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Sulmazole (AR-L 115-BS) 是一种小分子 cGMP-PDE抑制剂。Sulmazole 对 A1 腺苷受体具有竞争性抑制作用,可改善心脏指数,低肺毛细血管楔压,可用于研究心脏衰竭。
T6360 3-deazaneplanocin A HCl

Others; Histone Methyltransferase Chromatin/Epigenetic; Others
3-deazaneplanocin A HCl 是组蛋白甲基转移酶 (EZH2) 和 S-腺苷同型半胱氨酸水解酶 (AHCY) 抑制剂。
T24384 L-97-1

L97-1,L 97-1

L-97-1 is an antagonist of the adenosine A1 receptor.
T74651 L-Inosine

L-Inosine 是 L-构型形式的 Inosine。Inosine 是一种由腺苷分解代谢产生的内源性嘌呤核苷。Inosine 具有抗炎免疫调节,抗伤害和神经保护作用。
T74764 Adenosylhomocysteinase

Adenosylhomocysteinase (SAHH; AHCY) 是一种高度保守的酶。Adenosylhomocysteinase 可逆催化 S-腺苷同型半胱氨酸 (SAH) 生成腺苷和 L-同型半胱氨酸。血清外泌体 Adenosylhomocysteinase 水平可作为 HBV-LC 患者预后的生物标志物。
T69975 Istaroxime oxalate

Istaroxime, also known as PST-2744, is a positive inotropic agent that mediates its action through inhibition of sodium/potassium adenosine triphosphatase (Na+/K+ ATPase). Na+/K+ ATPase inhibition increases intracellular sodium levels, which reverses the driving force of the sodium/calcium exchanger, inhibiting calcium extrusion and possibly facilitating calcium entry. Additionally, Istaroxime increases intracellular calcium by improving the efficacy by which intracellular calcium triggers sarco...

化合物

L-Adenosine
Cat.No: T65008
Synonym:
Target:
TH-162
Cat.No: T26266
Synonym: L-PIA,(R)​-PIA,(R)​- PIA,(R)​-​PIA,L-2-N6-(Phenylisopropyl)adenosine
Target:
3’-Azido-3’-deoxy-beta-L-adenosine
Cat.No: TNU0351
Synonym:
Target:
Sulmazole
Cat.No: T28881
Synonym: Vardax,AR-L 115BS,AR-L 115-BS
Target: PDE, Parasite, Adenosine Receptor
3-deazaneplanocin A HCl
Cat.No: T6360
Synonym:
Target: Others, Histone Methyltransferase
L-97-1
Cat.No: T24384
Synonym: L97-1,L 97-1
Target:
L-Inosine
Cat.No: T74651
Synonym:
Target:
Adenosylhomocysteinase
Cat.No: T74764
Synonym:
Target:
Istaroxime oxalate
Cat.No: T69975
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4901 5'-Guanylic acid disodium salt

Guanosine 5'-monophosphate disodium salt,5'-鸟苷酸二钠,鸟苷钠5'-单磷酸,GMP-5

Others; Endogenous Metabolite Metabolism; Others
5'-Guanylic acid disodium salt (GMP-5) 由鸟嘌呤,核糖和磷酸组成,是信使 RNA 中的一种核苷酸单体。 鸟苷衍生物参与细胞内信号转导,并已鉴定存在于端粒,核糖体 DNA,免疫球蛋白重链转换区和原癌基因的控制区中的重复基因组序列中。
TN5193 Tubotaiwine

AChR Neuroscience
Tubotaiwine shows selective activity against L. infantum. Tubotaiwine and apparicine have affinity for adenosine receptors in the micromolar range and also have in-vivo analgesic activity in mice.

天然产物

5'-Guanylic acid disodium salt
Cat.No: T4901
Synonym: Guanosine 5'-monophosphate disodium salt,5'-鸟苷酸二钠,鸟苷钠5'-单磷酸,GMP-5
Target: Others, Endogenous Metabolite
Tubotaiwine
Cat.No: TN5193
Synonym:
Target: AChR
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