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Cat. No. Product Name Target Signaling Pathways
T13237L Ropsacitinib

Tyk2-IN-8,PF-06826647

Tyrosine Kinases Tyrosine Kinase/Adaptors
Ropsacitinib (PF-06826647) 是一种选择性TYK2抑制剂。Ropsacitinib 与Tyk2催化活性JH1结构域结合(IC50:17nM)。
T39858 NVP-BSK805 trihydrochloride

NVP-BSK805 trihydrochloride

NVP-BSK805 trihydrochloride is a potent ATP-competitive inhibitor of JAK2, exhibiting IC50 values of 0.48 nM, 31.63 nM, 18.68 nM, and 10.76 nM against JAK2 JH1, JAK1 JH1, JAK3 JH1, and TYK2 JH1, respectively.
T5049 NVP-BSK805

NVP-BSK805 2HCl,8-[3,5-二氟-4-(4-吗啉基甲基)苯基]-2-[1-(4-哌啶基)-1H-吡唑-4-基]喹喔啉,BSK 805

Tyrosine Kinases; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
NVP-BSK805 (BSK 805) 是 ATP 竞争性的 JAK2抑制剂,对 JAK1 JH1、 JAK2 JH1 (JAK 同源 1)、JAK3 JH1和 TYK2 JH1 的 IC50值分别为 31.63、0.48、8.68 和 10.76 nM。
T14687 Deucravacitinib

BMS-986165

Tyrosine Kinases; JAK; IFNAR; Interleukin Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Deucravacitinib (BMS-986165) 是一种高选择性、口服生物可利用的变构 TYK2 抑制剂,用于治疗自身免疫性疾病。它通过稳定调节 JH2 结构域来阻断受体介导的 Tyk2 激活,可抑制IL-12/23和 I 型IFN 途径。它选择性结合 TYK2 假激酶 (JH2) 结构域,IC50为1.0 nM。
T13235 Tyk2-IN-7

Others Others
Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).
T13232 TyK2-IN-2

PDE Metabolism
TyK2-IN-2 is a selective inhibitor of TYK2 (IC50s: 7 nM, 0.1 μM, and 0.05 μM for TYK2 JH2, IL-23, and IFNα).
T13234 Tyk2-IN-5

Others Others
Tyk2-IN-5 is a selective and orally active inhibitor of Tyk2 JH2 (Ki: 0.086 nM for Tyk2 JH2; IC50: 25 nM for IFNα).

化合物

Ropsacitinib
Cat.No: T13237L
Synonym: Tyk2-IN-8,PF-06826647
Target: Tyrosine Kinases
NVP-BSK805 trihydrochloride
Cat.No: T39858
Synonym: NVP-BSK805 trihydrochloride
Target:
NVP-BSK805
Cat.No: T5049
Synonym: NVP-BSK805 2HCl,8-[3,5-二氟-4-(4-吗啉基甲基)苯基]-2-[1-(4-哌啶基)-1H-吡唑-4-基]喹喔啉,BSK 805
Target: Tyrosine Kinases, JAK
Deucravacitinib
Cat.No: T14687
Synonym: BMS-986165
Target: Tyrosine Kinases, JAK, IFNAR, Interleukin
Tyk2-IN-7
Cat.No: T13235
Synonym:
Target: Others
TyK2-IN-2
Cat.No: T13232
Synonym:
Target: PDE
Tyk2-IN-5
Cat.No: T13234
Synonym:
Target: Others
TargetMol Loading
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