Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24449 |
Mepacrine
Haffkinine,Erion |
Others | Others |
Mepacrine (Erion) 是一种吖啶衍生物,以前广泛用作抗疟药。它在细胞生物学实验中用作磷脂酶A2的抑制剂。 | |||
T0942 |
Quinacrine dihydrochloride
疟疾平,Mepacrine dihydrochloride,阿的平,SN-390,Quinacrine 2HCl |
Apoptosis; Mitophagy; DNA; Phospholipase; Parasite; Autophagy; Histamine Receptor | Apoptosis; Autophagy; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience |
Quinacrine dihydrochloride (Mepacrine dihydrochloride) 是一种具有口服活性的抗疟剂,抑制 NF-κB 并激活 p53 信号转导,诱导肿瘤细胞发生凋亡,具有抗肿瘤和抗寄生虫活性。 |