Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24152 |
HTH-01-091
HTH-01091,HTH01-091,HTH 01-091,HTH 01091 |
Serine/threonin kinase; Pim; MELK; DYRK; CDK; RIP kinase | Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; JAK/STAT signaling; Metabolism; NF-κB; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
HTH-01-091 是一种强效且选择性的 maternal embryonic leucine zipper kinase (MELK) 抑制剂(IC50 :10.5 nM)。HTH-01-091 对PIM1/2/3、RIPK2、DYRK3、smMLCK 和 CLK2有抑制作用。HTH-01-091 可用于研究乳腺癌。 | |||
T73867 | HTH-01-091 TFA | ||
HTH-01-091 TFA 是一种强效且选择性的maternal embryonic leucine zipper kinase (MELK)抑制剂,其IC50为 10.5 nM。HTH-01-091 TFA 还能抑制PIM1/2/3、RIPK2、DYRK3、smMLCK 和CLK2。HTH-01-091 TFA 可用于乳腺癌研究。 |