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Search Results for " hif-1alpha inhibitor "

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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T36711 FM19G11

FM19G11,HIF-1alpha/2alpha Inhibitor

HIF Angiogenesis; Chromatin/Epigenetic
FM19G11 是一种低氧诱导因子 (HIF) α-亚基抑制剂(在低氧诱导的荧光素酶试验中 IC50 为 80 nM)。
T3494 LW6

HIF-1α inhibitor,CAY10585,LW8

Apoptosis; Dehydrogenase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Apoptosis; Chromatin/Epigenetic; Metabolism
LW6 (HIF-1α inhibitor) 是一种新型 HIF-1抑制剂,IC50值为 4.4 μM。它降低 HIF-1α蛋白表达,但不影响 HIF-1β 表达。
T4381 Lificiguat

利非西呱,YC-1

Others; Guanylate cyclase; HIF Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein; Others
Lificiguat (YC-1) 是一种不依赖一氧化氮的可溶性鸟苷酸环化酶激活剂和低氧诱导因子 1α 的抑制剂。
T70903 KRH102053

KRH102053 is a HIF-1alpha inhibitor. KRH102053 decreased the protein level of HIF-1alpha and the mRNA levels of HIF-regulated downstream target genes, such as vascular endothelial growth factor, aldolase A, enolase 1 and monocarboxylate transporter 4. Consistent with these results, KRH102053 also inhibited the rates of HIF-related migration and invasion of HOS cells as well as the degree of tube formation in human umbilical vein endothelium cells.

化合物

FM19G11
Cat.No: T36711
Synonym: FM19G11,HIF-1alpha/2alpha Inhibitor
Target: HIF
LW6
Cat.No: T3494
Synonym: HIF-1α inhibitor,CAY10585,LW8
Target: Apoptosis, Dehydrogenase, HIF/HIF Prolyl-Hydroxylase, HIF
Lificiguat
Cat.No: T4381
Synonym: 利非西呱,YC-1
Target: Others, Guanylate cyclase, HIF
KRH102053
Cat.No: T70903
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T21494 Oligomycin

HIF Angiogenesis; Chromatin/Epigenetic
Oligomycin 是一种抗真菌抗生素,是 H+-ATP 合成酶的抑制剂。Oligomycin 能够阻断氧化磷酸化和电子传递链。Oligomycin 对缺氧性肿瘤细胞 HIF-1alpha 表达具有抑制作用。

天然产物

Oligomycin
Cat.No: T21494
Synonym:
Target: HIF
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