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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T80393 Gramicidin S

Gramicidin soviet

Antibiotic Microbiology/Virology
Gramicidin S(Gramicidin Soviet)是一种阳离子环肽类抗生素,能破坏革兰氏阴性及革兰氏阳性细菌膜的完整性,并抑制细胞色素bd醌醇氧化酶。
T80388 Gramicidin B

Antibiotic Microbiology/Virology
Gramicidin B是一种由15个氨基酸组成的直链多肽,属于非核糖体肽类抗生素。
T74537 Antifungal agent 26

Antifungal agent 26, a derivative of gramicidin A, exhibits antifungal, antiviral, and antiparasitic activities through binding with polysaccharides containing D-mannose (Man) in pathogens.

化合物

Gramicidin S
Cat.No: T80393
Synonym: Gramicidin soviet
Target: Antibiotic
Gramicidin B
Cat.No: T80388
Synonym:
Target: Antibiotic
Antifungal agent 26
Cat.No: T74537
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1130 Gramicidin

短杆菌肽,Gramicidinum,Gramicidine,Gramicidina

MRP; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Gramicidin (Gramicidine) 是一种抗菌肽。它通过组装成膜中的通道,增加其对阳离子的渗透性。
T41042 Gramicidin C

Gramicidin C, a naturally occurring polypeptide antibiotic, is isolated from B. brevis var. G.B.
T36439 Gramicidin A

Antibacterial; HIF; Parasite Angiogenesis; Chromatin/Epigenetic; Microbiology/Virology
Gramicidin A 是一种从从 B. brevis 分离出来的多肽类抗生素。Gramicidin A 是一种高度疏水的通道形成离子载体,在人工膜中形成一价阳离子可渗透的通道。Gramicidin A 诱导缺氧诱导因子 1α (HIF-1α) 的降解,并能降低人肾细胞癌小鼠异种移植模型的生长。Gramicidin A 具有抗菌、抗疟活性以及溶血活性。
T2732 (-)-Epicatechin gallate

表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG

Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
(-)-Epicatechin gallate ((-)-Epicatechin 3-O-gallate) 抑制环加氧酶-1 的IC50值为 7.5 μM。

天然产物

Gramicidin
Cat.No: T1130
Synonym: 短杆菌肽,Gramicidinum,Gramicidine,Gramicidina
Target: MRP, Antibacterial, Antibiotic
Gramicidin C
Cat.No: T41042
Synonym:
Target:
Gramicidin A
Cat.No: T36439
Synonym:
Target: Antibacterial, HIF, Parasite
(-)-Epicatechin gallate
Cat.No: T2732
Synonym: 表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG
Target: Virus Protease, COX, Autophagy
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