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Cat. No. Product Name Target Signaling Pathways
T60521 Doxepin

作为三环类抗抑郁药,Doxepin 抑制血清素和去甲肾上腺素的再摄取。Doxepin 具有抗炎作用,可减少抗氧化应激。Doxepin 显示出对特应性皮炎和慢性荨麻疹的治疗效果,并且能改善认知过程和保护中枢神经系统。
T1540 Doxepin hydrochloride

Toruan,Doxepin HCl,Aponal,Novoxapin,盐酸多塞平

P450; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Doxepin hydrochloride (Aponal) 是一种可口服的三环抗抑郁剂,是选择性组胺受体 H1拮抗剂。它也是 CYP450抑制剂,抑制 CYP450 2C19和 CYP450 1A2。
T11088 Doxepin D3 Hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and
T37307 Nordoxepin hydrochloride

Doxepin is a tricyclic antidepressant. Desmethyldoxepin is the primary metabolite of doxepin, produced by metabolism at the liver. The metabolism of tricyclic antidepressants, including doxepin, is affected by a variety of factors, including age, genetics, and drug-drug interactions.

化合物

Doxepin
Cat.No: T60521
Synonym:
Target:
Doxepin hydrochloride
Cat.No: T1540
Synonym: Toruan,Doxepin HCl,Aponal,Novoxapin,盐酸多塞平
Target: P450, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Doxepin D3 Hydrochloride
Cat.No: T11088
Synonym:
Target: Histamine Receptor
Nordoxepin hydrochloride
Cat.No: T37307
Synonym:
Target:
TargetMol Loading
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