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4

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6993 Tauroursodeoxycholate sodium

牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)

Apoptosis; ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate sodium (TUDC) 是一种内质网应激抑制剂。Tauroursodeoxycholate sodium (TUDC) 抑制ERK,显著降低凋亡分子表达,如caspase-3和caspase-12。
T9154 Sodium taurodeoxycholate hydrate

牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate

Others Others
Sodium taurodeoxycholate hydrate (Taurodeoxycholic acid sodium salt monohydrate) 已用于一项研究,以评估亚胶束浓度的胆汁盐对脂质双层膜的影响。
T67974 Berberine ursodeoxycholate

HTD1801,BUDCA

Berberine ursodeoxycholate (HTD1801) 是一种口服有效的降血脂剂 ,是 Berberine 和 Ursodeoxycholic acid 的一种离子盐。Berberine ursodeoxycholate 具有广泛的代谢活性,可显著降低肝脏脂肪含量。Berberine ursodeoxycholate 可用于研究高脂血症、非酒精性脂肪性肝炎 (NASH) 和糖尿病。
T16998 Tauroursodeoxycholate dihydrate

牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate

ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate dihydrate is an endoplasmic reticulum stress inhibitor. Tauroursodeoxycholate also inhibits ERK. Tauroursodeoxycholate significantly decreases the expression of apoptosis molecules, such as caspase-3 and caspase-12.

化合物

Tauroursodeoxycholate sodium
Cat.No: T6993
Synonym: 牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)
Target: Apoptosis, ERK, Caspase
Sodium taurodeoxycholate hydrate
Cat.No: T9154
Synonym: 牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate
Target: Others
Berberine ursodeoxycholate
Cat.No: T67974
Synonym: HTD1801,BUDCA
Target:
Tauroursodeoxycholate dihydrate
Cat.No: T16998
Synonym: 牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate
Target: ERK, Caspase
Cat. No. Product Name Target Signaling Pathways
T5077 Deoxycholic acid sodium salt

脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid sodium salt (Sodium deoxycholate) 是 G 蛋白偶联胆汁酸受体TGR5的激活剂。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
T5254 Glycodeoxycholate Sodium

Sodium glycyldeoxycholate,Sodium glycodeoxycholate,Glycodeoxycholic acid sodium salt,脱氧甘胆酸钠

Others; Endogenous Metabolite Metabolism; Others
Glycodeoxycholate Sodium (Glycodeoxycholic acid sodium salt) 诱导肝细胞凋亡的机制与内切酶的DNA裂解有关。它是一种次级胆汁酸,由结肠环境中微生物菌群中存在的酶的作用产生。
T2532 Tauroursodeoxycholate

Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA

Apoptosis; ERK; P450; Caspase; Endogenous Metabolite Apoptosis; MAPK; Metabolism; Proteases/Proteasome
Tauroursodeoxycholate (UR 906),又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
T13916 Taurochenodeoxycholate-3-sulfate

Others Others
Taurochenodeoxycholate-3-sulfate is a bile salt found in urine.

天然产物

Deoxycholic acid sodium salt
Cat.No: T5077
Synonym: 脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
Glycodeoxycholate Sodium
Cat.No: T5254
Synonym: Sodium glycyldeoxycholate,Sodium glycodeoxycholate,Glycodeoxycholic acid sodium salt,脱氧甘胆酸钠
Target: Others, Endogenous Metabolite
Tauroursodeoxycholate
Cat.No: T2532
Synonym: Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA
Target: Apoptosis, ERK, P450, Caspase, Endogenous Metabolite
Taurochenodeoxycholate-3-sulfate
Cat.No: T13916
Synonym:
Target: Others
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