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Targets Recommended: Others

32

抑制剂 & 化合物

30

天然产物

8

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T10811 Chymase-IN-1

Others Others
Chymase-IN-1 是一个有效的,有选择性的,口服有活性的人肥大细胞糜蛋白酶抑制剂,IC50 为 29 nM。
TP1018L Urechistachykinin II acetate

Urechistachykinin II acetate(149097-04-1 free base),Uru-TK II acetate

Others Others
Urechistachykinin II acetate (Uru-TK II acetate)(149097-04-1 free base) 是一种从类胡萝卜素蠕虫中分离出来的无脊椎动物快速激肽相关肽 (TRPs),显示出抗菌活性而没有溶血作用。
TP1019L Urechistachykinin I acetate(149097-03-0 free base)

Uru-TK I acetate

Antibacterial Microbiology/Virology
Urechistachykinin I acetate(149097-03-0 free base) (Uru-TK I acetate) 是一种从类囊体线虫中分离出来的无脊椎动物加利宁相关肽 (TRP)。
T9417L gamma-preprotachykinin amide (72-92) acetate

gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)

Others Others
gamma-preprotachykinin amide (72-92) acetate 是一种 21 个氨基酸的肽,属于速激肽 (TK) 家族,在其 C 末端序列中包括神经激肽 A (NKA)。它对中枢 NK-2 受体的亲和力高于 NKA;它对 NK-1 受体的亲和力较低,但是,它有效地刺激唾液分泌,这是由 NK-1 受体激活介导的。
T73594 Chymotrypsin

Chymotrypsin A

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
Chymotrypsin (Chymotrypsin A) 是胰腺产生的丝氨酸蛋白酶,可切割芳香族氨基酸羧基侧的蛋白质链。
T21417 Dihydrotachysterol

Hytakerol,HSDB-3314,双氢速甾醇,HSDB3314,Parterol,HSDB 3314

Dihydrotachysterol (DHT) is a biologically active synthetic analog of vitamin D. It promotes intestinal absorption of active calcium and phosphate . It is also beneficial in the treatment of hypoparathyroidism.
T22928L Locustatachykinin I acetate

Others Others
Locustachykinin I acetate 是 Lacanobia 中脱酰胺酶的底物。它是一种从飞蝗中分离的昆虫速激肽相关肽。
T76157 Chymotrypsinogen

Chymotrypsinogen 是Chymotrypsin 的无活性前体。Chymotrypsinogen 是一种由胰腺产生的丝氨酸蛋白酶 (serine protease)。
T125775 Stachybotrin E

Stachybotrin E 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125775,CAS号为 1510813-72-5。
T26202 SP-Chymostatin B

alpha-Mapi

SP-Chymostatin B is a potent inhibitor of many proteases, including chymotrypsin, papain, chymotrypsin-like serine proteinases, chymases, and lysosomal cysteine proteinases. It weakly inhibits human leucocyte elastase. It is effective at a final concentra
T81919 Locustatachykinin II

Lom-TK II

Locustachykinin II (Lom-TK II)为具有同源性的昆虫神经肽,与脊椎动物的tachykinin肽家族相似。此化合物适用于研究昆虫的内分泌系统。
T80041 Tachyplesin I

Tachyplesin I为含17个氨基酸残基的β-发夹抗菌肽,对多种人类肿瘤细胞系具有细胞毒性,主要作用机制为破坏外细胞膜完整性。
T125839 Brachynoside

Brachynoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125839。
T126145 Teukotschyn

T125301 Chysin A

T9417 gamma-preprotachykinin amide (72-92)

gamma-preprotachykinin amide (72-92) 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T9417,CAS号为 114882-65-4。
T124366 Psilostachyin B

Psilostachyin B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124366,CAS号为 6995-02-4。
T75089 Selachyl alcohol

Selachyl alcohol是一种具有口服活性的降压剂,与抗高血压中性重髓质脂(ANRL)活性相似。这种烷基甘油化合物存在于鲨鱼鱼肝油混合物中,具有减少肺转移特性,可用于心血管疾病研究。
T125059 Xanthochymusside

T125165 Stachysterone D

Stachysterone D 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125165。
T34180 Psilostachyin C

NSC 106392

Psilostachyin c is a member of the class of compounds known as ambrosanolides and secoambrosanolides. Ambrosanolides and secoambrosanolides are sesquiterpene lactones from the Ambrosia family, with a backbone derivative of azuleno[6,5-b]furan-2-one (ambro
T39184 Tachysterol 3

Tachysterol 3 is a side product in vitamin D photosynthesis.
T24849 TachypleginA-2

tA 2,tA-2,tA2

TachypleginA-2 is a parasite motility and invasion inhibitor.
T12450 Chymase-IN-2

Others Others
Chymase-IN-2 is a modulator of chymase.
T126479 Brachystemidine F

Brachystemidine F 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126479,CAS号为 1050363-02-4。
T10026 Tachykinin angatonist 1

Tachykinin antagonist 1

Others Others
Tachykinin antagonist 1 is an antagonist of neurokinin receptors.
TP1019 Urechistachykinin I

Uru-TK I

Urechistachykinin I (Uru-TK I) is an invertebrate kalinin-related peptide (TRPs) isolated from thylakoid nematodes.
T22928 Locustatachykinin I

Others Others
Insect tachykinin-related peptide (TRP)
T24848 TachypleginA

Tachyplegin A,Tachyplegin-A

TachypleginA is a parasite motility and invasion inhibitor.
T125774 Stachybotrin F

Stachybotrin F 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125774,CAS号为 1510813-73-6。
TP1018 Urechistachykinin II

Uru-TK II

Urechistachykinin II (Uru-TK II) is an invertebrate rapid kinin-related peptide (TRPs) isolated from carotenoid worms.
T37312 Isotachysterol 3

Isotachysterol 3, an analog of 1,25-dihydroxy Vitamin D3, was found to enhance intestinal calcium transport and stimulate bone calcium mobilization in anephric rats[1].

化合物

Chymase-IN-1
Cat.No: T10811
Synonym:
Target: Others
Urechistachykinin II acetate
Cat.No: TP1018L
Synonym: Urechistachykinin II acetate(149097-04-1 free base),Uru-TK II acetate
Target: Others
Urechistachykinin I acetate(149097-03-0 free base)
Cat.No: TP1019L
Synonym: Uru-TK I acetate
Target: Antibacterial
gamma-preprotachykinin amide (72-92) acetate
Cat.No: T9417L
Synonym: gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)
Target: Others
Chymotrypsin
Cat.No: T73594
Synonym: Chymotrypsin A
Target: Serine/threonin kinase
Dihydrotachysterol
Cat.No: T21417
Synonym: Hytakerol,HSDB-3314,双氢速甾醇,HSDB3314,Parterol,HSDB 3314
Target:
Locustatachykinin I acetate
Cat.No: T22928L
Synonym:
Target: Others
Chymotrypsinogen
Cat.No: T76157
Synonym:
Target:
Stachybotrin E
Cat.No: T125775
Synonym:
Target:
SP-Chymostatin B
Cat.No: T26202
Synonym: alpha-Mapi
Target:
Locustatachykinin II
Cat.No: T81919
Synonym: Lom-TK II
Target:
Tachyplesin I
Cat.No: T80041
Synonym:
Target:
Brachynoside
Cat.No: T125839
Synonym:
Target:
Teukotschyn
Cat.No: T126145
Synonym:
Target:
Chysin A
Cat.No: T125301
Synonym:
Target:
gamma-preprotachykinin amide (72-92)
Cat.No: T9417
Synonym:
Target:
Psilostachyin B
Cat.No: T124366
Synonym:
Target:
Selachyl alcohol
Cat.No: T75089
Synonym:
Target:
Xanthochymusside
Cat.No: T125059
Synonym:
Target:
Stachysterone D
Cat.No: T125165
Synonym:
Target:
Psilostachyin C
Cat.No: T34180
Synonym: NSC 106392
Target:
Tachysterol 3
Cat.No: T39184
Synonym:
Target:
TachypleginA-2
Cat.No: T24849
Synonym: tA 2,tA-2,tA2
Target:
Chymase-IN-2
Cat.No: T12450
Synonym:
Target: Others
Brachystemidine F
Cat.No: T126479
Synonym:
Target:
Tachykinin angatonist 1
Cat.No: T10026
Synonym: Tachykinin antagonist 1
Target: Others
Urechistachykinin I
Cat.No: TP1019
Synonym: Uru-TK I
Target:
Locustatachykinin I
Cat.No: T22928
Synonym:
Target: Others
TachypleginA
Cat.No: T24848
Synonym: Tachyplegin A,Tachyplegin-A
Target:
Stachybotrin F
Cat.No: T125774
Synonym:
Target:
Urechistachykinin II
Cat.No: TP1018
Synonym: Uru-TK II
Target:
Isotachysterol 3
Cat.No: T37312
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1563 Dehydropachymic acid

Autophagy; Immunology/Inflammation related Autophagy; Immunology/Inflammation
Dehydropachymic acid 是从茯苓中分离出的一种三萜类天然产物,有抗炎活性。
T6S0619 Pachymic acid

3-O-Acetyltumulosic acid,茯苓酸

ERK; Akt Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Pachymic acid (3-O-Acetyltumulosic acid) 是来自茯苓的一种三萜,可抑制Akt 和ERK 信号传导途径。
T5620 Fenchyl Alcohol

Fenchol,葑醇

Others Others
Fenchyl Alcohol 是一种提取自道格拉斯松叶精油中的单萜醇,可用作香精。它能够显著的抑制绵羊和鹿瘤胃微生物的活性。
T5769 Stachydrine

Methyl hygrate betaine,水苏碱,L-stachydrine,Proline betaine,N,N-Dimethyl-L-proline

NF-κB; Endogenous Metabolite Metabolism; NF-κB
Stachydrine (N,N-Dimethyl-L-proline) 是中国草本植物益母草的主要成分,具有促进血液循环和消除血瘀的功效。Stachydrine (N,N-Dimethyl-L-proline) 能够抑制NF-κB 信号通路。
T5809 Stachyose hydrate

Stachyose,水苏糖

Others Others
Stachyose hydrate 是一种能够增强有益细菌的生长和活性的益生元。它具有降血糖作用,能够调节肠道微生物而改善炎症。
T37267 Pachybasin

Antibacterial Microbiology/Virology
Pachybasin 是一种蒽醌真菌代谢物。 Pachybasin 对大肠杆菌、枯草芽孢杆菌、M. luteus、S. cerevisiae、C. albicans、A. niger 和 A. flavus 具有抗菌活性,MIC 值为 64.0 μg/mL,对金黄色葡萄球菌具有抗菌活性 和尖孢镰刀菌,MIC 值分别为 32.0 和 16.0 μg/mL。
T3251 Stachydrine Hydrochloride

NF-κB NF-κB
Stachydrine hydrochloride 是Herba Leonuri 的主要活性成分,可以抑制NF-κB 信号通路。它可用于心血管疾病的研究,具有抗心肌肥大活性 。
T2713 Stachyose tetrahydrate

Stachyose,D-Stachyose tetrahydrate,水苏糖

Apoptosis; Others Apoptosis; Others
Stachyose tetrahydrate (D-Stachyose tetrahydrate) 是一种功能性低聚糖,可在肠道内产生有益物质或通过促进益生菌的增殖,间接防止结肠癌细胞生长,可作为益生元。
T40975 Stachyanthuside A

Stachyanthuside A, an ellagic acid glycoside, has been isolated from the leaves of Diplopanax stachyanthus.
TN4731 Pachyaximine A

Antifection Microbiology/Virology
Pachyaximine A possesses significant antibacterial activity against Escherichia coli, Staphylococcus aureus, Corynebacterium diphtheriae and Corynebacterium pyrogenes. (-)-Pachyaximine A demonstrates significant activity as antiestrogen binding site (AEBS
TN6481 Achyranthoside D

Achyranthoside D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6481,CAS号为 168009-91-4。
T82706 Clonostachydiol

Clonostachydiol为源于真菌Clonostachys cylindrospora(菌株FH-A 6607)的大分子内酯类驱虫药。
TN5128 Tetrachyrin

Others Others
Tetrachyrin是一种天然产物,属于菊科蟛蜞菊属,其产品编号为 TN5128,CAS号为 73483-88-2。Tetrachyrin可用作对照参考。
TN5057 Stachybotramide

LDL Metabolism
Stachybotramide preferentially stimulate the plasma cholesteryl ester transfer protein (CETP)-mediated transfer of cholesteryl esters (CE) from high density lipoprotein (HDL) to both very low density lipoprotein (VLDL) and low density lipoprotein (LDL).
T37451 Stachybotrysin B

Stachybotrysin B is a fungal metabolite originally isolated from S. chartarum and has antiviral and anticancer activities.1,2 It has antiviral activity against HIV in SupT1 cells (IC50 = 19.2 μM).1 Stachybotrysin B is cytotoxic to K562, HeLa, and HL-60 cells (IC50s = 21.72, 39.63, and 18.5 μM, respectively).2 |1. Zhao, J., Feng, J., Tan, Z., et al. Stachybotrysins A-G, phenylspirodrimane derivatives from the fungus Stachybotrys chartarum. J. Nat. Prod. 80(6), 1819-1826 (2017).|2. Ma, X.-h., Zhen...
TN6131 Leptostachyol acetate

Leptostachyol acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6131,CAS号为 35770-58-2。
TN6167 2-Demethoxyleptostachyol acetate

2-Demethoxyleptostachyol acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6167,CAS号为 139405-55-3。
T31767 Fenchyl acetate

NSC404295,NSC 404295,NSC-404295

Fenchyl acetate is a fragrance ingredient.
TN2032 Pachypodol

霍香黃酮醇

Antifection Microbiology/Virology
Pachypodol has antibacterial and antifungal activities against Bacillus subtilis, Staphylococcus aureus, Staphylococcus faecalis, Echerichia coli, Pseudomonas aeruginosa, Candida albicans, Candida krusei and Candida galabrata.
TN5058 Stachybotrolide

Others Others
Stachybotrolide is a natural product from Stachybotrys alternans.
TN3345 Achyranthoside C

Others Others
Achyranthoside C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3345,CAS号为 168009-90-3。
TN5357 Bistachybotrysin E

Bistachybotrysin E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5357,CAS号为 2231761-98-9。
T65444 Stachyose

Stachyose 是一种天然产物,可用于生命科学领域的相关研究,其产品编号为 T65444。
TN6180 6-Demethoxyleptostachyol acetate

6-Demethoxyleptostachyol acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6180,CAS号为 126298-48-4。
TN3536 Brachynoside heptaacetate

Others Others
Brachynoside heptaacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3536,CAS号为 144765-80-0。
TN4718 Orobanchyl acetate

Others Others
Orobanchyl acetate is a germination stimulant for root parasitic plants.
TN5059 Stachybotrylactam

Others Others
Stachybotrylactam has toxicity.
T82825 Brachyoside B

Brachyoside B,一种三萜皂苷,源自Astragalus wiedemannianus。
TN4732 Pachysamine M

Others Others
Pachysamine M shows inhibitory activities against multiple types of cancer cells.
TN1247 3-Epidehydropachymic acid

Others Others
3-Epidehydropachymic acid is a natural product

天然产物

Dehydropachymic acid
Cat.No: TN1563
Synonym:
Target: Autophagy, Immunology/Inflammation related
Pachymic acid
Cat.No: T6S0619
Synonym: 3-O-Acetyltumulosic acid,茯苓酸
Target: ERK, Akt
Fenchyl Alcohol
Cat.No: T5620
Synonym: Fenchol,葑醇
Target: Others
Stachydrine
Cat.No: T5769
Synonym: Methyl hygrate betaine,水苏碱,L-stachydrine,Proline betaine,N,N-Dimethyl-L-proline
Target: NF-κB, Endogenous Metabolite
Stachyose hydrate
Cat.No: T5809
Synonym: Stachyose,水苏糖
Target: Others
Pachybasin
Cat.No: T37267
Synonym:
Target: Antibacterial
Stachydrine Hydrochloride
Cat.No: T3251
Synonym:
Target: NF-κB
Stachyose tetrahydrate
Cat.No: T2713
Synonym: Stachyose,D-Stachyose tetrahydrate,水苏糖
Target: Apoptosis, Others
Stachyanthuside A
Cat.No: T40975
Synonym:
Target:
Pachyaximine A
Cat.No: TN4731
Synonym:
Target: Antifection
Achyranthoside D
Cat.No: TN6481
Synonym:
Target:
Clonostachydiol
Cat.No: T82706
Synonym:
Target:
Tetrachyrin
Cat.No: TN5128
Synonym:
Target: Others
Stachybotramide
Cat.No: TN5057
Synonym:
Target: LDL
Stachybotrysin B
Cat.No: T37451
Synonym:
Target:
Leptostachyol acetate
Cat.No: TN6131
Synonym:
Target:
2-Demethoxyleptostachyol acetate
Cat.No: TN6167
Synonym:
Target:
Fenchyl acetate
Cat.No: T31767
Synonym: NSC404295,NSC 404295,NSC-404295
Target:
Pachypodol
Cat.No: TN2032
Synonym: 霍香黃酮醇
Target: Antifection
Stachybotrolide
Cat.No: TN5058
Synonym:
Target: Others
Achyranthoside C
Cat.No: TN3345
Synonym:
Target: Others
Bistachybotrysin E
Cat.No: TN5357
Synonym:
Target:
Stachyose
Cat.No: T65444
Synonym:
Target:
6-Demethoxyleptostachyol acetate
Cat.No: TN6180
Synonym:
Target:
Brachynoside heptaacetate
Cat.No: TN3536
Synonym:
Target: Others
Orobanchyl acetate
Cat.No: TN4718
Synonym:
Target: Others
Stachybotrylactam
Cat.No: TN5059
Synonym:
Target: Others
Brachyoside B
Cat.No: T82825
Synonym:
Target:
Pachysamine M
Cat.No: TN4732
Synonym:
Target: Others
3-Epidehydropachymic acid
Cat.No: TN1247
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-01936 VEGFR3/FLT4 Protein, Mouse, Recombinant (His)

Flt-4,VEGFR-3,Chy,fms related tyrosine kinase 4,VEG...

Mouse HEK293 Cells
VEGFR3/FLT4 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 86.4 kDa and the accession number is P35917-1.
TMPY-01937 VEGFR3/FLT4 Protein, Mouse, Recombinant (hFc)

VEGFR-3,fms related tyrosine kinase 4,VEGFR3,Flt-4,AI323512,...

Mouse HEK293 Cells
VEGFR3/FLT4 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 112 kDa and the accession number is P35917-1.
TMPY-02574 Chymase 1 Protein, Human, Recombinant (His)

MCT1,chymase 1, mast cell,chymase,CYH

Human Baculovirus Insect Cells
The STR polymorphism in the CMA1 gene is associated with asthma and that this association is even stronger with atopic asthma. CMA1 and IL-4 in atopic asthma and for IL-4 in atopy in general. The local angiotensin II system (LAS) has numerous functions, including the regulation of growth and differentiation in the gastrointestinal tract. Angiotensin II (AngII) may be generated by angiotensin-I-converting enzyme (ACE) or mast cell chymase (CMA1) and plays an important role in inflammatory process...
TMPH-03618 Clotting factor C Protein, Tachypleus tridentatus, Recombinant (His & Myc)

FC,Limulus factor C,Clotting factor C

Tachypleus tridentatus E. coli
This enzyme is closely associated with an endotoxin-sensitive hemolymph coagulation system which may play important roles in both hemostasis and host defense mechanisms. Its active form catalyzes the activation of clotting factor B. Clotting factor C Protein, Tachypleus tridentatus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.8 kDa and the accession number is P28175.
TMPH-02581 Chymase 1 Protein, Mouse, Recombinant (His)

Mast cell protease 5,Mast cell protease I,Alpha-chy...

Mouse E. coli
Major secreted protease of mast cells with suspected roles in vasoactive peptide generation, extracellular matrix degradation, and regulation of gland secretion. Chymase 1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 29.2 kDa and the accession number is P21844.
TMPY-02480 Chymotrypsin C Protein, Human, Recombinant (His)

ELA4,CLCR,chymotrypsin C (caldecrin)

Human HEK293 Cells
Chymotrypsin C (abbreviated for CTRC), also known as caldecrin or elastase4, is a digestive enzyme of the peptidase S1 family. This enzyme is synthesized as an inactivate chymotrypsinogen. On cleavage by trypsin into two parts that activate each other by removing two small peptides in a trans-proteolysis, chymotrypsin C produced. N-linked glycosylation of human CTRC is required for efficient folding and secretion, however, the N-linked glycan is unimportant for enzyme activity or inhibitor bindi...
TMPH-03639 COX7A1 Protein, Trachypithecus cristatu, Recombinant (hFc)

Cytochrome c oxidase subunit VIIa-H,COX7A1,Cytochrome c oxid...

Trachypithecus cristatus HEK293 Cells
N/A. COX7A1 Protein, Trachypithecus cristatu, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 31.9 kDa and the accession number is Q9N234.
TMPH-00486 Chymase Protein, Canine, Recombinant (His & SUMO)

Chymase,Alpha-chymase,CMA1,Mast cell prote...

Canine E. coli
Chymase Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli.

重组蛋白

VEGFR3/FLT4 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01936
Species: Mouse
Expression System: HEK293 Cells
VEGFR3/FLT4 Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-01937
Species: Mouse
Expression System: HEK293 Cells
Chymase 1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02574
Species: Human
Expression System: Baculovirus Insect Cells
Clotting factor C Protein, Tachypleus tridentatus, Recombinant (His & Myc)
Cat.No: TMPH-03618
Species: Tachypleus tridentatus
Expression System: E. coli
Chymase 1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02581
Species: Mouse
Expression System: E. coli
Chymotrypsin C Protein, Human, Recombinant (His)
Cat.No: TMPY-02480
Species: Human
Expression System: HEK293 Cells
COX7A1 Protein, Trachypithecus cristatu, Recombinant (hFc)
Cat.No: TMPH-03639
Species: Trachypithecus cristatus
Expression System: HEK293 Cells
Chymase Protein, Canine, Recombinant (His & SUMO)
Cat.No: TMPH-00486
Species: Canine
Expression System: E. coli
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