Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1830 |
BX795
|
IκB/IKK; Chk; CDK; c-Kit; PDK; Autophagy | Autophagy; Cell Cycle/Checkpoint; NF-κB; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
BX795 是一种选择性PDK1抑制剂,也是相对特异性的TBK1和IKKɛ 抑制剂。它抑制 S6K1,Akt,PKCδ 和 GSK3β 的磷酸化,可调节自噬。 | |||
T70578 | BX-795 hydrochloride | ||
BX-795 hydrochloride is a TBK1 and IKKε inhibitor. BX-795 is a potential maternal embryonic leucine zipper kinase inhibitor. |