19
7
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14615 |
Biphenylindanone A
BINA |
GluR | Neuroscience |
Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders. | |||
T0888 |
Felbinac
Dapson,4-联苯乙酸,4-Biphenylacetic acid |
COX | Immunology/Inflammation; Neuroscience |
Felbinac (Dapson) 是非甾体抗炎药,可用于肌肉炎症和关节炎的研究。 | |||
T12241 |
Norbinaltorphimine dihydrochloride
nor-BNI dihydrochloride,Nor-BNI dihydrochloride,nor-Binaltorphimine dihydrochloride,Nor-Binaltorphimine dihydrochloride |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Norbinaltorphimine dihydrochloride是一种具有选择性和有效性的κ阿片受体 (κ opioid receptor) 拮抗剂,可在小鼠中诱导瘙痒相关反应。 | |||
TP2075L |
Bombinakinin M acetate
Bombinakinin M acetate(509151-65-9 free base) |
Bradykinin Receptor | GPCR/G Protein |
Bombinakinin M acetate 是一种有效的缓激肽受体激动剂,对哺乳动物动脉平滑肌缓激肽受体具有高度选择性,其效力比缓激肽高约 50 倍。 | |||
T0013 |
Mecarbinate
优多降,Dimecarbine,Dimecarbin,美卡比酯 |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
Mecarbinate (Dimecarbin) 是抗 HCV 试剂,也是中间体。 | |||
T31759 |
Felbinac Trometamol
L141,Felbinac,L-141,L 141 |
||
Felbinac Trometamol is an intravenous preparation used to treat severe postoperative pain. | |||
T23757 |
Ascorbic acid, rutoside drug combination
Rutinoscorbin,Rutascorbin,Ruta C 60,Cerutin |
||
Ascorbic acid, rutoside drug combination is used for treating diabetic retinopathy. | |||
TP2075 |
Bombinakinin M
|
||
Potent bradykinin receptor agonist. Highly selective for mammalian arterial smooth muscle bradykinin receptors, displaying ~ 50-fold greater potency than bradykinin. Elicits dose-dependent contractile effects in smooth muscle of guinea pig ileum (EC50 = 4 | |||
T6702L |
Terbinafine lactate
DRG-0286,Terbinafine hydrochloride,Lamisil Krem,SF 86-327 hydrochloride,Lamisil,Lamisil AT |
||
Terbinafine, a synthetic allylamine antifungal, inhibits ergosterol synthesis by inhibiting squalene epoxidase, an enzyme that is part of the fungal cell membrane synthesis pathway. | |||
T32536 |
l-Adrenalin ascorbinate
Tonhormon |
||
l-Adrenalin ascorbinate is a bioactive chemical. | |||
T66567 |
Diacetato[(R)-(+)-2,2'-bis(diphenylphosphino)-1,1'-binaphthyl]ruthenium(II)
|
||
Diacetato[(R)-(+)-2,2'-bis(diphenylphosphino)-1,1'-binaphthyl]ruthenium(II) 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66567,CAS号为 325146-81-4。 | |||
T64532 | Rac-Binap Pd G3 | ||
[2'-(Amino-κN)[1,1'-biphenyl]-2-yl-κC][[2'-(diphenylphosphino)[1,1'-binaphthalen]-2-yl]diphenylphosphine-κP](methanesulfonato-κO)palladium 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64532。 | |||
T75395 | alpha-2-3,6-sialidase (BiNanH2) | ||
alpha-2-3,6-sialidase (BiNanH2) 为一种生化研究常用的唾液酸转移酶,催化 α-2,3/2,6-唾液酸从 CMP-Neu5Ac 转移到半乳糖苷受体。 | |||
TP2225 |
Bombinakinin-GAP
|
Others | Others |
Bioactive bradykinin-related peptide | |||
T81573 |
Pabinafusp alfa
JR-141 |
||
Pabinafusp alfa (JR-141) 是由Iduronate 2-sulfatase和抗人转铁蛋白受体抗体结合而成的转铁蛋白受体靶向抗体。它具备穿透血脑屏障的能力,可防止粘多糖病II型(MPS II)小鼠中枢神经系统中硫酸肝素(HS)的积累。此外,Pabinafusp alfa能够促进小鼠的学习能力,并抑制中枢神经系统神经元的损伤。 | |||
T76202 | Recombinant Proteinase K | ||
Recombinant Proteinase K为一种serine protease,专门裂解脂肪族及芳香族氨基酸的羧基端肽键,适用于蛋白质消化与清除核酸制剂中的污染。 | |||
T79925 |
T4 UvsX Recombinase
|
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
T4 UvsX Recombinase 促进双链DNA模板上DNA复制的启动,通过催化模板DNA与同源单链DNA引物间的突触形成。此酶显著增强了T4 DNA聚合酶全酶在线性单链DNA模板上进行的回跳(发夹引物)DNA合成反应。 | |||
T71523 | Norbinaltorphimine | ||
nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist. | |||
T13946 |
Turbinaric acid
|
Others | Others |
Turbinaric acid, a secosqualene carboxylic acid with cytotoxic properties, originates from the brown alga Turbinaria ornata. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1411 |
Terbinafine hydrochloride
KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。 | |||
T6702 |
Terbinafine
Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067 |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Terbinafine (TDT 067) 是念珠菌属的角鲨烯环氧化酶有效的非竞争性抑制剂,Ki 值为 30 nM。它具有抗真菌感染活性。 | |||
TN3626 | Cerbinal | Antifection | Microbiology/Virology |
Cerbinal 是一种天然化合物,来源于非洲非洲菊的草本植物。它具有杀虫活性,是一种潜在的新型害虫防治剂。 | |||
T79953 |
Acetyl-binankadsurin A
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Acetyl-binankadsurin A(化合物5)是从南五味子(Kadsura longipedunculata)中提取的一种木脂素。该化合物对HIV-1蛋白酶表现出较低的抑制活性,其半抑制浓度(IC50)超过100 μg/mL。 | |||
T83117 |
Angeloylbinankadsurin A
|
||
Angeloylbinankadsurin A(化合物7)是一种从黑虎胡的EtOAc和CH2Cl2提取物中分离出的抗RA试剂,它在RA-FLS细胞上显示出显著的抑制活性(IC50=11.70 μM),同时对人类癌细胞系(Hela和BGC-823)表现出较低的毒性(IC50分别为19.9 μM和21.93 μM)。 | |||
TN2162 |
Rubinaphthin A
|
Others | Others |
Rubinaphthin A is a natural product from Rubia cordifolia. | |||
TN5495 | 3',3'''-Binaringenin | ||
3',3'''-Binaringenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5495,CAS号为 145399-99-1。 |