38
12
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24055 |
FAUC 213
FAUC213,FAUC-213 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
FAUC 213 是一种具有口服活性的‘、高度选择性的、可透过血脑屏障的多巴胺 D4受体完全拮抗剂,对 hD4.4的 Ki=2.2 nM。它对 D2和 D3受体的活性较低,对于 hD2、hD3的 Ki 分别为 3.4 μM、5.3 μM。它表现出非典型的抗精神病活性。 | |||
T1550 |
Thiamphenicol
甲砜霉素,Dextrosulphenidol,Thiophenicol |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。 | |||
T20525 |
Chloramphenicol palmitate
|
Antibacterial; Antibiotic | Microbiology/Virology |
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。 | |||
T7465 |
4-Methylbenzylidene camphor
Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC |
AChE | Neuroscience |
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。 | |||
T25239 |
Chloramphenicol stearate
Eusynthomycin,Chloramphenicol monostearate,Madomicetina |
||
Chloramphenicol stearate is an antibiotic useful for the therapy of numbers of bacterial infections. This includes an eye ointment to treat conjunctivitis. | |||
T74079 |
m-Chloramphenicol
|
||
m-Chloramphenicol (m-threo-Chloramphenicol) 是 Chloramphenicol 的一种杂质。Chloramphenicol 是一种广谱抗生素,是细菌蛋白质生物合成的有效抑制剂。 | |||
T10311 |
Amphotericin X1
两性霉素 X1 |
Others | Others |
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2 | |||
TF0050 |
Amphipol A8-35
|
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Amphipol A8-35 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0050,CAS号为 326856-53-5。 | |||
T72093 |
Thiamphenicol glycinate hydrochloride
甲砜霉素甘氨酸酯盐酸盐 |
||
Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。 | |||
T74061 | Amphotericin B methyl ester hydrochloride | ||
Amphotericin B methyl ester hydrochloride 是多烯类抗生素 Amphotericin B (A634250) 的甲酯衍生物。Amphotericin B methyl ester hydrochloride 是胆固醇结合物,具有显著的抗真菌活性。Amphotericin B methyl ester hydrochloride 干扰HIV-1颗粒的产生,抑制HIV-1的复制。 | |||
T35651 |
Bromamphenicol
|
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Bromamphenicol is a dibrominated derivative of the antibiotic chloramphenicol. It inhibits rat liver mitochondrial and E. coli protein synthesis by 90.6 and 98.8%, respectively, when used at a concentration of 93 μM, and inhibits DNA synthesis in human lymphoblastoid cells by 83% at 1 mM. Bromamphenicol can also bind to the major adhesin subunit DraE from E. coli. | |||
T73891 |
Amphotericin A
|
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Amphotericin A 是一种有效的抗真菌抗生素。 | |||
T64105 |
Voriconazole camphorsulfonate
|
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Voriconazole (UK-109496) camphorsulfonate 是一种二代广谱的三唑类抗真菌 (antifungal) 化合物,对真菌麦角甾醇的生物合成表现出抑制作用。Voriconazole camphorsulfonate 能够抑制由真菌细胞色素 P450 酶介导的 14-α-羊毛甾醇去甲基化作用,表现出抗真菌效果。 | |||
T65136 |
Camphorquinone
|
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Camphorquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65136,CAS号为 10373-78-1。 | |||
T66682 |
(1R,3S)-(+)-Camphoric acid
|
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(1R,3S)-(+)-Camphoric acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66682,CAS号为 124-83-4。 | |||
T71810 |
Thiamphenicol palmitate
|
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Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation. | |||
T20401 |
(-)-Isopinocampheol
l-Isopinocampheol |
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(-)-Isopinocampheol is a monoterpene and a component of several plant essential oils. It showed dual viricidal activity against herpes simplex virus 1. | |||
T65673 |
(+)-10,2-Camphorsultam
|
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(+)-10,2-Camphorsultam 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65673,CAS号为 108448-77-7。 | |||
T66968 |
(1S)-(+)-Camphor-10-sulphonic acid
|
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(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。 | |||
T30475 |
Bismuth camphocarbonate
Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth |
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Bismuth camphocarbonate is used for herpes zoster. | |||
T34895 |
Tocamphyl
Tocanfil,Biliphorin,Gallogen |
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Tocamphyl is a cholagogic agent that stimulates pancreatic exocrine and bile flow when administered in the duodenum. | |||
T30040 |
Amphocil
Amphotericin B cholesteryl sulfate |
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Amphocil is used to treat patients with invasive fungal infection. | |||
T25083 |
Amphotalide
RP 6171,RP-6171,RP6171,Schistomide |
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Amphotalide is an anthelminthic agent. | |||
T10309 |
Amphethinile
Amphetinile,CRC 82-07 |
Others | Others |
Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM. | |||
T30037 |
Amphidinolide C
|
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Amphidinolide C is a potent cytotoxic 25-membered macrolide from marine dinoflagellate Amphidinium sp. | |||
T24401 |
L-erythro-Chloramphenicol
L(+)-erythro-Chloramphenicol |
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L-erythro-Chloramphenicol functions as a potent inhibitor of electron transport. | |||
T131515 |
Picroside II (Amphicoside)
|
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Picroside II (Amphicoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131515。 | |||
T30041 |
Amphoglucamine
|
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Amphoglucamine is used in the combined chemotherapy of viral diseases. | |||
T65131 |
(+/-)-10-Camphorsulfonic Acid
|
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(+/-)-10-Camphorsulfonic Acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65131,CAS号为 5872-08-2。 | |||
T71443 |
Amphidinolide D
|
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Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction. | |||
T30036 |
Amphenidone
|
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Amphenidone is a Tranquilizer. | |||
T30038 |
Amphidinolide F
|
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Amphidinolide F is a new cytotoxic macrolide | |||
T66944 | (1R)-(-)-10-Camphorsulfonic acid | ||
(1R)-(-)-10-Camphorsulfonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66944,CAS号为 35963-20-3。 | |||
T20818 |
Propetamphos
Deadmag,Safrotin S 200 |
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Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice. | |||
T124427 |
Camphans?ure (+)-
|
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Camphans?ure (+)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124427,CAS号为 67111-66-4。 | |||
T65662 |
(1S)-(+)-(10-Camphorsulfonyl)oxaziridine
|
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(1S)-(+)-(10-Camphorsulfonyl)oxaziridine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65662,CAS号为 104322-63-6。 | |||
T10310 |
Amphotericin B methyl ester
|
Others | Others |
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV | |||
T30039 |
Amphimedine
|
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Amphimedine is a Pyridoacridine Marine Alkaloid. |
Cat. No. | Product Name | Target | Signaling Pathways |
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T8258 |
Chloramphenicol succinate sodium
Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。 | |||
TMS2262 |
(-)-CAMPHOR
L-Camphor,左旋樟脑 |
Others | Others |
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。 | |||
T20191 |
(-)-Camphoric acid
(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)- |
GluR | Neuroscience |
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。 | |||
T7959 |
(+)-ISOPINOCAMPHEOL
|
Others | Others |
(+)-ISOPINOCAMPHEOL 是一种天然产物。 | |||
T1205 |
Chloramphenicol
Chlornitromycin,Levomycetin,Chloromycetin,氯霉素 |
ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic | Chromatin/Epigenetic; Metabolism; Microbiology/Virology |
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。 | |||
T1067 |
Amphotericin B
NSC 527017,两性霉素B |
Antibiotic; Antifungal | Microbiology/Virology |
Amphotericin B (NSC-527017) 是一种多烯类抗真菌剂,对许多真菌物种具有广谱活性。Amphotericin B 不可逆地结合麦角甾醇,破坏细胞膜完整性,从而起到抗真菌活性。 | |||
T0882 |
(+)-Camphor
D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor |
Antibacterial; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。 | |||
T2952 |
Camphor
樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa |
Influenza Virus; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。 | |||
T25240 |
Chloramphenicol succinate
Paraxin succinate,Kemicetine succinate,CPSA |
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Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol. | |||
T82002 |
Juniper camphor
|
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Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。 | |||
TN4667 |
Norcamphor
|
Others | Others |
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。 | |||
T38588 |
Amphotericin B trihydrate
|
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Amphotericin B trihydrate, a polyene antibiotic, is derived from Streptomyces nodosus fermenter cultures. It exhibits antileishmanial properties. |