Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2479 |
Tyrphostin A9
Malonoben,Tyrphostin 9,SF 6847,AG 17,RG-50872 |
EGFR; VEGFR; Influenza Virus; PDGFR | Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Tyrphostin A9 (SF 6847) 是一种线粒体分裂诱导剂,是 PDGFR 抑制剂,具有抗流感病毒的活性。 | |||
T68822 |
Tyrphostin AG17
|
||
Tyrphostin AG17 is a biochemical that promotes adipocyte apoptosis in vivo and is an effective modulator of adipocyte differentiation and WAT hypertrophy in vitro and in vivo. It is thought to possibly be useful as a pharmacological obesity treatment. It is a tyrosine kinase antagonist that has also been found to inhibit tumor cell growth. | |||
T9121 |
AG-636
|
Dehydrogenase; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
AG-636 是一种选择性可逆和具有口服活性的二氢乳清酸脱氢酶(DHODH)抑制剂,IC50 为 17 nM,具有很强的抗癌作用。 |