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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T14116	ACP-105	Androgen Receptor	Endocrinology/Hormones
	ACP-105 是选择性的、可口服的雄激素受体调节剂 , 能够作用于野生型 AR (pEC50:9.0)和 T877A 突变型 AR (pEC50:9.3)。
T6946	Pimavanserin tartrate ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林	5-HT Receptor	GPCR/G Protein; Neuroscience
	Pimavanserin tartrate (Nuplazid) 是一种有效的5-HT 2A 受体反向激动剂，pIC50和 pKi 值分别为8.73和9.3，用于治疗与帕金森病相关的精神病。
T29614	ACP-0052 SL052,SL 052,SL-052,ACP 0052
	ACP-0052(SL-052, ACP-SL-052) is a photosensitizer based on hypoclintin that may be used in the treatment of prostate cancer.
T2076	Pimavanserin ACP-103,匹莫范色林	5-HT Receptor	GPCR/G Protein; Neuroscience
	Pimavanserin (ACP-103) 是特异性的 5-HT2A 受体反向激动剂，在基于细胞的功能测定中，平均 pIC50值为8.7。它是非典型抗精神病药，用于治疗帕金森病患者的幻觉和精神病。
T3626	Acalabrutinib ACP-196,阿可替尼	BTK	Angiogenesis; Tyrosine Kinase/Adaptors
	Acalabrutinib (ACP-196) 是一种不可逆的、高效的、具有口服活性、选择性的第二代BTK 抑制剂。它与 BTK 的 ATP 结合口袋中的 Cys481 共价结合。它在慢性淋巴细胞性白血病 (CLL) 小鼠模型中显示出强大的靶向作用和功效。
T3484	trans-ACPD Trans-(±)-ACP,1-amino-1,3-dicarboxycyclopentane,(±)-trans-ACPD	GluR	Neuroscience
	trans-ACPD ((±)-trans-ACPD) 是代谢型受体激动剂，可促进钙离子活动及产生内向电流。
TP1837	Acyl Carrier Protein (ACP) (65-74) Acyl Carrier Protein (ACP) 65-74
	Acyl Carrier Protein (ACP) (65-74) is an active acyl carrier protein (ACP) fragment.Acyl Carrier Protein (ACP) is a component of plastid-located plant fatty acid synthetase. It binds acyl groups covalently via the prosthetic group, 4-phosphopantetheine, d
T10240	ACP-5862	BTK	Angiogenesis; Tyrosine Kinase/Adaptors
	ACP-5862 is a major active and pyrrolidine ring-opened metabolite of Acalabrutinib (IC50: 5.0 nM for BTK). Acalabrutinib is an irreversible and highly selective BTK inhibitor (IC50: 3 nM; EC50: 8 nM).
T34657	SL-017 ACPSL-017,S-017,ACP-SL-017,ACP-SL017
	SL-017 (ACP-SL-017, ACPSL-017, ACP-SL-017) is a Hypocrellin-B (Hb) derivative and photosensitization agent that may be used to treat abnormal hair growth. SL017 targets the mitochondria and causes the mitochondrial membrane potential to collapse, producin
T71732	Fmoc-ε-Acp-OH
	Fmoc-ε-Acp-OH can be used as a PROTAC linker in the synthesis of PROTACs and other conjugation applications. Fmoc-ε-Acp-OH is an alkane chian with terminal Fmoc-protected amine and carboxylic acid groups. The Fmoc group can be deprotected under basic condition to obtain the free amine which can be used for further conjugations. The terminal carboxylic acid can react with primary amine groups in the presence of activators (e.g. EDC, or HATU) to form a stable amide bond.
T70840	Osemozotan Free Base
	Osemozotan Free Base is a 5-HT(1A) receptor agonist.
T70842	ACP1b
	ACP1b is an activator of ClpP protease.
TP1427L	ReACp53 acetate	p53	Apoptosis
	ReACp53 acetate 能够抑制 p53 amyloid 的形成, 挽救 p53 在癌细胞中的作用。
T75168	Homo-BacPROTAC7
	Homo-BacPROTAC7 是一个 ClpC1NTDBacPROTAC 降解剂，可以靶向 ClpC2。Homo-BacPROTAC7 能有效杀死 M. tuberculosis。
T22549	ACPT-I	Others	Others
	Agonist for group III mGlu receptors
T22488	(1S,3R)-ACPD	Others	Others
	group I and II mGlu receptor agonist
T22550	ACPT-II	Others	Others
	metabotropic receptor antagonist
T19178	ACPK	Others	Others
	ACPK is a pyrrolysine analogue bearing an azide residue.
T75171	BacPROTAC-1
	BacPROTAC-1 是一个 mSABacPROTAC 降解剂。BacPROTAC-1 对 mSA 和 ClpCNTD 具有高亲和力 (KD 分别为 3.9 μM 和 2.8 μM)。
TP1427	ReACp53
	ReACp53 is a cell-penetrating peptide, designed to inhibit p53 amyloid formation, resues p53 function in cancer cell lines and in organoids derived from high-grade serous ovarian carcinomas (HGSOC).
T75401	D-galactosyl-β1-3-N-acetyl-D-hexosamine phosphorylase (BiGalHexNAcP)
	D-galactosyl-β1-3-N-acetyl-D-hexosamine phosphorylase (BiGalHexNAcP)，属于CAZy糖苷水解酶GH112家族，主要应用于生化研究领域。该酶负责催化lacto-N-biose和lacto-N-neobiose的磷酸化反应，生成Gal-1-磷酸和相应的N-乙酰-D-己糖胺。
T75167	Homo-BacPROTAC6
	Homo-BacPROTAC6 是一个 ClpC1NTDBacPROTAC 降解剂，可以靶向 ClpC2。Homo-BacPROTAC7 能有效杀死M. tuberculosis。
T23080	NPEC-caged-(1S,3R)-ACPD	Others	Others
	group I and II mGlu receptor agonist
T61411	InhA-IN-4	Antibacterial	Microbiology/Virology
	InhA-IN-4 (TU14) 是一种有效的结核分枝杆菌InhA(烯酰 ACP 还原酶) 抑制剂，具有潜在的抗癌和抗增殖活性，可用于研究结核分枝杆菌感染。
T60866	InhA-IN-3	Antibacterial	Microbiology/Virology
	InhA-IN-3 (TU13) 是一种有效的结核分枝杆菌InhA(烯酰 ACP 还原酶) 抑制剂，具有潜在的抗癌和抗增殖活性，可用于研究结核分枝杆菌感染。
T4105L	AFN-1252 tosylate API-1252 tosylate
	AFN-1252 tosylate is an enoyl-ACP Reductase inhibitor.
T70835	（4R，9S)-AG 205
	AG-205 is a potent inhibitor of FabK, the enoyl-ACP reductase in Streptococcus pneumoniae.
T38125	Platencin
	Platencin is a natural, broad spectrum Gram-positive antibiotic isolated from S. platensis, which is also the source of platensimycin . Platencin inhibits two key enzymes in bacterial fatty acid synthesis, β-ketoacyl-ACP synthases II and III (FabF and FabH, respectively), unlike platensimycin which only targets FabF. The IC50 values for platencin against FabF and FabH are 1.95 and 3.91 μg/ml, respectively. It does not exhibit cross-resistance to antibiotic resistant bacterial strains, including ...

化合物

Cat.No: T14116

Target: Androgen Receptor

Pimavanserin tartrate

Cat.No: T6946

Synonym: ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林

Target: 5-HT Receptor

Cat.No: T29614

Synonym: SL052,SL 052,SL-052,ACP 0052

Cat.No: T2076

Synonym: ACP-103,匹莫范色林

Target: 5-HT Receptor

Cat.No: T3626

Synonym: ACP-196,阿可替尼

Target: BTK

Cat.No: T3484

Synonym: Trans-(±)-ACP,1-amino-1,3-dicarboxycyclopentane,(±)-trans-ACPD

Target: GluR

Acyl Carrier Protein (ACP) (65-74)

Cat.No: TP1837

Synonym: Acyl Carrier Protein (ACP) 65-74

Cat.No: T10240

Target: BTK

Cat.No: T34657

Synonym: ACPSL-017,S-017,ACP-SL-017,ACP-SL017

Fmoc-ε-Acp-OH

Cat.No: T71732

Osemozotan Free Base

Cat.No: T70840

Cat.No: T70842

ReACp53 acetate

Cat.No: TP1427L

Target: p53

Homo-BacPROTAC7

Cat.No: T75168

Cat.No: T22549

Target: Others

Cat.No: T22488

Target: Others

Cat.No: T22550

Target: Others

Cat.No: T19178

Target: Others

Cat.No: T75171

Cat.No: TP1427

D-galactosyl-β1-3-N-acetyl-D-hexosamine phosphorylase (BiGalHexNAcP)

Cat.No: T75401

Homo-BacPROTAC6

Cat.No: T75167

NPEC-caged-(1S,3R)-ACPD

Cat.No: T23080

Target: Others

Cat.No: T61411

Target: Antibacterial

Cat.No: T60866

Target: Antibacterial

AFN-1252 tosylate

Cat.No: T4105L

Synonym: API-1252 tosylate

（4R，9S)-AG 205

Cat.No: T70835

Cat.No: T38125

Cat. No.	Product Name	Target	Signaling Pathways
T4852	Trimyristin Trimyristoylglycerol,Tritetradecanoin,三肉豆蔻酸甘油酯,Glyceryl trimyristate,甘油三肉豆蔻酸酯,1,2,3-Tritetradecanoylglycerol	Phosphatase; Endogenous Metabolite; AChE	Metabolism; Neuroscience
	Trimyristin (Tritetradecanoin) 是一种 Myristica fragransHoutt 的有效成分，能够显著抑制乙酰胆碱酯酶 (AChE)，酸性和碱性磷酸酶 (ACP/ALP) 特性。它对 AChE，ACP 和 ALP 的 IC50分别为 0.11、0.16 和 0.18 mM。

天然产物

Cat.No: T4852

Synonym: Trimyristoylglycerol,Tritetradecanoin,三肉豆蔻酸甘油酯,Glyceryl trimyristate,甘油三肉豆蔻酸酯,1,2,3-Tritetradecanoylglycerol

Target: Phosphatase, Endogenous Metabolite, AChE

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