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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T27423	GNE-375 GNE375,GNE 375	Epigenetic Reader Domain; Carboxypeptidase; CDK	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Proteases/Proteasome
	GNE-375 是一种具有选择性和高效性的 BRD9 抑制剂，(IC50：5 nM)。GNE-375 抑制 BRD4、TAF1 和 CECR2，可用于研究表观遗传学耐药性。
T1463	Ramelteon 雷美替胺,TAK-375	Melatonin Receptor; MT Receptor	GPCR/G Protein; Neuroscience
	Ramelteon (TAK-375) 是强效高选择性和可口服的 MT1/MT2激动剂，Ki 值分别为 14 和 112 pM，有用于失眠症的研究潜力。
T39817	Msr-Ratio Msr-green,Msr-Ratio	Others	Others
	Msr-Ratio (Msr-green) (Msr-green) is a ratiometric fluorescent probe specifically designed for the detection of methionine sulfoxide reductase (MSR) activity. It has an excitation wavelength of 375 nm and an emission wavelength of 550 nm. This probe offers the ability to monitor the enzyme activity both in vitro and in live cells, making it a valuable tool for studying MSR function.
T19248	CP 375	Others	Others
	CP 375 is a Fe3+ chelating agent (log K1: 14.50).
T27587	IDX-375
	IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.
T37858	Dehydroergosterol 9,11-dehydro Ergosterol,DHE
	Dehydroergosterol is a naturally occurring, fluorescent analog of cholesterol (ex/em = 324/375 nm) that mimics the properties of cholesterol in cell membranes.[1] It is readily bound by cholesterol-binding proteins and has been used for real-time probing of the sterol environment and to elucidate intracellular sterol trafficking in living organisms.[1]
T41148	Phototrexate
	Phototrexate is a photoswitchable potent inhibitor of human dihydrofolate reductase (DHFR). Phototrexate is a photochromic analog of Methotrexate. Antifolate activity is switched on (cis-Phototrexate) by UVA (375 nm) light; it can be switched off (trans-Phototrexate) by blue or white light and by thermal relaxation in the dark.cis-Phototrexate (IC50 = 6 nM) significantly reduces the viability of HeLa cells compared withtrans-Phototrexate (IC50 = 34 μM).
T63391	Calpain Inhibitor-2
	Calpain Inhibitor-2 是具有亲脂性的钙蛋白酶抑制剂，与黑色素瘤细胞系（A-375和B-16F1）和PC-3前列腺癌细胞相比，他们在体外具有中等到良好的抗增殖效果。Calpain Inhibitor-2 中的化合物3，在基质胶细胞侵袭测定中以2μM 浓度能够抑制了80%的DU-145细胞侵袭。
T40895	Calmodulin antagonist-1
	Calmodulin antagonist-1 (W-7) is a calmodulin (CaM) antagonist that effectively inhibits calmodulin-activated Ca 2+ -phosphodiesterase (PDE) with an IC 50 of 28 μM. This compound also competitively inhibits trypsin-treated Ca 2+ -PDE with respect to cyclic GMP, exhibiting an IC 50 of 375 μM and a K i value of 300 μM.
T83937	Tricyclic cytosine tC
	Tricyclic cytosine tC 是一种用于在活细胞中成像 RNA 的荧光胞嘧啶类似物。当与共聚焦成像技术结合使用时，可用于研究单细胞分辨率下的 RNA 合成、降解和运输。激发/发射最大值 (λ) = 375/505 nm；消光系数 = 4000 M-1cm-1；量子产率 = 0.2。

化合物

GNE-375

Cat.No: T27423

Synonym: GNE375,GNE 375

Target: Epigenetic Reader Domain, Carboxypeptidase, CDK

Ramelteon

Cat.No: T1463

Synonym: 雷美替胺,TAK-375

Target: Melatonin Receptor, MT Receptor

Msr-Ratio

Cat.No: T39817

Synonym: Msr-green,Msr-Ratio

Synonym: 9,11-dehydro Ergosterol,DHE

Calmodulin antagonist-1

Cat.No: T40895

Synonym:

Target:

Tricyclic cytosine tC

Cat.No: T83937

Synonym:

Target:

Cat. No.	Product Name	Target	Signaling Pathways
T5S0055	Chelidonine Helidonine,Khelidonin,白屈菜碱,Stylophorin	Apoptosis; Others; Influenza Virus	Apoptosis; Microbiology/Virology; Others
	Chelidonine (Stylophorin) 是白屈菜中的一种异喹啉生物碱，有抗肿瘤和抗病毒作用。它可导致细胞周期 G2/M 停滞，诱导 caspase 依赖和非依赖性的细胞凋亡。

天然产物

Chelidonine

Cat.No: T5S0055

Synonym: Helidonine,Khelidonin,白屈菜碱,Stylophorin

Target: Apoptosis, Others, Influenza Virus

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