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Cat. No. Product Name Target Signaling Pathways
T6S0119 Dauricine

蝙蝠葛碱

Apoptosis; Others; NF-κB Apoptosis; NF-κB; Others
Dauricine 是存在于北豆根粉末中的一种双苯异喹啉生物碱,具有抗炎活性。它通过抑制NF-κB 激活,剂量依赖性地抑制结肠癌细胞的增值和侵袭,并诱导凋亡。
T3054 Daurisoline

蝙蝠葛苏林碱,(R,R)-Daurisoline

Others; Potassium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Others
Daurisoline ((R,R)-Daurisoline) 是一种 hERG 抑制剂,也是一种自噬阻滞剂。
T2S0118 Daurinoline

Calcium Channel; 5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a protective function on microcirculation of cerebral pia mater, which may be beneficial to relieve cerebral ischemic injury. Daurinoline could significantly reverse noradrenaline induced constriction of pial arterioles and venules, and increase the number of blood vessels which were decreased by noradrenaline.

天然产物

Dauricine
Cat.No: T6S0119
Synonym: 蝙蝠葛碱
Target: Apoptosis, Others, NF-κB
Daurisoline
Cat.No: T3054
Synonym: 蝙蝠葛苏林碱,(R,R)-Daurisoline
Target: Others, Potassium Channel, Autophagy
Daurinoline
Cat.No: T2S0118
Synonym:
Target: Calcium Channel, 5-HT Receptor, Histamine Receptor
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