Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6S0119 |
Dauricine
蝙蝠葛碱 |
Apoptosis; Others; NF-κB | Apoptosis; NF-κB; Others |
Dauricine 是存在于北豆根粉末中的一种双苯异喹啉生物碱,具有抗炎活性。它通过抑制NF-κB 激活,剂量依赖性地抑制结肠癌细胞的增值和侵袭,并诱导凋亡。 | |||
T3054 |
Daurisoline
蝙蝠葛苏林碱,(R,R)-Daurisoline |
Others; Potassium Channel; Autophagy | Autophagy; Membrane transporter/Ion channel; Others |
Daurisoline ((R,R)-Daurisoline) 是一种 hERG 抑制剂,也是一种自噬阻滞剂。 | |||
T2S0118 | Daurinoline | Calcium Channel; 5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a protective function on microcirculation of cerebral pia mater, which may be beneficial to relieve cerebral ischemic injury. Daurinoline could significantly reverse noradrenaline induced constriction of pial arterioles and venules, and increase the number of blood vessels which were decreased by noradrenaline. |