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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T25048 Algestone acetophenide

Neolutin,苯甲孕酮

Others Others
Algestone acetophenide (Neolutin) 是用于发情同步的孕酮,已被评估为与庚酸雌二醇联合使用的注射避孕药。它在治疗上也用作局部抗炎药,并在治疗痤疮时局部应用。
T0977 Medrysone

Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松

Glucocorticoid Receptor; Others Endocrinology/Hormones; Others
Medrysone (6α-Methyl-11β-hydroxyprogesterone) 是局部合成的糖皮质激素,具有代谢、抗炎和抗过敏特性,有潜力用于眼科的眼炎症研究。
T2597 Norgestrel

甲基炔诺酮,SH-850,FH 122-A,炔诺孕酮,WY-3707,SH-70850

Estrogen/progestogen Receptor; Reactive Oxygen Species Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
Norgestrel (WY-3707) 是一种孕酮的合成类似物,是一种口服避孕药中常见的化合物,也是一种神经保护性强抗氧化剂,能够防止光诱导的感光细胞中的ROS 的生成以及细胞死亡。
T9504 MAP4343

Microtubule Associated Cytoskeletal Signaling
MAP4343 是孕烯醇酮的 3-甲基醚衍生物。它在体外与微管相关蛋白 2 (MAP2) 结合并刺激微管蛋白聚合,从而增强神经突延伸和保护神经元免受神经毒剂的侵害。

化合物

Algestone acetophenide
Cat.No: T25048
Synonym: Neolutin,苯甲孕酮
Target: Others
Medrysone
Cat.No: T0977
Synonym: Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松
Target: Glucocorticoid Receptor, Others
Norgestrel
Cat.No: T2597
Synonym: 甲基炔诺酮,SH-850,FH 122-A,炔诺孕酮,WY-3707,SH-70850
Target: Estrogen/progestogen Receptor, Reactive Oxygen Species
MAP4343
Cat.No: T9504
Synonym:
Target: Microtubule Associated
Cat. No. Product Name Target Signaling Pathways
T5040 Medroxyprogesterone

甲羟孕酮,甲孕酮

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Medroxyprogesterone 是一种合成的人孕酮变体,是孕酮受体激动剂,用于治疗肾癌。在兽医实践中用作发情调节剂。
T1261 Medroxyprogesterone Acetate

Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
Medroxyprogesterone Acetate (Farlutin) 是广泛使用的合成类固醇,与雄激素,孕酮及糖皮质激素受体均有作用。
T16338 Norgestimate metabolite Norelgestromin

17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮

Drug Metabolite Metabolism
Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) 是norgestimate 的一种活性代谢物。它是用于避孕贴片的甾体孕激素,与雌激素乙炔雌二醇结合使用。
T1284 Megestrol acetate

SC10363,醋酸甲地孕酮,BDH1298

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。

天然产物

Medroxyprogesterone
Cat.No: T5040
Synonym: 甲羟孕酮,甲孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Medroxyprogesterone Acetate
Cat.No: T1261
Synonym: Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, Endogenous Metabolite
Norgestimate metabolite Norelgestromin
Cat.No: T16338
Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮
Target: Drug Metabolite
Megestrol acetate
Cat.No: T1284
Synonym: SC10363,醋酸甲地孕酮,BDH1298
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy
TargetMol Loading
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