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Cat. No. Product Name Target Signaling Pathways
TQ0118 Britannilactone

Desacetylinulicin,旋覆花内酯

Others Others
Britannilactone, extracted from the dried flower of Inula britannica L, significantly reduces melanin production in a dose-dependent manner (IC50: 15.5 uM).
TQ0169 Inulicin

1-O-Acetylbritannilactone,旋覆花内酯

FAK; NF-κB; COX; Src Angiogenesis; Cytoskeletal Signaling; Immunology/Inflammation; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors
Inulicin (1-O-Acetylbritannilactone) 是从欧亚旋覆花中提取的一种天然产物,可抑制 VEGF 介导的Src 和FAK 活化,抑制NF-κB 活化和易位,以及抑制 LPS 诱导的PGE2产生和COX-2表达。
T5793 Britannin

Apoptosis; AMPK; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Britannin 是分离于旋覆花的一种倍半萜内酯,可通过激活由 ROS 调节的 AMPK 来诱导肝癌细胞凋亡和自噬,具有抗增殖和抗炎活性。
TN1143 1-O-Acetyl britannilactone

NF-κB; COX Immunology/Inflammation; Neuroscience; NF-κB
1-O-Acetyl britannilactone shows antifungal, and anti-cancer activities, it suppresses angiogenesis and lung cancer cell growth possibly via regulating the VEGFR-Src-FAK signaling.
T75678 Tomentosin

Apoptosis Apoptosis
Tomentosin 是一种从里海旋覆花中提取出来倍半萜内酯,具有潜在的抗炎和抗癌活性,可促进胰腺癌细胞的凋亡并抑制增殖、迁移和侵袭。

天然产物

Britannilactone
Cat.No: TQ0118
Synonym: Desacetylinulicin,旋覆花内酯
Target: Others
Inulicin
Cat.No: TQ0169
Synonym: 1-O-Acetylbritannilactone,旋覆花内酯
Target: FAK, NF-κB, COX, Src
Britannin
Cat.No: T5793
Synonym:
Target: Apoptosis, AMPK, Autophagy
1-O-Acetyl britannilactone
Cat.No: TN1143
Synonym:
Target: NF-κB, COX
Tomentosin
Cat.No: T75678
Synonym:
Target: Apoptosis
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