4
11
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1432 |
Phenylbutazone
Butazolidine,保泰松 |
COX | Immunology/Inflammation; Neuroscience |
Phenylbutazone (Butazolidine) 是是非甾体类抗炎药,前列腺素 H 合酶过氧化物酶的还原辅助因子,可诱导肌肉盲样蛋白 1 表达,有用于强直性脊柱炎的研究潜力。 | |||
T0435 |
Sulfinpyrazone
(+/-)-Sulfinpyrazone,G-28315,苯磺保泰松,NSC 75925 |
COX | Immunology/Inflammation; Neuroscience |
Sulfinpyrazone (NSC-75925) 是一种口服有效的尿酸剂,具有抗血栓和血小板抑制作用。它可作用于慢性和间歇性痛风性关节炎。 | |||
T7710 |
MOFEBUTAZONE
|
Others | Others |
Mofebutazone 抑制前列腺素和白三烯的免疫释放。 | |||
T72177 |
Oxyphenbutazone monohydrate
羟布宗一水合物 |
||
Oxyphenbutazone monohydrate 是一种保泰松 (Phenylbutazone) 代谢物,具有抗炎作用。Oxyphenbutazone monohydrate 是一种具有口服活性的非选择性 COX 抑制剂。Oxyphenbutazone monohydrate 能选择性地杀死不复制的结核分枝杆菌 (Mycobaterium tuberculosis)。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2858 |
Baicalein
5,6,7-Trihydroxyflavone,黄芩素,黄芩黄素 |
Ferroptosis; Influenza Virus; ROS; Xanthine Oxidase | Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology |
Baicalein (5,6,7-Trihydroxyflavone) 是一种黄嘌呤氧化酶抑制剂,其IC50值为 3.12 μM。 | |||
T3S1866 |
Propyl gallate
没食子酸丙酯;3,4,5-三羟基苯甲酸丙酯、倍酸丙酯、五倍子酸丙酯,Tenox PG,没食子酸丙酯,n-Propyl gallate,Gallic acid propyl esterZ |
Antioxidant | oxidation-reduction |
Propyl gallate (Gallic acid propyl esterZ) 是常见的食品抗氧化剂。它能阻碍乙二醛、丙烯醛、甲基乙二醛的生成。 | |||
T22974 |
Methyl 2,5-dihydroxycinnamate
|
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Methyl 2,5-dihydroxycinnamate 是 erbstatin 类似物,是一种高效、稳定的 EGF 受体相关酪氨酸激酶的抑制剂。 | |||
T0311 |
Salicyl alcohol
α,2-Toluenediol,o-Methylolphenol,2-Hydroxybenzyl alcohol,水杨醇,邻羟基苄醇,Saligenin,Saligenol,Diathesin |
Others | Others |
Salicyl alcohol (2-Hydroxybenzyl alcohol) 是一种医药、香料、农药的合成中间体。 | |||
T3768 |
Epifriedelanol
表木栓醇,Epifriedelinol |
Others | Others |
Epifriedelanol (Epifriedelinol) 是一种分离自 Ulmus davidiana 根皮中的三萜类化合物,具有抗肿瘤作用,可以减缓人原始细胞的衰老。 | |||
T3S2152 |
23-Hydroxybetulinic acid
Anemosapogenin,23-羟基白桦酸 |
Others | Others |
23-Hydroxybetulinic acid (Anemosapogenin) 是一种具有抗癌作用的生物化合物。 | |||
T3871 |
Daucosterol
Alexandrin,Sitogluside,β-Sitosterol β-D-glucoside,Eleutheroside A,西托糖苷 |
Glucosidase | Metabolism |
Daucosterol (Sitogluside) 是天然的甾醇体类化合物。 | |||
T3794 |
Pentagalloylglucose
Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖 |
Influenza Virus | Microbiology/Virology |
1,2,3,4,6-O-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) 存在于多种植物中,具有重要的药理作用。Pentagalloylglucose 表现出显著的抗狂犬病病毒 (RABV) 活性。 | |||
TN2036 |
Paeonilactone B
(+)-Paeonilactone B |
NADPH-oxidase | Immunology/Inflammation |
Paeonilactone B ((+)-Paeonilactone B) 是一种来自白芍的单萜类化合物,具有神经保护活性,抑制氧化应激,在大鼠皮质细胞在抑制 H2O2 诱导的神经毒性。 | |||
TN1203 |
2,3,8-Tri-O-methylellagic acid
2,3,8-三邻甲基鞣花酸 |
Antifection | Microbiology/Virology |
2,3,8-tri-O-Methyl ellagic acid has antimicrobial activity agaist Vibro cholera, Staphylococcus aureus, Klebsiella pneumoniae, Pseudomonas aeruginosa, Bacillus cereus, Escherichia coli. | |||
TN1062 |
Peonidin chloride
|
ERK; COX | Immunology/Inflammation; MAPK; Neuroscience |
Peonidin chloride has antioxidant activity. Peonidin has show potent inhibitory and apoptotic effects on cancer cells in vitro, notably metastatic human breast cancer cells. |