首页工具

登录

搜索结果

Search Results for " urotensin "

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
TP2165	Urotensin II, mouse acetate (9047-55-6 free base) Urotensin II, mouse acetate	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II, mouse acetate (9047-55-6 free base) 是孤儿 GPR14 或 SENR 的内源性配体。它是一种强效血管收缩剂。
T37527L	[Orn8]-Urotensin II acetate	GPR	Endocrinology/Hormones; GPCR/G Protein
	[Orn8]-Urotensin II acetate 是一种 Urotensin 受体配体和 Urotensin 受体的部分激动剂。
TP1737L	Urotensin II (114-124), human acetate Urotensin II (114-124), human acetate(251293-28-4 free base)	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II (114-124), human acetate(251293-28-4 free base) 是一种 11 个氨基酸残基肽，是一种有效的血管收缩剂和孤儿受体 GPR14 的激动剂。
TP1199L	Urotensin I acetate (83930-33-0 Free base)	CRFR	GPCR/G Protein
	Urotensin I acetate 是一种 CRF 样神经肽，可作为 CRF 受体激动剂，对 CHO 细胞中的人 CRF1、人 CRF2 和大鼠 CRF2α 受体的 pEC50 分别为 11.46、9.36 和 9.85，对 CHO 细胞的 Kis 分别为 0.4、1.8 和 5.7 nM hCRF1、rCRF2α 和 mCRF2β 受体分别为。
T37527	[Orn8]-Urotensin II [Orn8]-Urotensin II

TP1199	Urotensin I Catostomus urotensin I
	Urotensin I is, 41-aa neuropeptide, acts as an agonist of CRF receptor with pEC50s of 11.46, 9.36 and 9.85 for human CRF1, human CRF2 and rat CRF2α receptors in CHO cells, and Kis of 0.4, 1.8, and 5.7 nM for hCRF1, rCRF2α and mCRF2β receptors, respectivel
T36483	Urotensin II-related peptide
	Urotensin II-related peptide 是人尾加压素 II 类似物。Urotensin II-related peptide 与 UT 受体具有高亲和力。
TP2166	Urotensin II, mouse TFA (9047-55-6 free base) Urotensin II, mouse TFA	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.
T36729	Urotensin II (goby) (trifluoroacetate salt)
	Urotensin II is a peptide vasoconstrictor and agonist of the urotensin (UT) receptor (Ki= 2.06 nM for the human recombinant receptor expressed in HEK293 cells).1It stimulates intracellular calcium mobilization in HEK293 cells expressing human and rat UT (EC50s = 0.47 and 0.78 nM, respectively) but decreases intracellular calcium concentration in goby (G. mirabilis) enterocytes when used at a concentration of 500 nM.2Urotensin II (20 mU/ml) stimulates active sodium and chloride absorption across ...
TP1816	Urotensin II, mouse
	Jump to search UTS2 Identifiers Aliases UTS2, PRO1068, U-II, UCN2, UII, urotensin 2 External IDs OMIM: 604097 MGI: 1346329 HomoloGene: 4939 GeneCards: UTS2 hide Gene location (Human) Chr. Chromosome 1 (human)[1] Band 1p36.23 Start 7,843,083 bp[1] En
TP1737	Urotensin II (114-124), human
	Urotensin II (114-124), human, is an 11-amino acid residue peptide that exhibits strong vasoconstrictor activity and acts as an agonist for the orphan receptor GPR14.
TP1415	Urotensin II (114-124), human TFA
	Urotensin II (114-124), human TFA, is an 11-amino acid residue peptide with a strong vasoconstrictor effect. This compound acts as an agonist for the orphan receptor GPR14.
T2058	Palosuran ACT-058362	GPR	Endocrinology/Hormones; GPCR/G Protein
	Palosuran (ACT-058362) 是人类 UT 受体的新型强效特异性拮抗剂，对表达人重组受体的 CHO 细胞膜的IC50值为 3.6 nM。它可改善糖尿病大鼠的胰腺和肾脏功能。
T75976	Urotensin I TFA
	Urotensin I (Catostomus urotensin I) TFA 是一种类 CRF 样肽，可作为 CRF 受体激动剂，在细胞实验中，对人 CRF1，CRF2和大鼠 CRF2α受体的 pEC50值分别为 11.46，9.36 和 9.85，对 hCRF1，rCRF2α和 mCRF2β受体的 Ki 值分别为 0.4，1.8 和 5.7 nM。
T23323	SB 611812	Neurotensin Receptor	GPCR/G Protein
	SB 611812 是 urotensin-II (UT) 的拮抗剂，可用于心血管疾病治疗的研究。
T75962	Urotensin II, mouse acetate
	Urotensin II, mouse acetate，是孤儿G蛋白偶联受体（GPR14或SENR）的一种内源性配体，具有显著的血管收缩活性并在中枢神经系统中发挥重要功能。
T75961	Urotensin II, mouse TFA
	Urotensin II, mouse TFA 为孤儿G蛋白偶联受体GPR14或SENR的内源性配体，具有强效血管收缩作用，并在中枢神经系统中发挥重要角色。
T38807L	[Lys8, Lys9]-Neurotensin (8-13) acetate	Neurotensin Receptor	GPCR/G Protein
	[Lys8, Lys9]-Neurotensin (8-13) acetate 是一种神经降压素类似物，通过激活 G 蛋白偶联受体 NTS1 和 NTS2 发挥镇痛作用，hNTS1 和 hNTS2 受体的 Ki 值分别为 0.33 nM 和 0.95 nM。
T7617L	Neurotensin(8-13) 3TFA(60482-95-3(free base))	Neurotensin Receptor	GPCR/G Protein
	Neurotensin(8-13) 3TFA(60482-95-3(free base)) 是神经降压素 (NT) 片段，神经降压素 (8-13) 导致细胞表面 NT1 受体 (NTR1) 密度降低。
TP2309	NEUROTENSIN TFA (39379-15-2 free base) Pyr-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH TFA（55508-42-4 free base),NEUROTENSIN TFA,神经加压素	Others	Others
	Neurotensin TFA (39379-15-2 free base) 是一种内源性 13 个氨基酸的神经肽，具有显着的阿片类非依赖性镇痛作用。它在大脑中充当神经递质，在肠道中充当激素，也充当神经调节剂。由于它与多种神经递质系统如多巴胺能、血清素能、谷氨酸能、GABA 能和胆碱能系统。它具有作为人体代谢物、有丝分裂原、神经递质和创伤的作用。
TP1310	Neurotensin	Neurotensin Receptor	GPCR/G Protein
	Neurotensin 是一种 13 个氨基酸的神经肽，参与调节促黄体激素和催乳素的释放，并与多巴胺能系统有显着的相互作用。它作为细胞有丝分裂原，作用于各种结肠直肠癌和胰腺癌。
T7617	Neurotensin(8-13) 神经降压素(8-13),Neurotensin(8-13)(3TFA)	Neurotensin Receptor	GPCR/G Protein
	Neurotensin(8-13) 是神经降压素的活性片段，可导致细胞表面 NT1 受体 (NTR1) 密度降低。
T76572	Acetyl neurotensin (8-13)
	Acetyl neurotensin (8-13) 是神经降压素类似物，具有完全结合和药理活性。
T38807	[Lys8, Lys9]-Neurotensin (8-13) JMV438,[Lys8, Lys9]-Neurotensin (8-13)
	[Lys8, Lys9]-Neurotensin (8-13) (JMV438) is a Neurotensin analog that elicits analgesic effects by activating the G protein-coupled receptors NTS1 and NTS2. The compound has K i values of 0.33 nM and 0.95 nM for hNTS1 and hNTS2 receptors, respectively.
TP2393	Neurotensin-related hexapeptide Lant-6
	Neurotensin-related hexapeptide exists in retinal ganglion cells and in their central projections in pigeons and may be utilized as a neuroactive substance by the central terminals of numerous retinal ganglion cells in birds.
T33656	Neurotensin (1-6)
	Neurotensin (1-6) affects dopamine release from striatum.
T40850	[D-Trp11]-Neurotensin [D-Trp11]-Neurotensin
	[D-Trp11]-Neurotensin is a compound that functions as a selective antagonist of Neurotensin (NT) in perfused rat hearts, while exhibiting full agonist properties in guinea pig atria and rat stomach strips. Additionally, this compound can inhibit hypotension induced by NT.
T22476	(±)-AC 7954 hydrochloride	Neurotensin Receptor	GPCR/G Protein
	(±)-AC 7954 hydrochloride是一种urotensin-II (UT)受体激活剂。
T27328	FL104 FL-104,FL 104	GPR	Endocrinology/Hormones; GPCR/G Protein
	FL104是小分子urotensin II 受体的有效激动剂，pEC50=7.11。
TP2104L	UFP 803 acetate	Neurotensin Receptor	GPCR/G Protein
	UFP 803 acetate 是一种有效的 urotensin-II (UT) 受体配体。 UFP-803 显示较低残留激动剂的活性。
TP1928L1	[Orn5]-URP acetate [Orn5]-URP acetate(782485-03-4 free base)	GPR	Endocrinology/Hormones; GPCR/G Protein
	[Orn5]-URP acetate 是一种有效的选择性 Urotensin-II receptor (UT) 拮抗剂 (pEC50 = 7.24)。 [Orn5]-URP 没有激动剂活性。
TP2106L	Urantide acetate(669089-53-6 free base)	Neurotensin Receptor	GPCR/G Protein
	Urantide acetate(669089-53-6 free base) 是一种选择性和竞争性的 urotensin-II (UT) 受体拮抗剂 (pKB = 8.3)。体外阻断 hU-II 诱导的胸主动脉收缩。对去甲肾上腺素或内皮素 1 诱导的收缩或乙酰胆碱诱导的松弛没有影响。在钙动员测定（在表达 hUT 受体的 CHO 细胞中）中表现为部分激动剂。
T12848	SB-657510	Others; Neurotensin Receptor	GPCR/G Protein; Others
	SB-657510 是 urotensin II (UII) receptor (UT) 拮抗剂。对于人，猴，猫，大鼠和小鼠的UT 的 Ki 值分别为 61、17、30、65 和 56 nM。SB-657510 通过抑制 UII 诱导的人类血管内皮细胞中炎性介质，如粘附分子，使细胞因子和组织因子上调从而发挥抗炎作用。SB 657510对糖尿病小鼠模型中糖尿病相关动脉粥样硬化疾病具有治疗作用。
T23326	SB 706375	Others	Others
	urotensin-II (UT) receptor antagonist
T28692	SB-436811 SB 436811
	SB-436811 is an antagonist of human urotensin-II receptor.
T26542	AC-7954
	AC-7954 is a potent and efficacious agonist of urotensin II receptor.
T71642	GSK-1562590
	GSK-1562590 is a urotensin-II receptor antagonist.
T22815	GSK 1562590 hydrochloride	Others	Others
	urotensin II (UT) receptor antagonist
T27441	GSK 1440115 GSK1440115,GSK-1440115
	GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma.
T75827	UFP-803 TFA
	UFP-803 TFA 是有效的urotensin-II receptor (UT)配体。UFP-803 TFA 具有较低的残留激动剂活性，因此它可以作为研究UT 系统在生理学和病理学中作用的重要工具。
T75828	[Orn5]-URP TFA
	[Orn5]-URP TFA 为Urotensin-II receptor (UT) 的有效且选择性纯拮抗剂，具pEC50值7.24，未呈现激动剂活性。
TP1928	[Orn5]-URP
	Urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.
T29077	Urolinin nWWK-Tyr(3-NO2)-Abu
	Urolinin is a linear peptidic Urotensin-II Receptor Agonist with low nanomolar potency as well as improved metabolic stability. Urolinin is a hexameric UIIR agonist with an EC50 of 4.75 nM and a metabolic stability of 1319 min, 6.3-fold higher than wild-t
TP2106	Urantide
	Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behav
TP2104	UFP-803 UFP 803
	Urotensin-II (UT) receptor ligand; behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonizes U-II induced contractions in the rat
T36373	Urocortin II (mouse) (trifluoroacetate salt)
	Urocortin II is a neuropeptide hormone and member of the corticotropin-releasing factor (CRF) family which includes mammalian CRF , urocortin , urocortin III , frog sauvagine, and piscine urotensin I.1 Mouse urocortin II shares 34 and 42% sequence homology with rat CRF and urocortin . It is expressed in mouse paraventricular, supraoptic, and arcuate nuclei of the hypothalamus, the locus coeruleus, and in motor nuclei of the brainstem and spinal ventral horn. Urocortin II selectively binds to CRF...
T35814	Urocortin III (human) (trifluoroacetate salt)
	Urocortin III is a neuropeptide hormone and member of the corticotropin-releasing factor (CRF) family which includes mammalian CRF , urocortin , urocortin II , frog sauvagine, and piscine urotensin I.1 Human urocortin III shares 90, 40, 37, and 21% identity to mouse urocortin III , mouse urocortin II , human urocortin , and mouse urocortin, respectively. Urocortin III selectively binds to type 2 CRF receptors (Kis = 21.7, 13.5, and >100 nM for rat CRF2α, rat CRF2β, and human CRF1, respectively)....

化合物

Urotensin II, mouse acetate (9047-55-6 free base)

Cat.No: TP2165

Synonym: Urotensin II, mouse acetate

Target: GPR

[Orn8]-Urotensin II acetate

Cat.No: T37527L

Target: GPR

Urotensin II (114-124), human acetate

Cat.No: TP1737L

Synonym: Urotensin II (114-124), human acetate(251293-28-4 free base)

Target: GPR

Urotensin I acetate (83930-33-0 Free base)

Cat.No: TP1199L

Target: CRFR

[Orn8]-Urotensin II

Cat.No: T37527

Synonym: [Orn8]-Urotensin II

Cat.No: TP1199

Synonym: Catostomus urotensin I

Urotensin II-related peptide

Cat.No: T36483

Urotensin II, mouse TFA (9047-55-6 free base)

Cat.No: TP2166

Synonym: Urotensin II, mouse TFA

Target: GPR

Urotensin II (goby) (trifluoroacetate salt)

Cat.No: T36729

Urotensin II, mouse

Cat.No: TP1816

Urotensin II (114-124), human

Cat.No: TP1737

Urotensin II (114-124), human TFA

Cat.No: TP1415

Cat.No: T2058

Synonym: ACT-058362

Target: GPR

Urotensin I TFA

Cat.No: T75976

Cat.No: T23323

Target: Neurotensin Receptor

Urotensin II, mouse acetate

Cat.No: T75962

Urotensin II, mouse TFA

Cat.No: T75961

[Lys8, Lys9]-Neurotensin (8-13) acetate

Cat.No: T38807L

Target: Neurotensin Receptor

Neurotensin(8-13) 3TFA(60482-95-3(free base))

Cat.No: T7617L

Target: Neurotensin Receptor

NEUROTENSIN TFA (39379-15-2 free base)

Cat.No: TP2309

Synonym: Pyr-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH TFA（55508-42-4 free base),NEUROTENSIN TFA,神经加压素

Target: Others

Cat.No: TP1310

Target: Neurotensin Receptor

Neurotensin(8-13)

Cat.No: T7617

Synonym: 神经降压素(8-13),Neurotensin(8-13)(3TFA)

Target: Neurotensin Receptor

Acetyl neurotensin (8-13)

Cat.No: T76572

[Lys8, Lys9]-Neurotensin (8-13)

Cat.No: T38807

Synonym: JMV438,[Lys8, Lys9]-Neurotensin (8-13)

Neurotensin-related hexapeptide

Cat.No: TP2393

Synonym: Lant-6

Neurotensin (1-6)

Cat.No: T33656

[D-Trp11]-Neurotensin

Cat.No: T40850

Synonym: [D-Trp11]-Neurotensin

(±)-AC 7954 hydrochloride

Cat.No: T22476

Target: Neurotensin Receptor

Cat.No: T27328

Synonym: FL-104,FL 104

Target: GPR

UFP 803 acetate

Cat.No: TP2104L

Target: Neurotensin Receptor

[Orn5]-URP acetate

Cat.No: TP1928L1

Synonym: [Orn5]-URP acetate(782485-03-4 free base)

Target: GPR

Urantide acetate(669089-53-6 free base)

Cat.No: TP2106L

Target: Neurotensin Receptor

Cat.No: T12848

Target: Others, Neurotensin Receptor

Cat.No: T23326

Target: Others

Cat.No: T28692

Synonym: SB 436811

Cat.No: T26542

Cat.No: T71642

GSK 1562590 hydrochloride

Cat.No: T22815

Target: Others

Cat.No: T27441

Synonym: GSK1440115,GSK-1440115

Cat.No: T75827

Cat.No: T75828

Cat.No: TP1928

Cat.No: T29077

Synonym: nWWK-Tyr(3-NO2)-Abu

Cat.No: TP2106

Cat.No: TP2104

Synonym: UFP 803

Urocortin II (mouse) (trifluoroacetate salt)

Cat.No: T36373

Urocortin III (human) (trifluoroacetate salt)

Cat.No: T35814

我们的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved. 沪ICP备20019793号-4

沪公网安备 31010602006700号

沪公网安备 31010602006700号

TargetMol Loading

联系我们

电话：

400-820-0310

邮箱：

service@tsbiochem.com

QQ：

2881945090（终端用户）

2885109491（经销商）

经销：

终端：

地址：

上海市静安区江场三路238号8楼