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Cat. No. Product Name Target Signaling Pathways
T6079 NVP-ADW742

ADW742,ADW,GSK 552602A

Apoptosis; IGF-1R Apoptosis; Tyrosine Kinase/Adaptors
NVP-ADW742 (ADW) 是一种具有口服活性,选择性的IGF-1R 酪氨酸激酶抑制剂,IC50为 0.17 μM。它抑制胰岛素受体,IC50为 2.8 μM,在肿瘤细胞中诱导多效性抗增殖/促凋亡。
T3549 Avadomide

CC 122

Apoptosis; E1/E2/E3 Enzyme; Ligand for E3 Ligase Apoptosis; PROTAC; Ubiquitination
Avadomide (CC 122) 是口服有效的cereblon 调节剂,可以调节 cereblon E3 连接酶活性,诱导弥漫性大 B 细胞淋巴瘤细胞凋亡,具有抗肿瘤和免疫调节活性。
TP1658L Type A Allatostatin I acetate

Type A Allatostatin I acetate(123209-95-0 free base)

Others Others
Type A Allatostatin I acetate(123209-95-0 free base) 是一种十三肽。 Allatostatin 是多效性神经肽,用于抑制昆虫保幼激素的合成。
T21244 NSI-189 Phosphate

NSI189 Phosphate,NSI 189 Phosphate,NSI-189磷酸盐

Others Others
NSI-189 Phosphate 是一种新型神经源性分子,具有多效性,包括临床前研究中证明的抗抑郁、促认知、突触和神经营养活性。其抗抑郁活性不依赖于单胺。
TP1658 Type A Allatostatin I

Type A Allatostatin I is a tridecapeptide that falls under the category of pleiotropic neuropeptides. These neuropeptides are known for their ability to inhibit the synthesis of juvenile hormone in insects.
T40528 Oxytocin free acid

9-Deamidooxytocin

Oxytocin free acid, also known as 9-Deamidooxytocin, is an analog of oxytocin where the glycinamide residue at position 9 has been substituted with a glycine residue. Oxytocin, a pleiotropic peptide hormone, has wide-ranging implications for general health, adaptation, development, reproduction, and social behavior.
T26688 Avadomide HCl

Avadomide hydrochloride,CC122, Avadomide HCl,CC-122,CC 122 HCl

Avadomide is an orally available pleiotropic pathway modulator with potential antineoplastic activity. CC-122 mimics an interferon response and has antitumor activity in DLBCL CC-122 binds Cereblon (CRBN) and promotes degradation of Ikaros and Aiolos in d
T82882 Binetrakin

Binetrakin (Interleukin 4 (human)) 是一种多效性细胞因子,源自T淋巴细胞,具有影响包括B细胞和T细胞在内的多种细胞类型的能力。它促进Th0细胞向Th2细胞的分化,广泛应用于各类生物学研究。
T82060 Interleukin-6 fragment (human)

Interleukin-6 fragment (human) 是一种多效性细胞因子,由淋巴细胞及非淋巴细胞产生。该分子的编码基因位于人类第7号染色体,长度大约为5 kb。Interleukin-6 fragment (human) 在免疫响应、急性相应、炎症过程、癌症治疗及血液造血方面均有重要的潜在应用。

化合物

NVP-ADW742
Cat.No: T6079
Synonym: ADW742,ADW,GSK 552602A
Target: Apoptosis, IGF-1R
Avadomide
Cat.No: T3549
Synonym: CC 122
Target: Apoptosis, E1/E2/E3 Enzyme, Ligand for E3 Ligase
Type A Allatostatin I acetate
Cat.No: TP1658L
Synonym: Type A Allatostatin I acetate(123209-95-0 free base)
Target: Others
NSI-189 Phosphate
Cat.No: T21244
Synonym: NSI189 Phosphate,NSI 189 Phosphate,NSI-189磷酸盐
Target: Others
Type A Allatostatin I
Cat.No: TP1658
Synonym:
Target:
Oxytocin free acid
Cat.No: T40528
Synonym: 9-Deamidooxytocin
Target:
Avadomide HCl
Cat.No: T26688
Synonym: Avadomide hydrochloride,CC122, Avadomide HCl,CC-122,CC 122 HCl
Target:
Binetrakin
Cat.No: T82882
Synonym:
Target:
Interleukin-6 fragment (human)
Cat.No: T82060
Synonym:
Target:
TargetMol Loading
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