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Search Results for " parenteral "

17

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8134 Cefathiamidine

Antibacterial; Antibiotic Microbiology/Virology
Cefathiamidine 是一种头孢菌素抗菌剂,可研究由易感细菌引起的感染,还可用于呼吸道、肝脏、五官感觉、尿路感染以及心内膜炎和败血症的研究。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T20720 Norethisterone enanthate

NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564

Estrogen/progestogen Receptor Endocrinology/Hormones
Norethisterone enanthate (NSC-9564) 是一种口服有效的长效的孕激素。
T31806 Flovagatran

TGN 255

Thrombin Proteases/Proteasome
Flovagatran (TGN 255) 是一种具有口服活性和有效性的凝血酶和肠外直接因子 II 抑制剂。Flovagatran 可用于研究静脉血栓栓塞。
T22314 Doripenem

Antibacterial; Antibiotic Microbiology/Virology
Doripenem 是对革兰氏阳性菌、阴性菌和厌氧菌有效的β-内酰胺广谱抗生素。
T9284 Dexketoprofen trometamol

COX Immunology/Inflammation; Neuroscience
Dexketoprofen trometamol 是一种改良的非选择性 COX 抑制剂,起效迅速,可作为口服和非肠道制剂使用。
T40475 Ceftobiprole medocaril

BAL5788,头孢比普酯

Antibacterial Microbiology/Virology
Ceftobiprole medocaril (BAL5788) 是 Ceftobiprole 的前药。Ceftobiprole 是一种广谱的头孢菌素,对耐甲氧西林金黄色葡萄球菌具有活性。
T60254 Calcium glycerophosphate

Phosphorylase Metabolism
Calcium glycerophosphate(CaGP)是肠道碱性磷酸酶 F3 的抑制剂 (intestinal alkaline phosphatase F3)。Calcium glycerophosphate 可作为全肠外营养溶液中钙和磷的来源。
T9422 Fosciclopirox

CPX-POM

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Fosciclopirox (CPX-POM) 利用靶向γ-分泌酶,抑制尿路上皮癌的生长。静脉给药后,它选择性地将活性代谢物 Ciclopirox 递送至整个尿路。Ciclopirox 在许多实体和血液恶性肿瘤中显示出抗癌活性。
T28552 Ro 09-1428

Ro-09-1428

Ro 09-1428, a parenteral cephalosporin, has high antipseudomonal activity.
T31528 Disodium sebacate

Sebacic Acid Disodium Salt,Decanedioic Acid Disodium Salt,Disodium Decanedioate

Disodium sebacate is a 10-carbon-atom dicarboxylic acid, proposed as substrate for parenteral nutrition. It has low toxicity.
T22433 Sulopenem

CP-70429,硫培南

Others Others
Sulopenem, an orally active, potent inhibitor of beta-lactamase, is a parenteral penem antibiotic with broad-spectrum activities against Gram-negative and Gram-positive bacteria.
T20107 Ertapenem

Invanz,MK0826,MK-0826,MK 0826

Ertapenem is a parenteral carbapenem. It has a broad spectrum of antimicrobial activity. It is highly resistant to inactivation by a wide variety of beta-lactamases.
T75298 Cefotiam dihydrochloride hydrate

Cefotiam (SCE-963) dihydrochloride hydrate,一种肠外头孢菌素类抗生素,对革兰氏阳性菌和革兰氏阴性菌展示出广谱活性。
T38872 Antibacterial agent 47

Antibacterial Agent 47 demonstrates potent antibacterial activity as an adjunct therapy to parenteral antibiotic Ceftazidime. By effectively reducing the minimum inhibitory concentration (MIC) of Ceftazidime, Antibacterial Agent 47 acts as a highly promising antimicrobial agent, thereby enhancing the overall efficacy of the treatment.
T75297 Cefotiam

Cefotiam (SCE-963)为肠外使用的头孢菌素类广谱抗生素,对革兰氏阳性菌和革兰氏阴性菌均有效。
T72141 Ceftobiprole medocaril sodium

头孢比普酯钠盐,BAL5788 sodium

Ceftobiprole medocaril (BAL5788) sodium 是 Ceftobiprole 的胃肠外前药。Ceftobiprole 是一种非肠道吡咯烷酮头孢菌素。Ceftobiprole 是一种广谱头孢菌素,对甲氧西林 (MRSA) 和耐万古霉素葡萄球菌 (VRSA) 和耐青霉素链球菌具有高水平的体外活性。Ceftobiprole 也抑制革兰氏阳性和革兰氏阴性病原体。

化合物

Cefathiamidine
Cat.No: T8134
Synonym:
Target: Antibacterial, Antibiotic
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Norethisterone enanthate
Cat.No: T20720
Synonym: NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564
Target: Estrogen/progestogen Receptor
Flovagatran
Cat.No: T31806
Synonym: TGN 255
Target: Thrombin
Doripenem
Cat.No: T22314
Synonym:
Target: Antibacterial, Antibiotic
Dexketoprofen trometamol
Cat.No: T9284
Synonym:
Target: COX
Ceftobiprole medocaril
Cat.No: T40475
Synonym: BAL5788,头孢比普酯
Target: Antibacterial
Calcium glycerophosphate
Cat.No: T60254
Synonym:
Target: Phosphorylase
Fosciclopirox
Cat.No: T9422
Synonym: CPX-POM
Target: Gamma-secretase
Ro 09-1428
Cat.No: T28552
Synonym: Ro-09-1428
Target:
Disodium sebacate
Cat.No: T31528
Synonym: Sebacic Acid Disodium Salt,Decanedioic Acid Disodium Salt,Disodium Decanedioate
Target:
Sulopenem
Cat.No: T22433
Synonym: CP-70429,硫培南
Target: Others
Ertapenem
Cat.No: T20107
Synonym: Invanz,MK0826,MK-0826,MK 0826
Target:
Cefotiam dihydrochloride hydrate
Cat.No: T75298
Synonym:
Target:
Antibacterial agent 47
Cat.No: T38872
Synonym:
Target:
Cefotiam
Cat.No: T75297
Synonym:
Target:
Ceftobiprole medocaril sodium
Cat.No: T72141
Synonym: 头孢比普酯钠盐,BAL5788 sodium
Target:
Cat. No. Product Name Target Signaling Pathways
T0224 Meropenem

美罗培南,SM 7338

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Meropenem (SM 7338) 是一种具有广谱抗菌活性的碳青霉烯抗生素,对敏感和耐药的淋病奈瑟氏球菌,流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL,0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T0012 Cinchonine

LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁

Apoptosis; P-gp; Parasite Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Cinchonine (LA40221) 是金鸡纳树皮中的一种天然产物。它可激活内质网应激诱导的人肝癌细胞凋亡。它是一种酰胺类局部麻醉剂。
T25240 Chloramphenicol succinate

Paraxin succinate,Kemicetine succinate,CPSA

Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol.

天然产物

Meropenem
Cat.No: T0224
Synonym: 美罗培南,SM 7338
Target: Others, Antibacterial, Antibiotic
Cinchonine
Cat.No: T0012
Synonym: LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁
Target: Apoptosis, P-gp, Parasite
Chloramphenicol succinate
Cat.No: T25240
Synonym: Paraxin succinate,Kemicetine succinate,CPSA
Target:
TargetMol Loading
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