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17

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1078 Nucleoprotein (396-404)

Nucleoprotein 396-404,NP 396

Nucleoprotein (396-404) refers to a specific fragment within the lymphocytic choriomeningitis virus (LCMV). This fragment, also known as the H-2D(b)-restricted immunodominant epitope, has been identified as a significant component of the viral antigen. It can be utilized as a valuable molecular model for studying viral antigens.
TP1077 Nucleoprotein (118-126)

Nucleoprotein 118-126,NP(118-126)

Nucleoprotein (118-126),a fragment of Nucleoprotein, is a 9-aa peptide .
TP2150 Nucleoprotein (396-404) (TFA)

NP 396 TFA

Others Others
Nucleoprotein (396-404) TFA is the 396 to 404 fragment of the lymphocytic choriomeningitis virus (LCMV). It is the H-2D(b)-restricted immunodominant epitope used as a molecular model of viral antigen.
T7330 Nucleozin

[4-(2-氯-4-硝基苯基)-1-哌嗪基](5-甲基-3-苯基-4-异噁唑基)-甲酮

Influenza Virus Microbiology/Virology
Nucleozin 靶向流感 A 核蛋白,这是一种病毒复制所必需的多功能 RNA 结合蛋白。
T0849 Pyrimethamine

Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶

DHFR; Antifolate; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Pyrimethamine (Pirimecidan) 是一种二氢叶酸还原酶的竞争性抑制剂,用作抗疟药。
TP1527 CEF8, Influenza Virus NP (383-391)

CEF8, Influenza Virus NP 383-391

Others Others
CEF8, Influenza Virus NP (383-391) 是一种甲型流感病毒核蛋白,含有 383-391 残基,是甲型流感病毒核蛋白中重要的 HLA-B*2705 限制性表位,与细胞毒性 T 淋巴细胞介导的免疫逃逸有关。
TP1822L CEF6 acetate(913545-15-0 free base)

Influenza Virus Microbiology/Virology
CEF6 acetate(913545-15-0 free base) 是 HLA-B7限制性流感病毒核蛋白表位,属于 CEF 对照肽。 CEF 对照肽长度为 8-12 个氨基酸,其序列来自人类巨细胞病毒、爱泼斯坦-巴尔病毒和流感病毒。
T7353 RSV604

(S)-1-(2-Fluorophenyl)-3-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea

RSV Microbiology/Virology
RSV604 ((S)-1-(2-Fluorophenyl)-3-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea) 是一种呼吸道合胞病毒抑制剂,可与 RSV 核蛋白结合,靶向核衣壳蛋白的 Kd 值为 1.6 μM。它对 RSV A 和 B 亚型的众多临床分离株有亚微摩尔活性,EC50平均值为 0.8 μM。
T70864 BMS-883559

BMS-883559 is a novel inhibitor of the influenza nucleoprotein (INF-NP).
TP1646 Influenza NP (147-155)

Influenza NP 147-155

This peptide is a H-2Kd-restricted epitope from Influenza nucleoprotein (147-155).
TP1596 CEF7, Influenza Virus NP (380-388)

CEF7, Influenza Virus NP 380-388

HLA-B*08 restricted influenza virus nucleoprotein epitope.
TP1632 Influenza NP (147-155) (TFA)

This peptide is a H2-Db-restricted epitope from Influenza nucleoprotein (147-155).
TP1644 Influenza A NP(366-374) Strain A/PR/8/35

This peptide is an H2-Db-restricted epitope from the Influenza A/PR/8/34 nucleoprotein.
TP1822 CEF6

CEF6, a HLA-B7 restricted influenza virus nucleoprotein epitope, belongs to the CEF control peptides. The CEF control peptides are 8-12 amino acids in length, with sequences derived from the human cytomegalovirus, Epstein-Barr virus and influenza virus.
T35887 MBD

MBD, a novel fluorescent probe (7-(p-Methoxybenzylamino)-4-nitrobenz-2,1,3-oxadiazole), is utilized to study the conformation of protein and nucleoprotein. Its application is extended to bacterial ribosomes, as well as bovine trypsinogen and trypsin. MBD exhibits significant fluorescence when it binds to the hydrophobic region of macromolecules [1][2].
T83046 Anti-Influenza agent 5

Influenza Virus Microbiology/Virology
Anti-Influenza agent 5 (Compound IIB-2)为查耳酮类衍生物,具有抑制流感病毒核输出的活性。该化合物能有效抑制对Oseltamivir具有耐药性的病毒株,主要通过阻断流感病毒核蛋白输出作用来抑制病毒复制。
T82071 Influenza NP (311-325)

Influenza NP (311-325) 是具有生物活性的肽段,对应于流感病毒核蛋白(NP)的311至325氨基酸。作为MHC II类限制性表位,它用于研究宿主在感染期间的免疫响应。该肽能在细胞内细胞因子检测中诱导强烈的γ干扰素(IFN-γ)产生,但不激活小鼠CD8 T细胞。谷氨酰胺(Q)或谷氨酸(E)位于N端时,焦谷氨酰(pGlu)肽可自发形成。Q或E向pGlu的自然转化及其疏水性γ-内酰胺环在肽的胃肠道蛋白酶稳定性中可能起作用。焦谷氨酰肽作为常见肽的一部分,在HPLC分析中评估肽的纯度。

化合物

Nucleoprotein (396-404)
Cat.No: TP1078
Synonym: Nucleoprotein 396-404,NP 396
Target:
Nucleoprotein (118-126)
Cat.No: TP1077
Synonym: Nucleoprotein 118-126,NP(118-126)
Target:
Nucleoprotein (396-404) (TFA)
Cat.No: TP2150
Synonym: NP 396 TFA
Target: Others
Nucleozin
Cat.No: T7330
Synonym: [4-(2-氯-4-硝基苯基)-1-哌嗪基](5-甲基-3-苯基-4-异噁唑基)-甲酮
Target: Influenza Virus
Pyrimethamine
Cat.No: T0849
Synonym: Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶
Target: DHFR, Antifolate, Parasite
CEF8, Influenza Virus NP (383-391)
Cat.No: TP1527
Synonym: CEF8, Influenza Virus NP 383-391
Target: Others
CEF6 acetate(913545-15-0 free base)
Cat.No: TP1822L
Synonym:
Target: Influenza Virus
RSV604
Cat.No: T7353
Synonym: (S)-1-(2-Fluorophenyl)-3-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea
Target: RSV
BMS-883559
Cat.No: T70864
Synonym:
Target:
Influenza NP (147-155)
Cat.No: TP1646
Synonym: Influenza NP 147-155
Target:
CEF7, Influenza Virus NP (380-388)
Cat.No: TP1596
Synonym: CEF7, Influenza Virus NP 380-388
Target:
Influenza NP (147-155) (TFA)
Cat.No: TP1632
Synonym:
Target:
Influenza A NP(366-374) Strain A/PR/8/35
Cat.No: TP1644
Synonym:
Target:
CEF6
Cat.No: TP1822
Synonym:
Target:
MBD
Cat.No: T35887
Synonym:
Target:
Anti-Influenza agent 5
Cat.No: T83046
Synonym:
Target: Influenza Virus
Influenza NP (311-325)
Cat.No: T82071
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2331 Eleutheroside B1

刺五加苷B1

Influenza Virus Microbiology/Virology
Eleutheroside B1是具有广谱抗人流感病毒的一种香豆素。它抑制多种趋化因子基因和流感病毒核蛋白基因的 mRNA 表达。它具有抗病毒、抗流感和抗炎活性,且细胞毒性小。

天然产物

Eleutheroside B1
Cat.No: TN2331
Synonym: 刺五加苷B1
Target: Influenza Virus
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