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Cat. No. Product Name Target Signaling Pathways
T5354 IRAK4-IN-7

CA-4948

IRAK Immunology/Inflammation; NF-κB
IRAK4-IN-7 (CA-4948) 是白介素 1 受体相关激酶 4 (IRAK4) 的选择性抑制剂,口服有活性。它可用于研究癌症以及炎症疾病。
T9924 Obinutuzumab

奥滨尤妥珠单抗,Obinutuzumab/afutuzumab

Others Others
Obinutuzumab (Obinutuzumab/afutuzumab)/afutuzumab 是一种新型糖工程化 II 型 CD20单克隆抗体,用于研究非霍奇金淋巴瘤。
T8380 Bendamustine

SDX105,宾达氮芥

Apoptosis; Others; DNA Alkylator/Crosslinker Apoptosis; DNA Damage/DNA Repair; Others
Bendamustine (SDX105) 是一种嘌呤类似物,是一种 DNA 交联剂,具有烷基化、抗癌和抗代谢作用。它可激活 DNA 损伤反应和细胞凋亡。
T35617 Mitoguazone

MGBG,Methyl-GAG

Apoptosis; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Mitoguazone (Methyl-GAG) 是一种可透过血脑屏障的选择性的 S-腺苷-蛋氨酸脱羧酶 (S-adenosyl-methionine decarboxylase) 抑制剂,可破坏多胺的生物合成。Mitoguazone 是一种具有抗肿瘤活性的合成多羰基衍生物,可抑制 HIV DNA 整合到单核细胞和巨噬细胞中的细胞 DNA 中,诱导细胞凋亡 (apoptosis)。Mitoguazone 具可用于预防急性白血病,霍奇金淋巴瘤和非霍奇金淋巴瘤。
T76692 Mosunetuzumab

BTCT-4465A

Others Others
Mosunetuzumab (BTCT-4465A) 是一种基于免疫球蛋白 G1 且靶向 CD20 (B 细胞) 和 CD3 (T 细胞) 的人源化抗体。Mosunetuzumab 重定向 T 细胞以接合和消除恶性 B 细胞,可用于研究复发或难治性 (R/R) B 细胞非霍奇金淋巴瘤 (B-NHL)和难治性滤泡性淋巴瘤。
T78686 Apoptosis inducer 11

Apoptosis Apoptosis
Apoptosisinducer 11(compound 3u)通过线粒体途径引发细胞凋亡。在非霍奇金淋巴瘤细胞系中,该化合物导致G2/M期停滞和S期显著减少。
T40901 Aderbasib

INCB007839,INCB7839

Aderbasib (INCB007839) is a highly potent and orally active hydroxamate-based inhibitor of ADAM10 and ADAM17, with low nanomolar affinity. This compound demonstrates strong antineoplastic activity and holds potential for cancer research in various areas, such as diffuse large B-cell non-Hodgkin lymphoma, HER2-positive breast cancer, gliomas, and more.
T78331 Epcoritamab

GEN3013

Epcoritamab (GEN3013) 是一种双特异性IgG1抗体,它能够将 CD3的T细胞引导至CD20阳性的肿瘤细胞,实现T细胞与肿瘤细胞的靶向联系。
T76768 Pinatuzumab

Pinatuzumab为针对CD22细胞表面抗原的单克隆抗体。作为合成抗体活性分子偶联物(ADC)成分,适用于非霍奇金淋巴瘤(NHL)等多种疾病的研究。
T76765 Veltuzumab

Veltuzumab (IMMU-106) 为一种针对CD20的人源化单克隆抗体。其在Daudi细胞系中显示出较低的EC50值,范围为0.08-0.09 μg/mL。Veltuzumab适用于非霍奇金淋巴瘤(NHL)等癌症的研究。
T82078 Iladatuzumab

MCDS0593A

Iladatuzumab (MCDS0593A) 为人源化IgG1抗CD79B单克隆抗体。该抗体作为ADC活性分子Iladatuzumab vedotin (DCDS0780A) 的构建模块,Iladatuzumab vedotin 展现出治疗B细胞非霍奇金淋巴瘤 (B-NHL) 的研究潜力。
T68485 Apilimod HCl

Apilimod dimesylate is a potent and selective PIKfyve inhibitor. It exhibits no significant activity at other lipid kinases and protein kinases, including PIP4K, PIP5K, mTOR, PI3K and PI4K. Apilimod dimesylate inhibits cellular entry by SARS-CoV-2, MERS-CoV and MHV S pseudovirions. It reduces the number of SARS-CoV-2-infected hiPSC-derived pneumocyte-like cells by 85% and inhibits SARS-CoV-2 replication in donor lung tissue. It also exhibits selective cytotoxicity in B-cell non-Hodgkin lymphoma ...
T73700 Daunorubicin citrate

Daunorubicin citrate(Daunomycin citrate)作为一种拓扑异构酶 II(topoisomerase II)抑制剂,展现出有效的抗肿瘤活性,通过抑制 DNA 和 RNA 合成(DNA and RNA synthesis)发挥作用。作为一种细胞毒性药物,Daunorubicin citrate 能够抑制癌细胞活性,并诱导细胞凋亡(apoptosis)和坏死(necrosis),属于蒽环类抗生素范畴。该化合物广泛应用于包括白血病、非霍奇金淋巴瘤、尤文氏肉瘤、维尔姆斯氏瘤在内的多种癌症和感染研究领域。

化合物

IRAK4-IN-7
Cat.No: T5354
Synonym: CA-4948
Target: IRAK
Obinutuzumab
Cat.No: T9924
Synonym: 奥滨尤妥珠单抗,Obinutuzumab/afutuzumab
Target: Others
Bendamustine
Cat.No: T8380
Synonym: SDX105,宾达氮芥
Target: Apoptosis, Others, DNA Alkylator/Crosslinker
Mitoguazone
Cat.No: T35617
Synonym: MGBG,Methyl-GAG
Target: Apoptosis, HIV Protease
Mosunetuzumab
Cat.No: T76692
Synonym: BTCT-4465A
Target: Others
Apoptosis inducer 11
Cat.No: T78686
Synonym:
Target: Apoptosis
Aderbasib
Cat.No: T40901
Synonym: INCB007839,INCB7839
Target:
Epcoritamab
Cat.No: T78331
Synonym: GEN3013
Target:
Pinatuzumab
Cat.No: T76768
Synonym:
Target:
Veltuzumab
Cat.No: T76765
Synonym:
Target:
Iladatuzumab
Cat.No: T82078
Synonym: MCDS0593A
Target:
Apilimod HCl
Cat.No: T68485
Synonym:
Target:
Daunorubicin citrate
Cat.No: T73700
Synonym:
Target:
TargetMol Loading
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