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Search Results for " muscarinic m1 receptor binding "

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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6707 Tiotropium Bromide hydrate

BA-679 BR hydrate,BA 679BR,噻托溴铵一水合物

AChR Neuroscience
Tiotropium Bromide hydrate (BA-679 BR hydrate) 是长效的毒蕈碱受体拮抗剂,可用于治疗慢性阻塞性气道疾病 (COPD)。
T23265 RS 67333 hydrochloride

RS 67333 (hydrochloride),RS 67333 HCl,盐酸RS67333

5-HT Receptor GPCR/G Protein; Neuroscience
RS 67333 hydrochloride (RO5203648) 是一种有效的、选择性的5-HT4 受体 (5-HT4R) 部分激动剂,在豚鼠纹状体中的 pKi 为 8.7。RS 67333 hydrochloride 对其他几种受体的亲和力较低,包括 5-HT1A、5-HT1D、5-HT2A、5-HT2C、多巴胺 D1、D2 和毒蕈碱 M1-M3 受体。RS 67333 hydrochloride 具有神经保护作用,可用于阿尔茨海默病研究。
T38895 Zanapezil free base

TAK-147 free base,Zanapezil free base

Zanapezil (TAK-147) is a powerful and selective inhibitor of acetylcholine esterase (AChE). It demonstrates significant and reversible inhibition of AChE activity in rat cerebral cortex homogenates (IC50 = 51.2 nM). Furthermore, Zanapezil exhibits moderate inhibition of muscarinic M1 and M2 receptor binding with Ki values of 234 and 340 nM, respectively. This compound holds promise for the investigation of the initial stages of Alzheimer's disease (AD).
T16443 PCS1055 dihydrochloride

Others Others
PCS1055 dihydrochloride is an effective, selective, and competitive muscarinic M4 receptor antagonist (IC50: 18.1 nM and a Kd: 5.72 nM). PCS1055 dihydrochloride is also a potent AChE inhibitor (IC50 s: 22 nM and 120 nM for electric eel and human AChE, res

化合物

Tiotropium Bromide hydrate
Cat.No: T6707
Synonym: BA-679 BR hydrate,BA 679BR,噻托溴铵一水合物
Target: AChR
RS 67333 hydrochloride
Cat.No: T23265
Synonym: RS 67333 (hydrochloride),RS 67333 HCl,盐酸RS67333
Target: 5-HT Receptor
Zanapezil free base
Cat.No: T38895
Synonym: TAK-147 free base,Zanapezil free base
Target:
PCS1055 dihydrochloride
Cat.No: T16443
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1653 Fustin

ERK; Beta Amyloid; AChR MAPK; Neuroscience
Fustin 是植物漆树 (Rhus verniciflua Stokes) 的植物性黄烷醇成分。 Fustin 对 6-羟基多巴胺诱导的神经元细胞死亡具有保护作用。

天然产物

Fustin
Cat.No: TN1653
Synonym:
Target: ERK, Beta Amyloid, AChR
TargetMol Loading
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