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3

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T10809 CHPG

Others Others
CHPG is a selective agonist of mGluR5. In BV2 microglial cells, it attenuates SO2-induced oxidative stress and inflammation through the TSG-6/NF-κB pathway.
T10809L CHPG hydrochloride

CHPG hydrochloride(170846-74-9 Free base)

ERK; NF-κB; GluR MAPK; Neuroscience; NF-κB
CHPG hydrochloride 是 mGluR5 的选择性激动剂。
T10808 CHPG sodium salt

NF-κB; GluR Neuroscience; NF-κB
CHPG sodium salt 是 mGluR5 的选择性激动剂,可激活 ERK 和 Akt 信号通路。 CHPG 钠盐可用于创伤性脑损伤的研究。

化合物

CHPG
Cat.No: T10809
Synonym:
Target: Others
CHPG hydrochloride
Cat.No: T10809L
Synonym: CHPG hydrochloride(170846-74-9 Free base)
Target: ERK, NF-κB, GluR
CHPG sodium salt
Cat.No: T10808
Synonym:
Target: NF-κB, GluR
Cat. No. Product Name Target Signaling Pathways
TN6714 Geranylgeraniol

FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095

Apoptosis Apoptosis
Geranylgeraniol (FT0626663) 是一种类异戊二烯,存在于水果、蔬菜和谷物中,包括大米。 Geranylgeraniol (FT0626663) 抑制生长并诱导各种肿瘤细胞的凋亡。 Geranylgeraniol (FT0626663) 保护单核细胞免受他汀类药物诱导的细胞毒性并抑制分枝杆菌的生长。
T82211 Herpotrichone B

Herpotrichone B exhibits potent anti-neuroinflammatory activity in BV-2 microglial cells induced by lipopolysaccharide (LPS), with a half-maximal inhibitory concentration (IC50) of 0.11μM.
TN5248 Voleneol

NOS; COX; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
1β,6α-Dihydroxyeudesm-4(15)-ene (Voleneol,DE) can attenuate the lipopolysaccharide (LPS)-induced inflammation in BV2 microglial cells, it also can dose-dependently suppress the protein expression of inducible nitric oxide synthase (iNOS) and cyclooxygenas

天然产物

Geranylgeraniol
Cat.No: TN6714
Synonym: FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095
Target: Apoptosis
Herpotrichone B
Cat.No: T82211
Synonym:
Target:
Voleneol
Cat.No: TN5248
Synonym:
Target: NOS, COX, Prostaglandin Receptor
TargetMol Loading
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