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Cat. No. Product Name Target Signaling Pathways
T21419 Diphenhydramine

苯海拉明,Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenhydramine (Syntedril) 是第一代具有抗胆碱能作用的H1 受体拮抗剂,它能透过血脑屏障。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T0059 Diphenylpyraline hydrochloride

盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。
T21390 Fexofenadine

Carboxyterfenadine,Telfast,非索非那定,MDL 16.455,Allegra

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fexofenadine (Carboxyterfenadine) 是一种抗组胺药物,用于治疗过敏症状,如鼻塞、花粉热和荨麻疹。与第一代抗组胺药相比,它通过血脑屏障并引起镇静的能力较差。
T1553 Chlorpheniramine maleate

马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Chlorpheniramine maleate (NCI-C55265) 是一种组胺 H1 拮抗剂,IC50为12 nM,用于过敏反应、花粉热、鼻炎、荨麻疹和哮喘。
T0785 Dexchlorpheniramine Maleate

S-(+)-Chlorpheniramine maleate salt,右泛醇,马来酸右氯苯那敏

Dopamine Receptor; 5-HT Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Dexchlorpheniramine Maleate (S-(+)-Chlorpheniramine maleate salt) 是一种具有抗胆碱能特性的抗组胺药,用于治疗花粉热或荨麻疹等过敏性疾病。
T0118 Mizolastine

SL 850324,咪唑司汀,咪唑斯汀

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mizolastine (SL 850324) 是组胺 H1 受体拮抗剂,IC50为 47 nM。它用于治疗过敏反应,如花粉热和荨麻疹等。
T4563 Thonzylamine

neohetramine,松齐拉敏

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂,具有抗组胺和抗过敏特性,可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。
T75276 Dexbrompheniramine

Dexbrompheniramine为口服活性H1受体拮抗剂(H1 receptor),具有抗组胺药属性,能够减轻天然化学组胺的作用。该化合物适用于花粉热与荨麻疹的研究。
T22983 Mizolastine dihydrochloride

Others Others
Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM). It also used in the treatment of hay fever, hives, and other allergic reactions.
T21247 Carbinoxamine

Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine

Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist.
T31396 Dexbrompheniramine maleate

D-Brompheniramine,Brompheniramine d-,Dexbrompheniraminum,Disophrol,Drixoral

Dexbrompheniramine is an antihistamine with anticholinergic properties. It is used to treat allergic diseases such as hay fever or urticaria. It can compete with histamine for H1 receptor sites on effector cells of the gastrointestinal tract, blood vessel
T69491 (E/Z)-Ensifentrine

(E/Z)-Ensifentrine is a potent and selective PDE3/4 inhibitor. (E/Z)-Ensifentrine acts as a long-acting inhibitor of the phosphodiesterase enzymes PDE-3 and PDE-4, producing both bronchodilator and antiinflammatory effects. It is being developed by Verona Pharma as a potential treatment for asthma and hay fever, and is currently in clinical trials.

化合物

Diphenhydramine
Cat.No: T21419
Synonym: 苯海拉明,Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255
Target: Histamine Receptor
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Diphenylpyraline hydrochloride
Cat.No: T0059
Synonym: 盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride
Target: Histamine Receptor
Fexofenadine
Cat.No: T21390
Synonym: Carboxyterfenadine,Telfast,非索非那定,MDL 16.455,Allegra
Target: Histamine Receptor
Chlorpheniramine maleate
Cat.No: T1553
Synonym: 马来酸氯苯那敏,NCI-C55265,Chlorphenamine maleate
Target: Histamine Receptor
Dexchlorpheniramine Maleate
Cat.No: T0785
Synonym: S-(+)-Chlorpheniramine maleate salt,右泛醇,马来酸右氯苯那敏
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine, Histamine Receptor
Mizolastine
Cat.No: T0118
Synonym: SL 850324,咪唑司汀,咪唑斯汀
Target: Histamine Receptor
Thonzylamine
Cat.No: T4563
Synonym: neohetramine,松齐拉敏
Target: Histamine Receptor
Dexbrompheniramine
Cat.No: T75276
Synonym:
Target:
Mizolastine dihydrochloride
Cat.No: T22983
Synonym:
Target: Others
Carbinoxamine
Cat.No: T21247
Synonym: Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine
Target:
Dexbrompheniramine maleate
Cat.No: T31396
Synonym: D-Brompheniramine,Brompheniramine d-,Dexbrompheniraminum,Disophrol,Drixoral
Target:
(E/Z)-Ensifentrine
Cat.No: T69491
Synonym:
Target:
TargetMol Loading
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