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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T8720	PRX-07034 hydrochloride PRX-07034	5-HT Receptor	GPCR/G Protein; Neuroscience
	PRX-07034 hydrochloride 是一种有效的高度选择性5-HT6受体拮抗剂，Ki 为 4-8 nM，IC50为 19 nM，可用于增强工作记忆和认知灵活性的研究。
T13995	1-Methyl-7-nitroisatoic anhydride 1M7	Others	Others
	1-Methyl-7-nitroisatoic anhydride (1M7) 是一种能够检测局部核苷酸的试剂。
T17906	Pomalidomide-amido-C4-amido-PEG2-C2-NH-Boc E3 Ligase Ligand-Linker Conjugates 53,Cereblon Ligand-Linker Conjugates 20	Others	Others
	Pomalidomide-amido-C4-amido-PEG2-C2-NH-Boc is a novel synthesized conjugate compound functioning as an E3 ligase ligand-linker in PROTAC technology. This compound incorporates a Pomalidomide-derived cereblon ligand, which binds selectively to the E3 ligase cereblon, and a 2-unit PEG linker, which provides stability and flexibility to the conjugate.
T74011	Mono(5-carboxy-2-ethylpentyl) phthalate
	Mono(5-carboxy-2-ethylpentyl) phthalate (MECPP)是Di-(2-ethylhexyl) phthalate (DEHP)的一种代谢产物，后者为硬质聚氯乙烯(PVC)中添加的主要增塑剂，以提升其柔韧性、耐温性、光学透明性、强度和抗扭结性。
T14593	Biotin-PEG3-Mal	Others	Others
	Biotin-PEG3-Mal is a biotinylated polyethylene glycol (PEG) derivative used as a linker in the synthesis of proteolysis targeting chimeras (PROTACs). By introducing the biotin moiety, it enables specific recognition and binding to target proteins. Additionally, the PEG spacer contributes to improved solubility and flexibility of the linker. This compound offers a valuable tool for constructing PROTACs, which hold great potential in targeted protein degradation strategies[1].
T62756	LY487379
	LY487379是一种选择性的人类 mGluR2 阳性异生调节剂（PAM）。LY487379 可提高谷氨酸刺激的 [35 S] GTPγS 结合，作用于 mGlu2 受体 (EC50: 1.7 μM) 和 mGlu3 受体 (EC50>10 μM)。LY487379 在大鼠模型中促使认知的灵活性，并诱导行为抑制。LY487379 能够用于研究精神分裂症。
T17331	(2-pyridyldithio)-PEG4 acid	Others	Others
	(2-Pyridyldithio)-PEG4 acid is a four-unit cleavable polyethylene glycol (PEG) linker specifically designed for the synthesis of antibody-drug conjugates (ADCs)[1]. It serves as a crucial component in the conjugation of antibodies and drugs, enabling targeted drug delivery and enhanced therapeutic efficacy. This linker possesses a (2-pyridyldithio) group at one end, facilitating the attachment of the linker to the specific site on the antibody molecule. The PEG4 chain provides the necessary flex...

化合物

PRX-07034 hydrochloride

Cat.No: T8720

Synonym: PRX-07034

Target: 5-HT Receptor

1-Methyl-7-nitroisatoic anhydride

Cat.No: T13995

Synonym: 1M7

Target: Others

Pomalidomide-amido-C4-amido-PEG2-C2-NH-Boc

Cat.No: T17906

Synonym: E3 Ligase Ligand-Linker Conjugates 53,Cereblon Ligand-Linker Conjugates 20

Target: Others

Mono(5-carboxy-2-ethylpentyl) phthalate

(2-pyridyldithio)-PEG4 acid

Cat.No: T17331

Synonym:

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T4797	DEHP Bis(2-ethylhexyl) phthalate,邻苯二甲酸二(2-乙基己)酯	Others; Endogenous Metabolite	Metabolism; Others
	DEHP (Bis(2-ethylhexyl) phthalate) 是内源性代谢产物的一种。
T0070	Pentoxifylline Oxpentifylline,PTX,己酮可可碱,BL-191	HIV Protease; PDE; Adenosine Receptor; Autophagy	Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂，具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。

天然产物

DEHP

Cat.No: T4797

Synonym: Bis(2-ethylhexyl) phthalate,邻苯二甲酸二(2-乙基己)酯

Target: Others, Endogenous Metabolite

Pentoxifylline

Cat.No: T0070

Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191

Target: HIV Protease, PDE, Adenosine Receptor, Autophagy

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