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Targets Recommended: Apoptosis HDAC

19

抑制剂 & 化合物

7

天然产物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T1888 Tacedinaline

Acetyldinaline,N-acetyldinaline,PD-123654,CI994,Goe-5549

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Tacedinaline (CI994) 是一种组蛋白脱乙酰酶抑制剂,抑制重组 HDAC 1, 2 和 3 的IC50值分别为 0.9,0.9,1.2 μM。
T1912 Dinaciclib

SCH 727965,PS-095760

Apoptosis; CDK Apoptosis; Cell Cycle/Checkpoint
Dinaciclib (SCH 727965) 是一种 CDK 抑制剂,抑制 CDK1、CDK2、CDK5 和 CDK9 (IC50=3/1/1/4 nM),具有选择性。Dinaciclib 具有潜在的抗肿瘤活性,可以抑制胸甘 (dThd) DNA 的整合。
T9256 N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine

Serine/threonin kinase; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine 是一种新型 2,6-naphthyridine,通过高通量筛选 (HTS) 鉴定为双蛋白激酶C/D (PKC/PKD) 抑制剂。
T5863 Indinavir sulfate

L735524 sulfate,MK-639 sulfate,硫酸茚地那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Indinavir sulfate (L735524 sulfate) 是一种 HIV 蛋白酶抑制剂。它抑制 HIV-1 蛋白酶,IC50 值为 0.41 nM,Ki 值为 0.24 nM。它也是SARS-CoV 3CLpro 抑制剂,IC50为 1.71 μM。
T3937 Methyl L-histidinate dihydrochloride

L-Histidine methyl ester dihydrochloride,L-组氨酸甲酯二盐酸盐

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
Methyl L-histidinate dihydrochloride (L-Histidine methyl ester dihydrochloride) 在Sprague-Dawley 大鼠胃中组氨酸脱羧酶的抑制作用被评估为 14CO2 产生减少,活性值为 1.8 μM。
T64437 5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine

5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64437。
T38451 Clodinafop-propargyl

Clodinafop-propargyl, a prominent member of aryloxyphenoxy-propionate herbicides, is employed for postemergence management of annual grasses in cereals, such as Avena, Lolium, Setaria, Phalaris, and Alopecurus spp.
TNU0894 2,6-Dichloro-3-nitro-4-pyridinamine

Heterocyclic Compounds - Pyridines; Intermediates and Building Blocks - Electrophiles, Nucleophiles
T69475 Dinalbuphine sebacate

Dinalbuphine sebacate is a long-lasting prodrug of nalbuphine, acting as a moderate-efficacy partial agonist or antagonist of the μ-opioid receptor and as a high-efficacy partial agonist of the κ-opioid receptor.
T65991 (S)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine

(S)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65991。
T70166 Indinavir monohydrate

Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.
T69231 Dinapsoline

Dinapsoline is a drug developed for the treatment of Parkinson's disease, that acts as a selective full agonist at the dopamine D1 receptor.
T25535 Indinavir, threo-

Threo-indinavir,Indinavir sulfate specified impurity C

Indinavir, threo- is a protease inhibitor utilized as a component of highly active antiretroviral treatment to HIV/AIDS.
T29294 1-Acridinamine

1-Aminoakridin,1-Aminoacridine

1-Acridinamine is a biochemical.
T68376 Indinavir lactone

Indinavir lactone is a protease inhibitor used as a component of highly active antiretroviral therapy to treat HIV/AIDS.
T65992 (R)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine

(R)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65992。
T67268 (S)-(3,5-Dioxa-4-phosphacyclohepta[2,1-a;3,4-a']dinaphthalen-4-yl)-5H-dibenz[b,f]azepine

(S)-(3,5-Dioxa-4-phosphacyclohepta[2,1-a;3,4-a']dinaphthalen-4-yl)-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67268,CAS号为 942939-38-0。
T31154 Cypridina luciferin

Cypridina luciferin is a bioactive chemical.
T5863L Indinavir

茚地那韦,MK-639,L 735 524,Crixivan

Indinavir (IDV) is an inhibitor of protease that is used as part of highly active antiretroviral therapy for the treatment of HIV/AIDS.

化合物

Tacedinaline
Cat.No: T1888
Synonym: Acetyldinaline,N-acetyldinaline,PD-123654,CI994,Goe-5549
Target: Apoptosis, HDAC
Dinaciclib
Cat.No: T1912
Synonym: SCH 727965,PS-095760
Target: Apoptosis, CDK
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
Cat.No: T9256
Synonym:
Target: Serine/threonin kinase, PKC
Indinavir sulfate
Cat.No: T5863
Synonym: L735524 sulfate,MK-639 sulfate,硫酸茚地那韦
Target: SARS-CoV, HIV Protease
Methyl L-histidinate dihydrochloride
Cat.No: T3937
Synonym: L-Histidine methyl ester dihydrochloride,L-组氨酸甲酯二盐酸盐
Target: HDAC
5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine
Cat.No: T64437
Synonym:
Target:
Clodinafop-propargyl
Cat.No: T38451
Synonym:
Target:
2,6-Dichloro-3-nitro-4-pyridinamine
Cat.No: TNU0894
Synonym:
Target:
Dinalbuphine sebacate
Cat.No: T69475
Synonym:
Target:
(S)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine
Cat.No: T65991
Synonym:
Target:
Indinavir monohydrate
Cat.No: T70166
Synonym:
Target:
Dinapsoline
Cat.No: T69231
Synonym:
Target:
Indinavir, threo-
Cat.No: T25535
Synonym: Threo-indinavir,Indinavir sulfate specified impurity C
Target:
1-Acridinamine
Cat.No: T29294
Synonym: 1-Aminoakridin,1-Aminoacridine
Target:
Indinavir lactone
Cat.No: T68376
Synonym:
Target:
(R)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine
Cat.No: T65992
Synonym:
Target:
(S)-(3,5-Dioxa-4-phosphacyclohepta[2,1-a;3,4-a']dinaphthalen-4-yl)-5H-dibenz[b,f]azepine
Cat.No: T67268
Synonym:
Target:
Cypridina luciferin
Cat.No: T31154
Synonym:
Target:
Indinavir
Cat.No: T5863L
Synonym: 茚地那韦,MK-639,L 735 524,Crixivan
Target:
Cat. No. Product Name Target Signaling Pathways
TN7180 2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-

4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C

Others Others
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- (Meridianin C)是一种海洋来源的天然产物,存在于Aplidium meridianum。
TN6740 Emodinanthrone

大黄素蒽酮,Emodin anthranol,Emodin anthrone,emodinol

Others; Antibiotic Microbiology/Virology; Others
Emodinanthrone 是一种蒽醌类化合物,是大黄素的前体,具有抗生素活性。它抑制大肠杆菌膜囊泡中呼吸驱动的溶质转运。
TN5766 Nandinaside A

Nandinaside A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5766,CAS号为 1813517-23-5。
TN2916 3-Acetoxy-4,7(11)-cadinadien-8-one

Others Others
3-Acetoxy-4,7(11)-cadinadien-8-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2916,CAS号为 104975-02-2。
TN2488 1,3,5-Cadinatriene-3,8-diol

Others Others
1,3,5-Cadinatriene-3,8-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2488,CAS号为 941227-27-6。
TN3253 7alpha-Hydroxy-4,11-cadinadiene-3,8-dione

Others Others
7alpha-Hydroxy-4,11-cadinadiene-3,8-dione 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3253,CAS号为 1423809-64-6。
TN5365 10β-Hydroxycadina-4,11(13)-dien-12,8β-olide

10β-Hydroxycadina-4,11(13)-dien-12,8β-olide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5365,CAS号为 35001-23-1。

天然产物

2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-
Cat.No: TN7180
Synonym: 4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C
Target: Others
Emodinanthrone
Cat.No: TN6740
Synonym: 大黄素蒽酮,Emodin anthranol,Emodin anthrone,emodinol
Target: Others, Antibiotic
Nandinaside A
Cat.No: TN5766
Synonym:
Target:
3-Acetoxy-4,7(11)-cadinadien-8-one
Cat.No: TN2916
Synonym:
Target: Others
1,3,5-Cadinatriene-3,8-diol
Cat.No: TN2488
Synonym:
Target: Others
7alpha-Hydroxy-4,11-cadinadiene-3,8-dione
Cat.No: TN3253
Synonym:
Target: Others
10β-Hydroxycadina-4,11(13)-dien-12,8β-olide
Cat.No: TN5365
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-00613 DNA polymerase II Protein, E. coli, Recombinant (His & Myc)

DNA polymerase II,polB,dinA,Pol II

E. coli E. coli
Thought to be involved in DNA repair and/or mutagenesis. Its processivity is enhanced by the beta sliding clamp (dnaN) and clamp loader.

重组蛋白

DNA polymerase II Protein, E. coli, Recombinant (His & Myc)
Cat.No: TMPH-00613
Species: E. coli
Expression System: E. coli
TargetMol Loading
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