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Cat. No. | Product Name | Target | Signaling Pathways |
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T1888 |
Tacedinaline
Acetyldinaline,N-acetyldinaline,PD-123654,CI994,Goe-5549 |
Apoptosis; HDAC | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Tacedinaline (CI994) 是一种组蛋白脱乙酰酶抑制剂,抑制重组 HDAC 1, 2 和 3 的IC50值分别为 0.9,0.9,1.2 μM。 | |||
T1912 |
Dinaciclib
SCH 727965,PS-095760 |
Apoptosis; CDK | Apoptosis; Cell Cycle/Checkpoint |
Dinaciclib (SCH 727965) 是一种 CDK 抑制剂,抑制 CDK1、CDK2、CDK5 和 CDK9 (IC50=3/1/1/4 nM),具有选择性。Dinaciclib 具有潜在的抗肿瘤活性,可以抑制胸甘 (dThd) DNA 的整合。 | |||
T9256 |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
|
Serine/threonin kinase; PKC | Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine 是一种新型 2,6-naphthyridine,通过高通量筛选 (HTS) 鉴定为双蛋白激酶C/D (PKC/PKD) 抑制剂。 | |||
T5863 |
Indinavir sulfate
L735524 sulfate,MK-639 sulfate,硫酸茚地那韦 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Indinavir sulfate (L735524 sulfate) 是一种 HIV 蛋白酶抑制剂。它抑制 HIV-1 蛋白酶,IC50 值为 0.41 nM,Ki 值为 0.24 nM。它也是SARS-CoV 3CLpro 抑制剂,IC50为 1.71 μM。 | |||
T3937 |
Methyl L-histidinate dihydrochloride
L-Histidine methyl ester dihydrochloride,L-组氨酸甲酯二盐酸盐 |
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Methyl L-histidinate dihydrochloride (L-Histidine methyl ester dihydrochloride) 在Sprague-Dawley 大鼠胃中组氨酸脱羧酶的抑制作用被评估为 14CO2 产生减少,活性值为 1.8 μM。 | |||
T64437 | 5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine | ||
5-(11bR)-Dinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepin-4-yl-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64437。 | |||
T38451 |
Clodinafop-propargyl
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Clodinafop-propargyl, a prominent member of aryloxyphenoxy-propionate herbicides, is employed for postemergence management of annual grasses in cereals, such as Avena, Lolium, Setaria, Phalaris, and Alopecurus spp. | |||
TNU0894 |
2,6-Dichloro-3-nitro-4-pyridinamine
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Heterocyclic Compounds - Pyridines; Intermediates and Building Blocks - Electrophiles, Nucleophiles | |||
T69475 |
Dinalbuphine sebacate
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Dinalbuphine sebacate is a long-lasting prodrug of nalbuphine, acting as a moderate-efficacy partial agonist or antagonist of the μ-opioid receptor and as a high-efficacy partial agonist of the κ-opioid receptor. | |||
T65991 | (S)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine | ||
(S)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65991。 | |||
T70166 |
Indinavir monohydrate
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Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability. | |||
T69231 |
Dinapsoline
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Dinapsoline is a drug developed for the treatment of Parkinson's disease, that acts as a selective full agonist at the dopamine D1 receptor. | |||
T25535 |
Indinavir, threo-
Threo-indinavir,Indinavir sulfate specified impurity C |
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Indinavir, threo- is a protease inhibitor utilized as a component of highly active antiretroviral treatment to HIV/AIDS. | |||
T29294 |
1-Acridinamine
1-Aminoakridin,1-Aminoacridine |
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1-Acridinamine is a biochemical. | |||
T68376 | Indinavir lactone | ||
Indinavir lactone is a protease inhibitor used as a component of highly active antiretroviral therapy to treat HIV/AIDS. | |||
T65992 | (R)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine | ||
(R)-4-Phenoxydinaphtho[2,1-d:1',2'-f][1,3,2]dioxaphosphepine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65992。 | |||
T67268 |
(S)-(3,5-Dioxa-4-phosphacyclohepta[2,1-a;3,4-a']dinaphthalen-4-yl)-5H-dibenz[b,f]azepine
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(S)-(3,5-Dioxa-4-phosphacyclohepta[2,1-a;3,4-a']dinaphthalen-4-yl)-5H-dibenz[b,f]azepine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67268,CAS号为 942939-38-0。 | |||
T31154 |
Cypridina luciferin
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Cypridina luciferin is a bioactive chemical. | |||
T5863L |
Indinavir
茚地那韦,MK-639,L 735 524,Crixivan |
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Indinavir (IDV) is an inhibitor of protease that is used as part of highly active antiretroviral therapy for the treatment of HIV/AIDS. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN7180 |
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-
4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C |
Others | Others |
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- (Meridianin C)是一种海洋来源的天然产物,存在于Aplidium meridianum。 | |||
TN6740 |
Emodinanthrone
大黄素蒽酮,Emodin anthranol,Emodin anthrone,emodinol |
Others; Antibiotic | Microbiology/Virology; Others |
Emodinanthrone 是一种蒽醌类化合物,是大黄素的前体,具有抗生素活性。它抑制大肠杆菌膜囊泡中呼吸驱动的溶质转运。 | |||
TN5766 |
Nandinaside A
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Nandinaside A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5766,CAS号为 1813517-23-5。 | |||
TN2916 |
3-Acetoxy-4,7(11)-cadinadien-8-one
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Others | Others |
3-Acetoxy-4,7(11)-cadinadien-8-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2916,CAS号为 104975-02-2。 | |||
TN2488 |
1,3,5-Cadinatriene-3,8-diol
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Others | Others |
1,3,5-Cadinatriene-3,8-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2488,CAS号为 941227-27-6。 | |||
TN3253 |
7alpha-Hydroxy-4,11-cadinadiene-3,8-dione
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Others | Others |
7alpha-Hydroxy-4,11-cadinadiene-3,8-dione 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3253,CAS号为 1423809-64-6。 | |||
TN5365 | 10β-Hydroxycadina-4,11(13)-dien-12,8β-olide | ||
10β-Hydroxycadina-4,11(13)-dien-12,8β-olide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5365,CAS号为 35001-23-1。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-00613 |
DNA polymerase II Protein, E. coli, Recombinant (His & Myc)
DNA polymerase II,polB,dinA,Pol II |
E. coli | E. coli |
Thought to be involved in DNA repair and/or mutagenesis. Its processivity is enhanced by the beta sliding clamp (dnaN) and clamp loader. |