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Search Results for " antiangiogenesis "

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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22436 Takeda-6d

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
Takeda-6d 是一种新型、有效的 DFG-out RAF/血管内皮生长因子受体 2 (VEGFR2) 抑制剂,IC50 分别为 7.0 nM 和 2.2 nM。
TQ0317 R1530

R-1530,R 1530

VEGFR; FGFR; FLT; PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
R1530 是一种多激酶抑制剂,具有抗肿瘤和抗血管生成活性。它是具有口服活性的有丝分裂/血管生成高效双重作用抑制剂, 抑制 VGFR2、FGFR1作用的 IC50分别为 10 nM 和 28 nM。
T7945 SU14813

VEGFR; PDGFR; c-Kit Angiogenesis; Tyrosine Kinase/Adaptors
SU14813 是一种多靶点受体酪氨酸激酶抑制剂,能够抑制 VEGFR2 (IC50:50 nM),VEGFR1 (IC50:2 nM),PDGFRβ (IC50:4 nM),KIT (IC50:15 nM)。
T29173 YF-452

YF-452 inhibits tumor growth through antiangiogenesis by suppressing VEGF receptor 2 signaling.
T69813 AZD-6126

AZD6126, also known as ANG-453, a water-soluble phosphate prodrug of N-acetylcolchinol with potential antiangiogenesis and antineoplastic activities. AZD-6126 is an angiogenesis inhibitor and tubulin inhibitor potentially for the treatment of solid tumours. AZD6126 is converted in vivo into N-acetylcolchinol. N-acetylcolchinol binds to and destabilizes the tubulin cytoskeleton of endothelial cells in tumor blood vessels, which may result in tumor endothelial cel apoptosis, the selective occlusio...

化合物

Takeda-6d
Cat.No: T22436
Synonym:
Target: VEGFR
R1530
Cat.No: TQ0317
Synonym: R-1530,R 1530
Target: VEGFR, FGFR, FLT, PDGFR
SU14813
Cat.No: T7945
Synonym:
Target: VEGFR, PDGFR, c-Kit
YF-452
Cat.No: T29173
Synonym:
Target:
AZD-6126
Cat.No: T69813
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0227 Sinensetin

Pedalitin permethyl ether,甜橙素

TNF; PGE Synthase Apoptosis; Immunology/Inflammation
Sinensetin (Pedalitin permethyl ether) 是从水果中发现的一种甲基化黄酮,有很强的抗血管和抗炎症的能力。

天然产物

Sinensetin
Cat.No: T4S0227
Synonym: Pedalitin permethyl ether,甜橙素
Target: TNF, PGE Synthase
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