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Cat. No. Product Name Target Signaling Pathways
T6713 Ulipristal

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Ulipristal 是性孕酮受体 (progesterone receptor) 的选择性调节剂。它能够与孕激素受体结合,抑制 PR 介导的基因表达,降低生殖系统中孕激素的活性。
T2527 Ulipristal acetate

Ulipristal,醋酸乌利司他,CDB-2914

Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy Autophagy; Endocrinology/Hormones; Others
Ulipristal acetate (CDB-2914) 是一种具有抗孕酮活性的选择性孕酮受体调节剂。它可抑制子宫平滑肌瘤病的生长。它通过抑制或延迟排卵和影响子宫内膜组织,可用作紧急避孕药。
T1541 Drospirenone

ZK 3059,屈螺酮,Dihydrospirorenone

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; COX Endocrinology/Hormones; Immunology/Inflammation; Neuroscience; Others
Drospirenone (ZK 3059) 是spironolactone 的类似物,是一种合成的孕酮。
T21256 Algestone

Alphasone

Algestone is a synthetic progestational dihydroxy derivative with anti-inflammatory properties.

化合物

Ulipristal
Cat.No: T6713
Synonym:
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Ulipristal acetate
Cat.No: T2527
Synonym: Ulipristal,醋酸乌利司他,CDB-2914
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Drospirenone
Cat.No: T1541
Synonym: ZK 3059,屈螺酮,Dihydrospirorenone
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, COX
Algestone
Cat.No: T21256
Synonym: Alphasone
Target:
TargetMol Loading
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