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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T23797 Bis(diazoacetyl)butane

1,4-Bis-diazoacetylbutane,Supermutagen,1,4-Bis(diazoacetyl)butane,DAB (mutagen)

Bis(diazoacetyl)butane is a mutagen and traditionally related to radio-mimetic chemical mutagens due to the similarity of appearance of mutagenic action of this mutagen and physical mutagens. It also has anti-tumor and carcinogenic activity.
T82620 DAB tetrahydrochloride dihydrate

3,3-Diaminobenzidine tetrahydrochloride dihydrate

3,3-Diaminobenzidine tetrahydrochloride dehydrate 作为染料,在组织化学(HC)及免疫组织化学(IHC)中应用广泛。该化合物主要用于过氧化物酶体染色和线粒体细胞色素c氧化酶活性的检测。

化合物

Bis(diazoacetyl)butane
Cat.No: T23797
Synonym: 1,4-Bis-diazoacetylbutane,Supermutagen,1,4-Bis(diazoacetyl)butane,DAB (mutagen)
Target:
DAB tetrahydrochloride dihydrate
Cat.No: T82620
Synonym: 3,3-Diaminobenzidine tetrahydrochloride dihydrate
Target:
Cat. No. Product Name Target Signaling Pathways
T2895 Lupeol

Fagarasterol,羽扇豆醇,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol

Apoptosis; Androgen Receptor; Akt Apoptosis; Cytoskeletal Signaling; Endocrinology/Hormones; PI3K/Akt/mTOR signaling
Lupeol (Monogynol B) 是一个活跃的五环三萜,具有抗氧化剂、抗肿瘤和抗炎活性。它是一种雄激素受体抑制剂,可研究癌症,特别是雄激素依赖表型和去势抵抗表型的前列腺癌。
T2863 p-Coumaric acid

para-Coumaric Acid,4-Hydroxycinnamic acid,trans-4-Hydroxycinnamic acid,对香豆酸,Trans-p-Coumaric acid,4-Coumaric acid,P-Hydroxycinnamic acid

Endogenous Metabolite; Antibiotic Metabolism; Microbiology/Virology
p-Coumaric acid (para-Coumaric Acid) 是肉桂酸的丰富异构体,具有抗诱变和抗肿瘤特性。
T5746 Dictamine

Dictamnine,Dectamine,白鲜碱

Apoptosis; Anti-infection; Antibacterial; Antifungal Apoptosis; Microbiology/Virology
Dictamine (Dectamine) 显示抗胆碱酯酶、抗炎、致突变、抗菌和抗真菌活性。 它具有在人子宫颈、结肠和口腔癌细胞中发挥细胞毒性的能力。
TN1711 Gossypetin

Antioxidant; p38 MAPK; MAPK; Antibacterial MAPK; Microbiology/Virology; oxidation-reduction
Gossypetin 是一种可从Rhodiola rosea Linn.中提取的六羟基化的类黄酮,是一种有效的 MKK3 和 MKK6 抑制剂,可强烈减弱 MKK3/6-p38 信号传导途径。Gossypetin 具有抗突变、抗动脉粥样硬化、抗氧化以及细胞保护和抗菌作用,它通过下调溶酶体酪蛋白酶 K 的活性和诱导肌动蛋白环破骨细胞中的自噬相关蛋白来抑制骨吸收。

天然产物

Lupeol
Cat.No: T2895
Synonym: Fagarasterol,羽扇豆醇,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol
Target: Apoptosis, Androgen Receptor, Akt
p-Coumaric acid
Cat.No: T2863
Synonym: para-Coumaric Acid,4-Hydroxycinnamic acid,trans-4-Hydroxycinnamic acid,对香豆酸,Trans-p-Coumaric acid,4-Coumaric acid,P-Hydroxycinnamic acid
Target: Endogenous Metabolite, Antibiotic
Dictamine
Cat.No: T5746
Synonym: Dictamnine,Dectamine,白鲜碱
Target: Apoptosis, Anti-infection, Antibacterial, Antifungal
Gossypetin
Cat.No: TN1711
Synonym:
Target: Antioxidant, p38 MAPK, MAPK, Antibacterial
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