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12

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1108 Allergen Gal d 4 (46-61), chicken

Lysozyme C (46-61) (chicken)

Allergen Gal d 4 (46-61), chicken is a hen egg white lysozyme peptide.
T22596 BADGE

PPAR DNA Damage/DNA Repair; Metabolism
BADGE 是一种标准化的化学过敏原。它的生理作用是通过增加组胺释放和细胞介导的免疫来实现的。
T14377 AZD5423

Glucocorticoid Receptor Endocrinology/Hormones
AZD5423 是可吸入的非甾体糖皮质激素受体选择性调节剂,能够有效降改善轻度过敏性哮喘患者的过敏原诱导反应。
T68173 ZD-2138

Ici-D2138

Lipoxygenase Metabolism
ZD-2138是一种有效且具有选择性的5-脂氧合酶(5-LOX)的特异性抑制剂,抑制了过敏原诱导的肺支气管收缩,可减少豚鼠孤立气道的神经诱发性快速激肽能收缩。ZD-2138可用来治疗哮喘疾病。
T81805 Mevonlerbart

Mevlonlerbart是针对Felcat allergen 1的特异性IgG4κ类抗体。Felcat allergen 1为一过敏原蛋白。
T82371 Freneslerbart

Freneslerbart为针对Felcat allergen 1的IgG4κ类抗体,后者为一过敏原蛋白。
T70107 Olcorolimus

Olcorolimus inhibits single allergen-induced allergic inflammation such as eosinophilic and lymphocytic infiltration and mRNA expression for interleukin (IL)-4 and IL-5
T81561 Palmitoyl tripeptide-8

Palmitoyl tripeptide-8,一种生物活性肽,具抗敏感功能,常作为化妆品成分应用。
T11482 GSK2245035

Others Others
GSK2245035 is a highly selective intranasal TLR7 agonist with preferential Type-1 interferon (IFN)-stimulating properties (pEC50s: 9.3 and 6.5 for IFNα and TFNα). It effectively suppresses allergen-induced Th2 cytokine production in human peripheral blood
T82820 Bremzalerbart

Bremzalerbart为针对主要桦树花粉过敏原Bet v 1-A的BETVIA的人源IgG4单克隆抗体。
T82946 Atisnolerbart

Atisnolerbart为一种靶向BETVIA的人源IgG4抗体,其中BETVIA指的是桦树花粉过敏原Bet v 1-A的主要成分。
T35457 (±)12(13)-DiHOME

(±)12(13)-DiHOME,Isoleukotoxin diol

(±)12(13)-DiHOME is the diol form of (±)12(13)-EpOME , a cytochrome P450-derived epoxide of linoleic acid also known as isoleukotoxin. [1] It is formed from 12(13)-EpOME by soluble epoxide hydrolase (sEH) in neutrophils. [2] 12(13)-DiHOME is toxic to Sf21 cells expressing sEH and to lacZ-expressing control cells, unlike isoleukotoxin, which is only toxic to cells containing sEH.[1] [2] Levels of 12(13)-DiHOME are increased in rat spinal cord following burn injury, and it enhances cold tolerance...

化合物

Allergen Gal d 4 (46-61), chicken
Cat.No: TP1108
Synonym: Lysozyme C (46-61) (chicken)
Target:
BADGE
Cat.No: T22596
Synonym:
Target: PPAR
AZD5423
Cat.No: T14377
Synonym:
Target: Glucocorticoid Receptor
ZD-2138
Cat.No: T68173
Synonym: Ici-D2138
Target: Lipoxygenase
Mevonlerbart
Cat.No: T81805
Synonym:
Target:
Freneslerbart
Cat.No: T82371
Synonym:
Target:
Olcorolimus
Cat.No: T70107
Synonym:
Target:
Palmitoyl tripeptide-8
Cat.No: T81561
Synonym:
Target:
GSK2245035
Cat.No: T11482
Synonym:
Target: Others
Bremzalerbart
Cat.No: T82820
Synonym:
Target:
Atisnolerbart
Cat.No: T82946
Synonym:
Target:
(±)12(13)-DiHOME
Cat.No: T35457
Synonym: (±)12(13)-DiHOME,Isoleukotoxin diol
Target:
Cat. No. Product Name Target Signaling Pathways
T4S0398 Rosin

松香树脂

p38 MAPK MAPK
Rosin 分离自松木或松树桩中,是一种频繁接触的过敏原,能够导致过敏性接触性皮炎。
T0834 Ethylparaben

Ethyl 4-hydroxybenzoate,Ethyl parahydroxybenzoate,羟苯乙酯,尼泊金乙酯

Antibacterial; Antifungal Microbiology/Virology
Ethylparaben (Ethyl parahydroxybenzoate) 是一种标准化的化学过敏原。 对羟基苯甲酸乙酯的生理作用是通过增加组胺释放和细胞介导免疫来实现的。
T0927 Butylparaben

Butyl 4-hydroxybenzoate,Butyl parahydroxybenzoate,尼泊金丁酯,对羟基苯甲酸丁酯

Endogenous Metabolite; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Butylparaben (Butyl 4-hydroxybenzoate) 是一种标准化的化学过敏原,可增加组胺释放和细胞介导的免疫。
T1297 Eugenol

丁香酚,4-Allylguaiacol,Allylguaiacol,4-Allyl-2-methoxyphenol,Eugenic acid

Apoptosis; Ferroptosis; Reactive Oxygen Species; Antibacterial; Parasite Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Eugenol (Allylguaiacol) 是一种从丁香中发现的精油,抑制脂质的过氧化,具有抗菌,驱虫和抗氧化活性。
T0908 Chlorquinaldol

5,7-Dichloro-8-hydroxy-2-methylquinoline,Chloquinan,氯喹那多

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Chlorquinaldol (5,7-Dichloro-8-hydroxy-2-methylquinoline) 是一种抗菌剂, 有潜力研究局部皮肤病症和阴道感染。
T5320 Tulipalin A

α-methylene-γ-butyrolactone,2-Methylenebutyrolactone,2-甲烯基丁内酯

Others; Drug Metabolite Metabolism; Others
Tulipalin A (α-methylene-γ-butyrolactone) 是来源于郁金香鳞茎的有毒糖苷。Tulipalin A 是引起过敏性接触皮炎的致敏性致敏物 (causative allergen),在低剂量影响免疫细胞的功能,例如 Jurkat T 细胞。

天然产物

Rosin
Cat.No: T4S0398
Synonym: 松香树脂
Target: p38 MAPK
Ethylparaben
Cat.No: T0834
Synonym: Ethyl 4-hydroxybenzoate,Ethyl parahydroxybenzoate,羟苯乙酯,尼泊金乙酯
Target: Antibacterial, Antifungal
Butylparaben
Cat.No: T0927
Synonym: Butyl 4-hydroxybenzoate,Butyl parahydroxybenzoate,尼泊金丁酯,对羟基苯甲酸丁酯
Target: Endogenous Metabolite, Antibacterial, Antibiotic
Eugenol
Cat.No: T1297
Synonym: 丁香酚,4-Allylguaiacol,Allylguaiacol,4-Allyl-2-methoxyphenol,Eugenic acid
Target: Apoptosis, Ferroptosis, Reactive Oxygen Species, Antibacterial, Parasite
Chlorquinaldol
Cat.No: T0908
Synonym: 5,7-Dichloro-8-hydroxy-2-methylquinoline,Chloquinan,氯喹那多
Target: Antibacterial, Antibiotic, Antifungal
Tulipalin A
Cat.No: T5320
Synonym: α-methylene-γ-butyrolactone,2-Methylenebutyrolactone,2-甲烯基丁内酯
Target: Others, Drug Metabolite
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