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Cat. No. Product Name Target Signaling Pathways
T4S1999 Valepotriate

戊曲酯/缬草素,Valtrate

Apoptosis; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Valepotriate (Valtrate) 是从蜘蛛香分离而来的一种天然产物,是一类新的细胞毒剂和抗肿瘤剂,对 HTC 肝癌细胞是非常有效的细胞毒剂。 它可能对焦虑的精神症状具有潜在的抗焦虑作用。
TN4341 IVHD-valtrate

Mdm2; BCL; PARP; Caspase; p53 Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
VHD-valtrate has anticancer effects against human ovarian cancer cells in vitro and in vivo, it is a potential therapeutic agent for ovarian cancer, providing a basis for development of the compound as a novel chemotherapeutic agent.
T8803 Valtrate hydrine B4

Valtrate hydrine B4 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T8803,CAS号为 18296-48-5。
TJP2872 Acevaltrate

Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate

ATPase; Others Membrane transporter/Ion channel; Others
Acevaltrate (Acevaltratum) 对人小细胞肺癌细胞系 GLC(4) 和人结肠直肠癌细胞系 COLO 320 具有高细胞毒性,IC50 值为 1-6 uM。它抑制大鼠肾和脑半球中 Na+/K+-ATP 酶活性,IC50分别为 22.8 和 42.3 μM。
TN3844 Didrovaltrate

Calcium Channel Membrane transporter/Ion channel; Metabolism
Didrovaltrate shows cytotoxic against human cancer cell lines. Didrovaltrate blocks I(Ca-L) in a concentration-dependent manner and probably inhibits I(Ca-L) in its inactive state, which may contribute to its cardiovascular effect.
TN3646 Chlorovaltrate K

Others Others
Chlorovaltrate K shows moderate cytotoxicity against lung adenocarcinoma (A 549), metastatic prostate cancer (PC-3M), colon cancer (HCT-8) and hepatoma (Bel 7402) cell lines with IC50 values of 0.89-9.76 uM.
TN4352 Jatamanvaltrate B

Others Others
Jatamanvaltrate B shows cytotoxicity against lung adenocarcinoma (A549), metastatic prostate cancer (PC-3M), colon cancer (HCT-8),and hepatoma (Bel7402) cell lines.
TN5249 Volvaltrate B

Others Others
Volvaltrate B shows cytotoxic activity against the lung adenocarcinoma (A549), metastatic prostate cancer (PC-3M), colon cancer (HCT-8), and hepatoma (Bel7402) cell lines, with IC50 values of 8.5, 2.0, 3.2, and 6.1 uM, respectively.
TN1024 Baldrinal

Others Others
Baldrinal, valtrate, and acevaltrate are the quality control compounds of Valeriana jatamansi Jones.

天然产物

Valepotriate
Cat.No: T4S1999
Synonym: 戊曲酯/缬草素,Valtrate
Target: Apoptosis, HIV Protease
IVHD-valtrate
Cat.No: TN4341
Synonym:
Target: Mdm2, BCL, PARP, Caspase, p53
Valtrate hydrine B4
Cat.No: T8803
Synonym:
Target:
Acevaltrate
Cat.No: TJP2872
Synonym: Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate
Target: ATPase, Others
Didrovaltrate
Cat.No: TN3844
Synonym:
Target: Calcium Channel
Chlorovaltrate K
Cat.No: TN3646
Synonym:
Target: Others
Jatamanvaltrate B
Cat.No: TN4352
Synonym:
Target: Others
Volvaltrate B
Cat.No: TN5249
Synonym:
Target: Others
Baldrinal
Cat.No: TN1024
Synonym:
Target: Others
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