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Cat. No. | Product Name | Target | Signaling Pathways |
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T11937L |
m-Tyramine hydrobromide
|
Others | Others |
m-Tyramine hydrobromide, an endogenous trace amine neuromodulator, influences both the adrenergic and dopaminergic receptors. | |||
T13622 |
Cholestyramine
Colestyramine,考来烯胺,Cholestyramine resin |
Others | Others |
Cholestyramine (Cholestyramine resin) 是一种胆汁酸结合树脂,能够抑制肠胆汁酸吸收导致增加粪便胆汁酸排泄,提高胆固醇胆汁酸合成。 | |||
T126368 |
N-Tetracosanoyltyramine
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N-Tetracosanoyltyramine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126368。 | |||
T5327 |
Amezinium methylsulfate
Amezinium metilsulfate,甲磺美嗪,Amezinium (methylsulfate),Lu-1631 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Amezinium methylsulfate (Lu-1631) 具有多种机制,包括刺激 α 和 β-1 受体以及抑制去甲肾上腺素和酪胺的摄取。 | |||
T69270 |
Amezinium
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Amezinium is a sympathomimetic drug used for the treatment of low blood pressure. It has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake. | |||
T1488L |
Procarbazine free base
CB 400-497,NSC-77213,Ro 4-6467/1,Ro 4-6467,Procarbazine |
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Procarbazine is an antineoplastic chemotherapy drug for the treatment of Hodgkin's lymphoma and certain brain cancers. The drug is metabolized and activated in the liver. It also inhibits MAO thus increasing the effects of sympathomimetics, TCAs, and tyra | |||
T71910 |
Racemic rasagiline
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Racemic rasagiline,也称为 AGN-1135,是一种单胺氧化酶 B 型抑制剂(MAOI)。然而,在食用富含酪胺的食物的患者中,这种药物的应用可能导致致命的高血压危象。TVP-1022是雷沙吉兰的(S)异构体,具有心脏保护剂的作用。 | |||
T73614 | Tyrosine decarboxylase | ||
Tyrosine decarboxylase (TDC; TyrDC),即酪氨酸脱羧酶,广泛存在于植物、昆虫和不同微生物中,常用于生化研究。Tyrosine decarboxylase 是一种5'-磷酸吡哆醛 (PLP) 依赖性脱羧酶,可以催化酪氨酸中羧基的去除,产生酪胺和二氧化碳。 | |||
T36521 |
Alaproclate (hydrochloride)
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Alaproclate is a selective serotonin reuptake inhibitor (SSRI).1,2 It inhibits depletion of serotonin (5-HT) induced by 4-methyl-α-ethyl-m-tyramine in rat cerebral cortex, hippocampus, hypothalamus, and striatum (EC50s = 18, 4, 8, and 12 mg/kg, respectively).1 Alaproclate inhibits NMDA-evoked currents and depolarization-induced voltage-dependent potassium currents in rat hippocampal neurons (IC50s = 1.1 and 6.9 μM, respectively) and does not inhibit GABA-evoked currents when used at concentratio... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3095 |
Tyramine
4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine |
MAO; Endogenous Metabolite | Metabolism; Neuroscience |
Tyramine (Uteramine) 是天然存在于体内或某些食物中的氨基酸。Tyramine 有助于调节血压。 | |||
T7851 |
Tyramine hydrochloride
盐酸酪胺,酪胺盐酸盐 |
Others; Endogenous Metabolite | Metabolism; Others |
Tyramine hydrochloride 是一种氨基酸,有助于调节血压。其中 Tyramine 天然存在于体内,并存在于某些食物中。 | |||
T11937 |
m-Tyramine
|
Others | Others |
m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator. | |||
TN6457 |
N-trans-caffeoyltyramine
Trans-N-Caffeoyltyramine,N-(E)-Caffeoyl-lambda-tyramine,N-cis-Caffeoyltyramine,Typheramide |
Immunology/Inflammation related | Immunology/Inflammation |
N-trans-caffeoyltyramine (Trans-N-Caffeoyltyramine) 是炎症反应的调节剂,可用于慢性炎症性疾病治疗的研究。 | |||
TN7064 |
Candicine
4-Hydroxy-N-Benzeneethanaminium,N, N, N-trimethyltyramine chloride,Candicin,N-Methylhordenine,Tyramine Impurity 1,4-羟基-N,N,N-三甲基-苯乙铵,2-(4-hydroxyphenyl)ethyl-trimethylazanium |
Others | Others |
Candicine (N, N, N-trimethyltyramine chloride) 是来自 Stapelia gigantea 的天然产品。 | |||
T82407 | Feruloyl tyramine | ||
Feruloyl tyramine 为一酰胺类化合物,可从大麻籽乙醇提取物中分离。在小鼠侧脑室注射该化合物,可引发体温降低及运动协调障碍。 | |||
T37341 |
N-Acetyltyramine
|
Antibacterial | Microbiology/Virology |
N-Acetyltyramine 是一种群体感应抑制剂,由溶藻弧菌 M3-10 产生。N-Acetyltyramine 可以抑制C. violaceumATCC 12472 的群体感应。它可以逆转阿霉素耐药白血病 P388 细胞的耐药性。 | |||
TN7042 |
N-methyltyramine
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Adrenergic Receptor | GPCR/G Protein; Neuroscience |
N-methyltyramine 是一种从豆科植物大叶相思中分离出的生物碱,是一种 α2-肾上腺素受体拮抗剂,通过酶促肾上腺素合成调节肾上腺素能受体,可用于研究肠道疾病。 | |||
TN3669 |
Cis-N-Feruloyltyramine
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Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Cis-N-Feruloyltyramine 是一种天然存在的化合物,存在于各种植物中,对 P-388癌细胞系具有细胞毒性。 Cis-N-Feruloyltyramine 是体外前列腺素(PG)合成的抑制剂。 | |||
TN4618 |
N-trans-Sinapoyltyramine
|
Others | Others |
N-trans-Sinapoyltyramine 对 HeLa 人癌细胞系表现出强烈的选择性细胞毒性,IC50 值为 9.77 ± 1.25 μm。 | |||
T12142 |
N-Caffeoyl O-methyltyramine
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Glucosidase | Metabolism |
N-Caffeoyl O-methyltyramine 是一种生物碱,分离自Cuscuta reflexa,能够较大程度抑制α-葡萄糖苷酶的活性(IC50:103.58 μM)。 | |||
TN1030 |
N-p-trans-Coumaroyltyramine
N-反式对香豆酰基酪胺,N-反式-对香豆酰酪胺 |
AChE; Parasite | Microbiology/Virology; Neuroscience |
N-p-trans-Coumaroyltyramine 是从蓼属植物中分离出的肉桂酰苯乙酰胺,是一种乙酰胆碱酯酶抑制剂,IC50 为 122 μM。它具有抗锥虫活性,对T. brucei rhodesiense 作用的 IC50值为 13.3 µM。 | |||
T3S0645 |
N-trans-Feruloyltyramine
Feruloyltyramine,N-Feruloyltyramine,Moupinamide,N-反式阿魏酰酪胺 |
Others; COX | Immunology/Inflammation; Neuroscience; Others |
N-trans-Feruloyltyramine (Feruloyltyramine) 是从大麻中分离得到的一种生物碱,是COX1和COX2的抑制剂,具有抗氧化和抗炎活性。 | |||
T4710 |
3-Methoxytyramine hydrochloride
3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐 |
Others; Endogenous Metabolite; Drug Metabolite | Metabolism; Others |
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 是多巴胺的无活性代谢物,能够活化痕量胺相关受体1 。 | |||
T8269 |
3-Methoxytyramine
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Others; Endogenous Metabolite | Metabolism; Others |
3-Methoxytyramine 是一种神经调节剂,是 3-羟基酪胺/多巴胺的细胞外代谢产物。 | |||
TN4617 |
N-trans-Feruloyl-3-methoxytyramine
|
Others | Others |
N-trans-Feruloyl-3-methoxytyramine shows significantly DPPH radical scavenging activities. | |||
T5263 |
p-Hydroxymandelic acid
4-羟基扁桃酸,4-Hydroxymandelic acid |
Others; Endogenous Metabolite | Metabolism; Others |
p-Hydroxymandelic acid (4-Hydroxymandelic acid) 是有价值的芳香类化学品,常用于生产药物和食品添加剂。 |