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抑制剂 & 化合物

8

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Cat. No. Product Name Target Signaling Pathways
T67757 (9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one

Immunology/Inflammation related Immunology/Inflammation
(9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one 是青藤碱的主要代谢物。青藤碱是来源于青藤的代谢物。(9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one 显示出抗炎活性。

化合物

(9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one
Cat.No: T67757
Synonym:
Target: Immunology/Inflammation related
Cat. No. Product Name Target Signaling Pathways
T2726 Sinomenine

Cucoline,Kukoline,青藤碱

Apoptosis; Others; NF-κB; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; NF-κB; Others
Sinomenine (Kukoline) 是来自汉防己的一种生物碱,是 μ 阿片受体激活剂,也是NF-κB 活化的阻断剂。
TN7068 Sinomenine N-oxide

Others Others
Sinomenine N-oxide 是青藤碱循环代谢机制的主要代谢产物之一。
T2921 Sinomenine hydrochloride

盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride

Apoptosis; NF-κB; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; NF-κB
Sinomenine hydrochloride (Kukoline hydrochloride) 是来自汉防己的一种生物碱,是NF-κB 活化的阻断剂。Sinomenine 也是一种 μ 阿片受体激活剂。
T2996 Tetrandrine

NSC-77037,d-Tetrandrine,Hanfangchin A,粉防己碱,Fanchinine,Sinomenine A,汉防己甲素

Potassium Channel; Calcium Channel Membrane transporter/Ion channel; Metabolism
Tetrandrine (Sinomenine A) 是来自粉防己的一种双苯基异喹啉生物碱,可抑制电压门控钙离子通道 (ICa) 和 Ca2+激活的钾离子通道。
T83255 7(R)-7,8-Dihydrosinomenine

7(R)-7,8-Dihydrosinomenine是从青藤中分离出的异喹啉生物碱,具备抗破骨细胞活性。
T83481 1,1′-Disinomenine

1,1'-Disinomenine,一种从Sinomenium acutum茎部分离得到的生物碱,对A549和Hela细胞表现出较弱的抑制效果。
T83449 14-Episinomenine

14-Episinomenine为Stephania cepharantha所含生物碱,具可提取性质。
T3S1319 (+)-Magnoflorine

Escholin,Magnoflorine,Thalictrin,Escholine,木兰花碱

Others; Antifungal Microbiology/Virology; Others
(+)-Magnoflorine (Thalictrin) 是从 Acoruscalamus 中分到的一种阿朴啡生物碱,可以减少 C. albicans 生物膜的形成,具有抗真菌、抗氧化、抗糖尿病、镇静和抗焦虑的作用。

天然产物

Sinomenine
Cat.No: T2726
Synonym: Cucoline,Kukoline,青藤碱
Target: Apoptosis, Others, NF-κB, Opioid Receptor, Autophagy
Sinomenine N-oxide
Cat.No: TN7068
Synonym:
Target: Others
Sinomenine hydrochloride
Cat.No: T2921
Synonym: 盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride
Target: Apoptosis, NF-κB, Opioid Receptor, Autophagy
Tetrandrine
Cat.No: T2996
Synonym: NSC-77037,d-Tetrandrine,Hanfangchin A,粉防己碱,Fanchinine,Sinomenine A,汉防己甲素
Target: Potassium Channel, Calcium Channel
7(R)-7,8-Dihydrosinomenine
Cat.No: T83255
Synonym:
Target:
1,1′-Disinomenine
Cat.No: T83481
Synonym:
Target:
14-Episinomenine
Cat.No: T83449
Synonym:
Target:
(+)-Magnoflorine
Cat.No: T3S1319
Synonym: Escholin,Magnoflorine,Thalictrin,Escholine,木兰花碱
Target: Others, Antifungal
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