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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0351 Risperidone

Risperidal,R 64 766,利培酮

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂,对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。
T0351L Risperidone Mesylate

Risperidone Mesylate salt

Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.
T12734 Risperidone E-oxime

Others Others
Risperidone E-oxime is an impurity of Risperidone. Risperidone is a serotonin blocker of 5-HT2 receptor, P-Glycoprotein inhibitor and potent dopamine D2 receptor antagonist(Kis of 4.8, 5.9 nM for 5-HT2A and dopamine D2 receptor, respectively ).
T62661 Risperidone hydrochloride

Risperidone hydrochloride (R 64 766 hydrochloride) 是一种 5-HT2 受体的阻断剂,P-糖蛋白 (P-Glycoprotein) 的抑制剂和 dopamine D2 受体的拮抗剂,其能够作用于 5-HT2A (Ki: 4.8 nM) 和 dopamine D2 (Ki: 5.9 nM)受体。
T73715 Risperidone-d

Risperidone-d4是 Risperidone 的氘代物。Risperidone 是5-HT2受体的阻断剂,P-糖蛋白(P-Glycoprotein)的抑制剂 和dopamine D2受体的拮抗剂,其对 5-HT2A 和 dopamine D2受体的Ki 值分别为 4.8,5.9 nM。

化合物

Risperidone
Cat.No: T0351
Synonym: Risperidal,R 64 766,利培酮
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, P-gp
Risperidone Mesylate
Cat.No: T0351L
Synonym: Risperidone Mesylate salt
Target:
Risperidone E-oxime
Cat.No: T12734
Synonym:
Target: Others
Risperidone hydrochloride
Cat.No: T62661
Synonym:
Target:
Risperidone-d
Cat.No: T73715
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0076 Paliperidone

9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。

天然产物

Paliperidone
Cat.No: T0076
Synonym: 9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
TargetMol Loading
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