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Cat. No. | Product Name | Target | Signaling Pathways |
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T0351 |
Risperidone
Risperidal,R 64 766,利培酮 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂,对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。 | |||
T0351L |
Risperidone Mesylate
Risperidone Mesylate salt |
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Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker. | |||
T12734 |
Risperidone E-oxime
|
Others | Others |
Risperidone E-oxime is an impurity of Risperidone. Risperidone is a serotonin blocker of 5-HT2 receptor, P-Glycoprotein inhibitor and potent dopamine D2 receptor antagonist(Kis of 4.8, 5.9 nM for 5-HT2A and dopamine D2 receptor, respectively ). | |||
T62661 |
Risperidone hydrochloride
|
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Risperidone hydrochloride (R 64 766 hydrochloride) 是一种 5-HT2 受体的阻断剂,P-糖蛋白 (P-Glycoprotein) 的抑制剂和 dopamine D2 受体的拮抗剂,其能够作用于 5-HT2A (Ki: 4.8 nM) 和 dopamine D2 (Ki: 5.9 nM)受体。 | |||
T73715 |
Risperidone-d
|
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Risperidone-d4是 Risperidone 的氘代物。Risperidone 是5-HT2受体的阻断剂,P-糖蛋白(P-Glycoprotein)的抑制剂 和dopamine D2受体的拮抗剂,其对 5-HT2A 和 dopamine D2受体的Ki 值分别为 4.8,5.9 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0076 |
Paliperidone
9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。 |