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Cat. No. Product Name Target Signaling Pathways
T0849 Pyrimethamine

Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶

DHFR; Antifolate; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Pyrimethamine (Pirimecidan) 是一种二氢叶酸还原酶的竞争性抑制剂,用作抗疟药。
T0930 Sulfadiazine

Sulphadiazine,磺胺嘧啶

Antibacterial; Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。
T0836 Sulfadoxine

周效磺胺,磺胺多辛,Sulphadoxine

DHFR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Proteases/Proteasome
Sulfadoxine (Sulphadoxine) 是磺胺类化合物,常与pyrimethamine 结合起到抗疟疾作用。它抑制HIV 在外周血单核细胞中的复制。
T17257 WR99210

DHFR; Antifolate; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
WR99210 是一种有效的、可口服的且毒性较低的二氢叶酸还原酶 (DHFR) 抑制剂 (IC50<0.075 nM)。WR99210 具有较好的抗寄生虫活性,对间日疟原虫和恶性疟原虫株 (包括耐 Pyrimethamine  的恶性疟原虫株) 以及弓形虫有良好的抑制作用。
T69089 Trimethoprim sulfate

Trimethoprim sulfate is a pyrimidine inhibitor of dihydrofolate reductase, it is an antibacterial related to PYRIMETHAMINE. The interference with folic acid metabolism may cause a depression of hematopoiesis. It is potentiated by SULFONAMIDES and the TRIMETHOPRIM-SULFAMETHOXAZOLE COMBINATION is the form most often used. It is sometimes used alone as an antimalarial. TRIMETHOPRIM RESISTANCE has been reported.

化合物

Pyrimethamine
Cat.No: T0849
Synonym: Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶
Target: DHFR, Antifolate, Parasite
Sulfadiazine
Cat.No: T0930
Synonym: Sulphadiazine,磺胺嘧啶
Target: Antibacterial, Antibiotic, Parasite, Autophagy
Sulfadoxine
Cat.No: T0836
Synonym: 周效磺胺,磺胺多辛,Sulphadoxine
Target: DHFR, HIV Protease, Antibiotic, Parasite, Autophagy
WR99210
Cat.No: T17257
Synonym:
Target: DHFR, Antifolate, Antibacterial
Trimethoprim sulfate
Cat.No: T69089
Synonym:
Target:
TargetMol Loading
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