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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T23133 Pentamidine

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine 是抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T1654 Pentamidine isethionate

Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine isethionate (Pentamidine diisethionate) 是抗微生物剂,会干扰 DNA 的生物合成。它抑制寄生虫Leishmania infantum,IC50为 2.5 μM。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它有抗肿瘤和抗菌活性。
T23132 Pentamidine dihydrochloride

喷他脒二盐酸盐,MP-601205 dihydrochloride

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine dihydrochloride (MP-601205 dihydrochloride) 是一种抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T32891 l-Primaquine

BRN0019337,BRN-0019337,BRN 0019337

l-Primaquine is used to treat and prevent malaria and to treat Pneumocystis pneumonia.
T16428 Pafuramidine

DB289

Others Others
Pafuramidine is an orally bioavailable prodrug of furamidine. It has activity against Pneumocystis pneumonia (IC50 value: 4.5 nM)
T19198 Atovaquone-d4

阿托伐醌D4

Others Others
Atovaquone D4 is the deuterium-labeled Atovaquone. Atovaquone is a medication used to treat or prevent pneumocystis babesia, malaria, toxoplasmosis, and pneumonia.
T39862 Trimethoprim lactate

Trimethoprim lactic is a bacteriostatic antibiotic and an orally active dihydrofolate reductase inhibitor. Trimethoprim lactic is active against a wide range of Gram-positive and Gram-negative aerobic bacteria . Trimethoprim lactic has the potential for urinary tract infections, Shigellosis and Pneumocystis pneumonia treatment.
T75291 Trimethoprim hydrochloride

Trimethoprim hydrochloride 是一种口服活性的抑菌抗生素,同时也是二氢叶酸还原酶抑制剂。它对多种革兰氏阳性及革兰氏阴性需氧细菌有效。用于尿路感染、志贺氏菌病和肺孢子菌肺炎的研究。与锌联合使用时,可抑制甲型流感病毒对鸡胚的感染。

化合物

Pentamidine
Cat.No: T23133
Synonym:
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Pentamidine isethionate
Cat.No: T1654
Synonym: Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Pentamidine dihydrochloride
Cat.No: T23132
Synonym: 喷他脒二盐酸盐,MP-601205 dihydrochloride
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
l-Primaquine
Cat.No: T32891
Synonym: BRN0019337,BRN-0019337,BRN 0019337
Target:
Pafuramidine
Cat.No: T16428
Synonym: DB289
Target: Others
Atovaquone-d4
Cat.No: T19198
Synonym: 阿托伐醌D4
Target: Others
Trimethoprim lactate
Cat.No: T39862
Synonym:
Target:
Trimethoprim hydrochloride
Cat.No: T75291
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1153 Trimethoprim

NIH 204,BW 56-72,甲氧苄啶,NSC-106568

DHFR; DNA/RNA Synthesis; Antifolate; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Trimethoprim (NSC-106568) 是抑菌抗生素,也是具有口服活性的二氢叶酸还原酶抑制剂。它对多种革兰氏阳性和革兰氏阴性需氧细菌具有活性,可用于尿路感染,肺孢子菌肺炎和志贺氏菌病的研究。

天然产物

Trimethoprim
Cat.No: T1153
Synonym: NIH 204,BW 56-72,甲氧苄啶,NSC-106568
Target: DHFR, DNA/RNA Synthesis, Antifolate, Antibacterial, Antibiotic
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