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Targets Recommended: Apoptosis HDAC

6

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T1890 Pracinostat

SB939

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Pracinostat (SB939) 是一种组蛋白去乙酰化酶抑制剂,对 HDACs 的IC50值为 40-140 nM,可用于研究癌症。
T2262 Itanapraced

CHF5074,CSP-1103

Beta Amyloid; Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Itanapraced (CHF5074) 是新型γ-secretase 调节剂,能够降低 Aβ42 (IC50=3.6 nM) 和 Aβ40 (IC50=18.4 nM) 分泌。
T21371 Apraclonidine hydrochloride

Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum

Adrenergic Receptor GPCR/G Protein; Neuroscience
Apraclonidine hydrochloride (ALO 2145) 是一种 α2-肾上腺素能激动剂和弱的 α-1 肾上腺素能受体激动剂。 Apaclonidine hydrochloride 可降低人眼的眼内压,可用于青光眼治疗的研究。
T13451L Mapracorat

BOL-303242X,ZK-245186

Others Others
Mapracorat is a novel non-steroidal selective agonist of glucocorticoid receptor.
T13451 (S)-Mapracorat

(S)-ZK-245186,(S)-BOL-303242X

Others Others
(S)-Mapracorat is a selective and less active agonist of glucocorticoid receptor.
T60350 Apraclonidine

Apraclonidine (ALO 2145) 是一种选择性α2和弱 α1 受体激动剂,可有效降低人眼的眼内压。Apraclonidine 也是一种局部滴眼液。

化合物

Pracinostat
Cat.No: T1890
Synonym: SB939
Target: Apoptosis, HDAC
Itanapraced
Cat.No: T2262
Synonym: CHF5074,CSP-1103
Target: Beta Amyloid, Gamma-secretase
Apraclonidine hydrochloride
Cat.No: T21371
Synonym: Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum
Target: Adrenergic Receptor
Mapracorat
Cat.No: T13451L
Synonym: BOL-303242X,ZK-245186
Target: Others
(S)-Mapracorat
Cat.No: T13451
Synonym: (S)-ZK-245186,(S)-BOL-303242X
Target: Others
Apraclonidine
Cat.No: T60350
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-01555 PRAC Protein, Human, Recombinant (His & SUMO)

PRAC,C17orf92

Human E. coli
The PRAC gene is located on chromosome 17 at position 17q21, about 4 kbp downstream from the homeodomain Hoxb-13 gene. The pathogenesis of PCa may be due to the expression levels of PRAC protein, and this protein can serve as a potential biomarker for the management of PCa.

重组蛋白

PRAC Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPY-01555
Species: Human
Expression System: E. coli
TargetMol Loading
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