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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1890 |
Pracinostat
SB939 |
Apoptosis; HDAC | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Pracinostat (SB939) 是一种组蛋白去乙酰化酶抑制剂,对 HDACs 的IC50值为 40-140 nM,可用于研究癌症。 | |||
T2262 |
Itanapraced
CHF5074,CSP-1103 |
Beta Amyloid; Gamma-secretase | Neuroscience; Proteases/Proteasome; Stem Cells |
Itanapraced (CHF5074) 是新型γ-secretase 调节剂,能够降低 Aβ42 (IC50=3.6 nM) 和 Aβ40 (IC50=18.4 nM) 分泌。 | |||
T21371 |
Apraclonidine hydrochloride
Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Apraclonidine hydrochloride (ALO 2145) 是一种 α2-肾上腺素能激动剂和弱的 α-1 肾上腺素能受体激动剂。 Apaclonidine hydrochloride 可降低人眼的眼内压,可用于青光眼治疗的研究。 | |||
T13451L |
Mapracorat
BOL-303242X,ZK-245186 |
Others | Others |
Mapracorat is a novel non-steroidal selective agonist of glucocorticoid receptor. | |||
T13451 |
(S)-Mapracorat
(S)-ZK-245186,(S)-BOL-303242X |
Others | Others |
(S)-Mapracorat is a selective and less active agonist of glucocorticoid receptor. | |||
T60350 |
Apraclonidine
|
||
Apraclonidine (ALO 2145) 是一种选择性α2和弱 α1 受体激动剂,可有效降低人眼的眼内压。Apraclonidine 也是一种局部滴眼液。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01555 |
PRAC Protein, Human, Recombinant (His & SUMO)
PRAC,C17orf92 |
Human | E. coli |
The PRAC gene is located on chromosome 17 at position 17q21, about 4 kbp downstream from the homeodomain Hoxb-13 gene. The pathogenesis of PCa may be due to the expression levels of PRAC protein, and this protein can serve as a potential biomarker for the management of PCa. |