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55

抑制剂 & 化合物

3

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Cat. No. Product Name Target Signaling Pathways
TP2496 Octapeptide-2 Acetate

Octapeptide-2 Acetate(1374396-34-5 Free base)

Others Others
Octapeptide-2 Acetate 作为一种促进毛发生长的活性物质,是一种双层封装的仿生肽,有助于促进细胞生长和迁移。它通过激活毛囊的干细胞来促进头发生长。 它比天然蛋白质更稳定且作用时间更长。
TP1616L Hsp70-derived octapeptide acetate

Hsp70-derived octapeptide acetate(736171-62-3 free base)

Others Others
Hsp70-derived octapeptide acetate (Hsp70-derived octapeptide acetate)(736171-62-3 free base) 是一组含有四肽重复 (TPR) 的蛋白质,已显示与 70 kDa 热休克同源蛋白 (hsc70) 的 C 末端结构域相互作用。在本研究中,含 TPR 的蛋白质,包括 hsc70 相互作用蛋白 (CHIP)、TPR1 和人富含谷氨酰胺的 TPR 含蛋白 (hSGT) 的 C 端,对 DnaJ 和 hsc70 对荧光素酶重折叠的影响进行了调查。
TP2204L CCK Octapeptide, non-sulfated acetate

CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)

cholecystokinin GPCR/G Protein
CCK Octapeptide, non-sulfated acetate 是一种合成的胆囊收缩素脱硫酸肽。
T39170 Cholecystokinin Octapeptide, desulfated TFA

CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA

Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.
TP2204 Cholecystokinin Octapeptide, desulfated

CCK Octapeptide, non-sulfated

Others Others
Non-sulfated form of the C-terminal octapeptide of CCK
TP1198 Sincalide ammonium

SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium

cholecystokinin GPCR/G Protein
Sincalide ammonium (CCK-8 ammonium) 是一种有效的氨基酸多肽激素胆囊收缩素 (CCK) 的类似物,是保留了 CCK 的大部分生物活性的活性片段。Sincalide ammonium 促进胆汁的分泌,使胆囊收缩并使 Oddi 的括约肌松弛,从而促进胆汁排入十二指肠。Sincalide ammonium 可通过注射促进胆囊收缩,常用于辅助诊断胆囊、胰腺疾病和胆囊造影术。
TP1197 Sincalide

SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide

Others Others
Sincalide (CCK-8) 是一种速效的胆囊收缩素的氨基酸多肽激素类似物,可在胆囊造影术中静脉使用。它的肝胆生理作用是增加胆汁的分泌,使胆囊收缩并使 Oddi 的括约肌松弛,从而使胆汁排入十二指肠。它是一种通过注射促进胆囊收缩并帮助诊断胆囊和胰腺疾病的药物。
TP1616 Hsp70-derived octapeptide

A group of tetratricopeptide repeat (TPR)-containing proteins has been shown to interact with the C-terminal domain of the 70 kDa heat-shock cognate protein (hsc70). In the present study, the effect of the TPR-containing proteins, including the C-terminus
TP2386 Ige octapeptide (497-504)

Ige octapeptide (497-504) is a bioactive chemical.
TP2389 Laminin B1 octapeptide P-8

Asp-pro-gln-tyr-ile-gln-ser-arg,Dpgyigsr

Laminin B1 octapeptide P-8 is a synthetic laminin B1 chain octapeptide with laminin receptor binding ability.
T80204 Octapeptide-2

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Octapeptide-2, 已报道作为化妆品成分,是一种具促进毛发生长功能的生物活性肽。
T7615 Xenopsin

爪蟾肽,Xenopsin(2TFA)

Others Others
Xenopsin (Xenopsin(2TFA)) 是一种神经降压素样八肽,来自于非洲爪蟾皮肤,能够抑制胃泌素刺激的胃酸分泌。
T4119 Octreotide Acetate

醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)

Somatostatin GPCR/G Protein
Octreotide Acetate (Sandostatin) 是一种长期有效的合成生长抑素八肽类似物,可抑制生长激素的分泌。
T7615L Xenopsin 2TFA(51827-01-1(free base)

Others Others
Xenopsin 2TFA(51827-01-1(free base) 是一种以前从两栖动物皮肤中分离出来的神经降压素样八肽。
TP1114L Leucokinin VIII acetate

Leucokinin 8

Others Others
Leucokinin VIII acetate (Leucokinin 8) 是一种从蟑螂头部提取物中分离的利尿八肽。
TP1785L Peptide T acetate(106362-32-7 free base)

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Peptide T acetate(106362-32-7 free base) 是一种来自 HIV-1 gp120 V2 区域的八肽。它是一种合成八肽,其可能的作用机制是 gp120 对 CD4 受体的竞争性抑制以及与血管肠肽受体的结合和抑制细胞因子作用。
TP1074L Neuropeptide FF acetate(99566-27-5 free base)

NPFF acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) 是属于 RF 酰胺家族的八肽。 NPFF 与 G 蛋白偶联受体 NPFF (1) 和 NPFF (2) 相互作用。
TP1605L1 Allatostatin IV TFA(123338-13-6 free base)

Others Others
Allatostatin IV TFA(123338-13-6 free base) 是一种八肽胺,是在昆虫中发现的抑制(allatostatins)或刺激(allatotropins)保幼激素(JH)合成的调节肽家族的成员。
T7497L C3a 70-77 2TFA(63555-63-5(free base))

Complement 3a (70-77)

Complement System Immunology/Inflammation
C3a 70-77 2TFA(63555-63-5(free base)) (Complement 3a (70-77)) 是对应于 C3a 的 COOH 末端的八肽。
TP2446L Angiotensin amide acetate

血管紧张素胺,Angiotensin amide acetate(53-73-6 Free base)

Others Others
Angiotensin amide acetate 是Angiotensin amide 的衍生物。Angiotensin amide 是一种八肽酰胺,可以通过血管收缩来提高血压。
T7497L1 C3a 70-77 acetate

C3a 70-77 acetate (63555-63-5 Free base)

Others Others
C3a 70-77 acetate 是对应于 C3a 的 COOH 末端的八肽乙酸酯,具有 C3a 的特异性和 1% 至 2% 的生物活性。
TP1346 CYN 154806 TFA

CYN 154806 TFA

Somatostatin GPCR/G Protein
CYN 154806 TFA(183658-72-2 free base) 是一种环状八肽,是一种有效的选择性生长抑素 sst2 受体拮抗剂。对于重组 sst2、sst1、sst3、sst4 和 sst5 受体,pIC50 值分别为 8.58、5.41、6.07、5.76 和 6.48。
T2584L1 Octreotide HCl

Octreotide hydrochloride, (-)-,Octreotide hydrochloride

Octreotide HCl is a potent, long-acting synthetic SOMATOSTATIN octapeptide analog that inhibits the secretion of growth hormone.
TP1838 Xenin

Xenin is a 25 amino acid peptide that has been identified in human gastric mucosa in the search for a counterpart to the amphibian octapeptide xenopsin.
T30642 BW 633C

BW 633-C,BW633C BW-633-C,BW633-C,BW-633C

BW 633C is a octapeptide with aminoalcohol (AA) linkage between Leu & Val.
T34273 RC 161

RC-161,RC161

RC 161 is a somatostatin octapeptide analog.
T7497 C3a (70-77)

Complement 3a (70-77),C3a 70-77

Complement System Immunology/Inflammation
C3a (70-77) 是对应于 C3a 的 COOH 末端的八肽。
TP2446 Angiotensin amide

Angiotensinamide,Hypertensine,Angiotensin,NSC 107678,NSC-107678

Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.
T34591 Sdz 204-090

Sdz 204-090 is a cyclic octapeptide analog of somatostatin.
T20403 Dynorphin A (1-8)

PH-8P,Dynorphin (1-8)

Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.
T25087 Angiopeptin

血管抑肽,D-Nal-cys-tyr-trp-lys-val-cys-thr-NH2,Bim 23014 C

Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.
TP2401 Peptide T amide

D-Ala(1)-peptide T amide

Peptide T amide is an octapeptide segment of HIV envelope gp120 and is used in AIDS therapy.
T34867 Thymoctonan

Thymic humoral factor gamma 2

Thymoctonan, as a synthetic octapeptide thymic hormone, can repair immunodeficiency of mice cured of plasmacytoma by melphalan.
TP1785 Peptide T

Peptide T is an octapeptide from the V2 region of HIV-1 gp120. Peptide T is a synthetic octapeptide whose possible mechanism of action is the competitive inhibition of gp120 to the CD4 receptor as well as binding to vasointestinal peptide receptors and in
TP1114 Leucokinin VIII

Leucokinin 8

Leucokinin VIII is an diuretic octapeptide isolated form head extracts of the cockroach.
T15105 Dexloxiglumide

Others Others
Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors.
T76403 [Glp5] Substance P (5-11)

[Glp5] Substance P (5-11)为一八肽,为大鼠中枢神经系统(CNS)主要P物质片段之一,局部调节大鼠纹状体多巴胺释放。
T15711L Larazotide

AT 2347,AT2347,AT-2347

Larazotide is an octapeptide paracellular permeability inhibitor whose structure is derived from a protein (zonula occludens toxin) secreted by Vibrio cholerae for treatment of Coeliac disease.
T82142 Hymenistatin I

Hymenistatin I,一种环八肽[c-(-Pro-Pro-Tyr-Val-Pro-Leu-Ile-ile-Ile-)],具有免疫抑制活性,影响体液和细胞免疫应答。
TP1873 Peptide T TFA

Peptide T (TFA) is an octapeptide derived from the V2 region of HIV-1 gp120. It serves as a ligand for the CD4 receptor, effectively inhibiting the binding of HIV to the CD4 receptor.
TP1482 Xenopsin TFA (51827-01-1 free base)

Xenopsin TFA

Xenopsin TFA is a neurotensin-like octapeptide derived from the skin of xenopus xenopus.Xenopsin TFA is an inhibitor of tetrachloroside to stimulate gastric acid secretion.
T25155 Biphalin

D-ENK,Dala(2),D-Enk-O

Biphalin is a synthetic opioid octapeptide with a palindromic sequence that has high analgesic activity. Biphalin shows a potent affinity for μ and δ-opioid receptors and a significant to κ-receptor.
TP1605 Allatostatin IV

Allatostatin IV, an octapeptide amine, is a member of the allatoregulatory peptide family found in insects which either inhibit (allatostatins) or stimulate (allatotropins) juvenile hormone (JH) synthesis.
T82930 Autoinducing Peptide I

Autoinducing Peptide I为金黄色葡萄球菌分泌的环状八肽,主要用于疫苗研究领域。
T25481 H 77

H77,H-77

H 77 is a new effective renin inhibitor. H 77 is angiotensinogen (6-13)-octapeptide in which the peptide bond -CO-NH- at the Leu(9)-Leu(11) linkage is replaced by a -CH2-NH- bond.
T81585 Oxyntomodulin (human, mouse, rat)

Proglucagon (33-69)

Oxyntomodulin (human, mouse, rat) (Proglucagon (33-69)) 是由胰高血糖素前体产生,融合了完整胰高血糖素序列和C端八肽,含37个氨基酸。
T76618 VPLSLYSG

VPLSLYSG 是一种可被基质金属蛋白酶-9 (MMP-9)、MMP-1和MMP-2降解的八肽。VPLSLYSG 在MMP 底物中有潜在应用。
T75844 BIM-23056 TFA

BIM23056 TFA为线性八肽类化合物,作为sst3与sst5生长抑素受体的有效拮抗剂,其Ki值分别为10.8和5.7。
T75966 C3a (70-77) (TFA)

C3a (70-77) TFA (Complement 3a (70-77) TFA) 为COOH末端对应C3a的八肽,具有C3a的特异性且生物活性约为1至2%。
T80765 Xenopsin TFA

Xenopsin TFA是一种神经降压素样八肽,源自非洲爪蟾皮肤。该化合物能够抑制胃泌素刺激的胃酸分泌。

化合物

Octapeptide-2 Acetate
Cat.No: TP2496
Synonym: Octapeptide-2 Acetate(1374396-34-5 Free base)
Target: Others
Hsp70-derived octapeptide acetate
Cat.No: TP1616L
Synonym: Hsp70-derived octapeptide acetate(736171-62-3 free base)
Target: Others
CCK Octapeptide, non-sulfated acetate
Cat.No: TP2204L
Synonym: CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)
Target: cholecystokinin
Cholecystokinin Octapeptide, desulfated TFA
Cat.No: T39170
Synonym: CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA
Target:
Cholecystokinin Octapeptide, desulfated
Cat.No: TP2204
Synonym: CCK Octapeptide, non-sulfated
Target: Others
Sincalide ammonium
Cat.No: TP1198
Synonym: SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium
Target: cholecystokinin
Sincalide
Cat.No: TP1197
Synonym: SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide
Target: Others
Hsp70-derived octapeptide
Cat.No: TP1616
Synonym:
Target:
Ige octapeptide (497-504)
Cat.No: TP2386
Synonym:
Target:
Laminin B1 octapeptide P-8
Cat.No: TP2389
Synonym: Asp-pro-gln-tyr-ile-gln-ser-arg,Dpgyigsr
Target:
Octapeptide-2
Cat.No: T80204
Synonym:
Target: Reactive Oxygen Species
Xenopsin
Cat.No: T7615
Synonym: 爪蟾肽,Xenopsin(2TFA)
Target: Others
Octreotide Acetate
Cat.No: T4119
Synonym: 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)
Target: Somatostatin
Xenopsin 2TFA(51827-01-1(free base)
Cat.No: T7615L
Synonym:
Target: Others
Leucokinin VIII acetate
Cat.No: TP1114L
Synonym: Leucokinin 8
Target: Others
Peptide T acetate(106362-32-7 free base)
Cat.No: TP1785L
Synonym:
Target: Others, HIV Protease
Neuropeptide FF acetate(99566-27-5 free base)
Cat.No: TP1074L
Synonym: NPFF acetate
Target: Neuropeptide Y Receptor
Allatostatin IV TFA(123338-13-6 free base)
Cat.No: TP1605L1
Synonym:
Target: Others
C3a 70-77 2TFA(63555-63-5(free base))
Cat.No: T7497L
Synonym: Complement 3a (70-77)
Target: Complement System
Angiotensin amide acetate
Cat.No: TP2446L
Synonym: 血管紧张素胺,Angiotensin amide acetate(53-73-6 Free base)
Target: Others
C3a 70-77 acetate
Cat.No: T7497L1
Synonym: C3a 70-77 acetate (63555-63-5 Free base)
Target: Others
CYN 154806 TFA
Cat.No: TP1346
Synonym: CYN 154806 TFA
Target: Somatostatin
Octreotide HCl
Cat.No: T2584L1
Synonym: Octreotide hydrochloride, (-)-,Octreotide hydrochloride
Target:
Xenin
Cat.No: TP1838
Synonym:
Target:
BW 633C
Cat.No: T30642
Synonym: BW 633-C,BW633C BW-633-C,BW633-C,BW-633C
Target:
RC 161
Cat.No: T34273
Synonym: RC-161,RC161
Target:
C3a (70-77)
Cat.No: T7497
Synonym: Complement 3a (70-77),C3a 70-77
Target: Complement System
Angiotensin amide
Cat.No: TP2446
Synonym: Angiotensinamide,Hypertensine,Angiotensin,NSC 107678,NSC-107678
Target:
Sdz 204-090
Cat.No: T34591
Synonym:
Target:
Dynorphin A (1-8)
Cat.No: T20403
Synonym: PH-8P,Dynorphin (1-8)
Target:
Angiopeptin
Cat.No: T25087
Synonym: 血管抑肽,D-Nal-cys-tyr-trp-lys-val-cys-thr-NH2,Bim 23014 C
Target:
Peptide T amide
Cat.No: TP2401
Synonym: D-Ala(1)-peptide T amide
Target:
Thymoctonan
Cat.No: T34867
Synonym: Thymic humoral factor gamma 2
Target:
Peptide T
Cat.No: TP1785
Synonym:
Target:
Leucokinin VIII
Cat.No: TP1114
Synonym: Leucokinin 8
Target:
Dexloxiglumide
Cat.No: T15105
Synonym:
Target: Others
[Glp5] Substance P (5-11)
Cat.No: T76403
Synonym:
Target:
Larazotide
Cat.No: T15711L
Synonym: AT 2347,AT2347,AT-2347
Target:
Hymenistatin I
Cat.No: T82142
Synonym:
Target:
Peptide T TFA
Cat.No: TP1873
Synonym:
Target:
Xenopsin TFA (51827-01-1 free base)
Cat.No: TP1482
Synonym: Xenopsin TFA
Target:
Biphalin
Cat.No: T25155
Synonym: D-ENK,Dala(2),D-Enk-O
Target:
Allatostatin IV
Cat.No: TP1605
Synonym:
Target:
Autoinducing Peptide I
Cat.No: T82930
Synonym:
Target:
H 77
Cat.No: T25481
Synonym: H77,H-77
Target:
Oxyntomodulin (human, mouse, rat)
Cat.No: T81585
Synonym: Proglucagon (33-69)
Target:
VPLSLYSG
Cat.No: T76618
Synonym:
Target:
BIM-23056 TFA
Cat.No: T75844
Synonym:
Target:
C3a (70-77) (TFA)
Cat.No: T75966
Synonym:
Target:
Xenopsin TFA
Cat.No: T80765
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T38649 Lyciumin A

Lyciumin A, a cyclic octapeptide, possesses inhibitory properties against proteases, renin, and angiotensin-converting enzyme. It holds potential for hypertension research.
T79958 Isocrenatoside

Angiotensin-converting Enzyme (ACE) Metabolism
Isocrenatoside (compound 6)为环状八肽,具有ACE抑制活性。该化合物可通过乙醇提取Microtoena prainiana茎部分离纯化。研究显示,1 mg/mL浓度下,Isocrenatoside的ACE抑制效率高达99.3%。
T75646 Moroidin

Moroidin是一种双环八肽,隶属于荨麻疹科环肽科,有效抑制纯化的微管蛋白聚合,表现为微管蛋白聚合抑制剂。此外,Moroidin对包括A549人肺癌细胞在内的多种癌细胞显示出细胞毒性作用,能诱导细胞凋亡。

天然产物

Lyciumin A
Cat.No: T38649
Synonym:
Target:
Isocrenatoside
Cat.No: T79958
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
Moroidin
Cat.No: T75646
Synonym:
Target:
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