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Cat. No. Product Name Target Signaling Pathways
T60509 Maprotiline

Maprotiline 能够抑制细胞的增殖和转移,具有抗癌作用。 Maprotiline 通过靶向 ERK 信号通路和 CRABP1 诱导癌细胞凋亡。 Maprotiline 是一种高度选择性的去甲肾上腺素再摄取阻滞剂,具有有效的抗抑郁作用 [1][2]。
T0172 Maprotiline hydrochloride

Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil

5-HT Receptor; Adrenergic Receptor; AChR; Norepinephrine; Autophagy; Histamine Receptor Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Maprotiline hydrochloride (Psymion) 是一种桥环四环类抗抑郁药,是去甲肾上腺素重吸收抑制剂。
T70960 Maprotiline-d3 hydrochloride

Maprotiline-d3 is intended for use as an internal standard for the quantification of maprotiline by GC- or LC-MS. Maprotiline is a tricyclic antidepressant. It binds to the norepinephrine transporter (NET) and is selective for NET over the serotonin and dopamine transporters. Maprotiline also binds to the serotonin (5-HT) receptor subtype 5-HT2A, as well as histamine H1, muscarinic acetylcholine, α1-adrenergic, and dopamine D2 receptors. In vivo, maprotiline inhibits norepinephrine reuptake in r...
T70958 Dov-Val-Dil-OH TFA

Dov-Val-Dil-OH is a useful chemical intermediate for synthesis of auristatin-related compounds, such as Monomethyl auristatin E (MMAE), Auristatins are antimitotic agents which inhibits cell division by blocking the polymerisation of tubulin.
T24852 Tamitinol

EMD 21 657,Emd21657,Emd 21657,Emd-21657

Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.
T25698 Levoprotiline

Levoprotilinum

Levoprotiline 一种抗抑郁的化合物,它是 Oxaprotiline 的 R-(-)对映体,作用与 Oxaprotiline 相当,并且作用起效潜伏期较短。它是第二代抗抑郁药马普替林的继任者。

化合物

Maprotiline
Cat.No: T60509
Synonym:
Target:
Maprotiline hydrochloride
Cat.No: T0172
Synonym: Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil
Target: 5-HT Receptor, Adrenergic Receptor, AChR, Norepinephrine, Autophagy, Histamine Receptor
Maprotiline-d3 hydrochloride
Cat.No: T70960
Synonym:
Target:
Dov-Val-Dil-OH TFA
Cat.No: T70958
Synonym:
Target:
Tamitinol
Cat.No: T24852
Synonym: EMD 21 657,Emd21657,Emd 21657,Emd-21657
Target:
Levoprotiline
Cat.No: T25698
Synonym: Levoprotilinum
Target:
TargetMol Loading
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