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Cat. No. Product Name Target Signaling Pathways
T2516 Amuvatinib

MP470,HPK 56

Apoptosis; FLT; c-Met/HGFR; c-RET; DNA/RNA Synthesis; PDGFR; c-Kit Angiogenesis; Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Tyrosine Kinase/Adaptors
Amuvatinib (MP470) 是一种多靶点酪氨酸激酶抑制剂,对突变 c-Kit,PDGFRα,Flt3,c-Met 和 c-Ret 具有活性。它还是一种 DNA 修复抑制剂,靶向蛋白 DNA 修复 RAD51,从而破坏 DNA 损伤修复,具有抗肿瘤活性。
T14282 Amuvatinib hydrochloride

HPK 56 hydrochloride,MP470 hydrochloride

Others Others
Amuvatinib hydrochloride (MP470 hydrochloride) is an orally bioavailable multi-targeted tyrosine kinase inhibitor with potent activity against mutant c-Kit, PDGFRα, Flt3, c-Met and c-Ret and is also a DNA repair suppressor through suppression of DNA repai

化合物

Amuvatinib
Cat.No: T2516
Synonym: MP470,HPK 56
Target: Apoptosis, FLT, c-Met/HGFR, c-RET, DNA/RNA Synthesis, PDGFR, c-Kit
Amuvatinib hydrochloride
Cat.No: T14282
Synonym: HPK 56 hydrochloride,MP470 hydrochloride
Target: Others
TargetMol Loading
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