Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0825 |
Ebselen
SPI-1005,PZ-51,依布硒,CCG-39161 |
Phosphatase; Virus Protease; Calcium Channel; COX; HIV Protease | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Ebselen (CCG-39161) 是一种谷胱甘肽过氧化物酶模拟物,是电压依赖性钙通道阻断剂。它抑制Mpro 和COVID-19病毒,是HIV-1衣壳 CTD 二聚化的抑制剂,具有抗炎、抗癌和抗氧化活性。 | |||
T27235 |
Ebselen oxide
|
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Ebselen oxide is a dose-dependent inhibitor of HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, and HDAC9. | |||
T39020 |
Carboxyebselen
Carboxyebselen,HOOC-Ebs |
NOS | Immunology/Inflammation |
Carboxyebselen (HOOC-Ebs) 是一种内皮型一氧化氮合酶 (eNOS) 抑制剂,具有有效性和选择性。 | |||
T33407 |
MitoEbselen-2 chloride
MitoPeroxidase-2,MitoPeroxidase 2,MitoEbselen 2,MitoEbselen-2 |
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MitoEbselen-2 is a radiation mitigator which reduces lipid hydroperoxides and prevents apoptotic cell death. When administered 24 hours postirradiation, MitoEbselen-2 was shown to increase the survival of mice exposed to whole body γ-irradiation. |