Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6484 |
EI1
KB-145943,Ezh2 inhibitor |
Apoptosis; Histone Methyltransferase | Apoptosis; Chromatin/Epigenetic |
EI1 (Ezh2 inhibitor) 是一种EZH2抑制剂,能够作用于 EZH2 (WT) 和 EZH2 (Y641F),IC50值分别为 15 nM 和 13 nM。 | |||
T71871 |
EI-1
|
||
EI-1 is an inhibitor of Hepatitis C virus entry. | |||
T6196 |
PP1
EI 275,AGL 1872 |
Apoptosis; EGFR; Bcr-Abl; Src; c-Kit | Angiogenesis; Apoptosis; Cytoskeletal Signaling; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
PP1 (AGL 1872) 是一种选择性有效 Src 家族抑制剂,抑制 Lck 和Fyn,IC50分别为 5 和 6 nM。 |